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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 17, 2013, Pages 4832-4836

Novel selective inhibitors of aminopeptidases that generate antigenic peptides

(6) Papakyriakou, Athanasios a,b Zervoudi, Efthalia b Theodorakis, Emmanuel A a Saveanu, Loredana c Stratikos, Efstratios b Vourloumis, Dionisios b

a UNIVERSITY OF CALIFORNIA (United States)

b INSTITUTE OF NANOSCIENCE AND NANOTECHNOLOGY (Greece)

c INSERM (France)

Author keywords

Endoplasmic reticulum aminopeptidase; ERAP1; ERAP2; IRAP; Molecular modeling; Rational design; Selective inhibitor

Indexed keywords

AMINOPEPTIDASE;

ANTIGEN PRESENTATION; ARTICLE; COMPETITIVE INHIBITION; ENDOPLASMIC RETICULUM; HUMAN; MOLECULAR DOCKING; NUCLEOPHILICITY; STATIC ELECTRICITY;

ENDOPLASMIC RETICULUM AMINOPEPTIDASE; ERAP1; ERAP2; IRAP; MOLECULAR MODELING; RATIONAL DESIGN; SELECTIVE INHIBITOR;

AMINOPEPTIDASES; CYSTINYL AMINOPEPTIDASE; DRUG DESIGN; ENDOPLASMIC RETICULUM; ENZYME INHIBITORS; HUMANS; MODELS, MOLECULAR;

EID: 84881368000 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.07.024 Document Type: Article

Times cited : (26)

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