Identification and characterization of a new chemotype of noncovalent SENP inhibitors

ACS Chemical Biology

Volumn 8, Issue 7, 2013, Pages 1435-1441

  Madu, Ikenna G ^a   Namanja, Andrew T ^a   Su, Yang ^a   Wong, Steven ^a   Li, Yi Jia ^a   Chen, Yuan ^a  

^a CITY OF HOPE NATIONAL MEDICAL CENTER   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ANTINEOPLASTIC AGENT; PROTEINASE INHIBITOR; SMALL UBIQUITIN RELATED MODIFIER PROTEASE INHIBITOR; SUMO 1 PROTEIN; SUMO 2 PROTEIN; SUMO PROTEIN; UNCLASSIFIED DRUG;

ANTINEOPLASTIC ACTIVITY; ARTICLE; CELL CYCLE PROGRESSION; CELL TRANSPORT; CONTROLLED STUDY; DNA DAMAGE; DRUG IDENTIFICATION; DRUG STRUCTURE; ENZYME INHIBITION; ENZYME KINETICS; NUCLEAR MAGNETIC RESONANCE; PRIORITY JOURNAL;

CATALYTIC DOMAIN; ELECTROPHORESIS, POLYACRYLAMIDE GEL; ENDOPEPTIDASES; ENZYME ACTIVATION; ENZYME INHIBITORS; HELA CELLS; HUMANS; INHIBITORY CONCENTRATION 50; MAGNETIC RESONANCE SPECTROSCOPY; MODELS, CHEMICAL; SMALL MOLECULE LIBRARIES;

EID: 84880516465     PISSN: 15548929     EISSN: 15548937     Source Type: Journal    
DOI: 10.1021/cb400177q     Document Type: Article

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