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Volumn 8, Issue 8, 2013, Pages 1322-1329

Structure-based design of small-molecule ligands of phosphofructokinase-2 activating or inhibiting glycolysis

(8) Pyrkov, Timothy V a Sevostyanova, Irina A b Schmalhausen, Elena V b Shkoporov, Andrei N c Vinnik, Andrei A a Muronetz, Vladimir I b Severin, Fedor F b Fedichev, Peter O a,d

a Quantum Pharmaceuticals (Russian Federation)

b MOSCOW STATE UNIVERSITY (Russian Federation)

c PIROGOV RUSSIAN NATIONAL RESEARCH MEDICAL UNIVERSITY (Russian Federation)

d MOSCOW INSTITUTE OF PHYSICS AND TECHNOLOGY (Russian Federation)

Author keywords

Cancer; Drug design; Glycolysis; Metabolism; Phosphofructokinases

Indexed keywords

6 PHOSPHOFRUCTO 2 KINASE; FRUCTOSE 2,6 BISPHOSPHATE;

ANTIPROLIFERATIVE ACTIVITY; ARTICLE; BINDING AFFINITY; BREAST CANCER; CELL LYSATE; CELL PROLIFERATION; COLON ADENOCARCINOMA; COMPUTER AIDED DESIGN; GLYCOLYSIS; HUMAN; HUMAN CELL; HYDROGEN BOND; IN VITRO STUDY; LUNG ADENOCARCINOMA; MOLECULAR DOCKING; NONHUMAN; PRIORITY JOURNAL; RAT; STRUCTURE ACTIVITY RELATION;

EID: 84881026405 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201300154 Document Type: Article

Times cited : (9)

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