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Volumn 14, Issue 1, 2013, Pages 141-150

Effect of counterions on physicochemical properties of prazosin salts

Author keywords

prazosin; preformulation; salt form; salt screening

Indexed keywords

COUNTERION; PRAZOSIN;

EID: 84878575159     PISSN: None     EISSN: 15309932     Source Type: Journal    
DOI: 10.1208/s12249-012-9889-x     Document Type: Article
Times cited : (11)

References (32)
  • 1
    • 0017623487 scopus 로고
    • Pharmaceutical salts
    • 833720 10.1002/jps.2600660104 1:CAS:528:DyaE2sXmtVCnsw%3D%3D
    • Berge SM, Bighley LM, Monkhouse DC. Pharmaceutical salts. J Pharm Sci. 1977;66:1-19.
    • (1977) J Pharm Sci , vol.66 , pp. 1-19
    • Berge, S.M.1    Bighley, L.M.2    Monkhouse, D.C.3
  • 2
    • 34249088975 scopus 로고    scopus 로고
    • Structure, solubility, screening, and synthesis of molecular salts
    • 17455329 10.1002/jps.20927 1:CAS:528:DC%2BD2sXltVGqs7k%3D
    • Black SN, Collier EA, Davey RJ, Roberts RJ. Structure, solubility, screening, and synthesis of molecular salts. J Pharm Sci. 2007;96:1053-68.
    • (2007) J Pharm Sci , vol.96 , pp. 1053-1068
    • Black, S.N.1    Collier, E.A.2    Davey, R.J.3    Roberts, R.J.4
  • 3
    • 1042284962 scopus 로고    scopus 로고
    • A procedure for salt selection and optimization
    • H. Stahl C.G. Wermuth (eds) Wiley-VCH Inc. Weinheim
    • Bowker MJ. A procedure for salt selection and optimization. In: Stahl PH, Wermuth CG, editors. Handbook of pharmaceutical salts: properties, selection and use. Weinheim: Wiley-VCH Inc.; 2002. p. 161-89.
    • (2002) Handbook of Pharmaceutical Salts: Properties, Selection and Use , pp. 161-189
    • Bowker, M.J.1
  • 4
    • 0035835965 scopus 로고    scopus 로고
    • Changing the salt, changing the drug
    • Davies G. Changing the salt, changing the drug. Pharm J. 2001;266:322-3.
    • (2001) Pharm J , vol.266 , pp. 322-323
    • Davies, G.1
  • 5
    • 0023032232 scopus 로고
    • Salt selection for basic drugs
    • 10.1016/0378-5173(86)90055-4 1:CAS:528:DyaL2sXjvVarsA%3D%3D
    • Gould PL. Salt selection for basic drugs. Int J Pharm. 1986;33:201-17.
    • (1986) Int J Pharm , vol.33 , pp. 201-217
    • Gould, P.L.1
  • 6
    • 34548032742 scopus 로고    scopus 로고
    • Salt formation to improve drug solubility
    • 17619064 10.1016/j.addr.2007.05.010 1:CAS:528:DC%2BD2sXpsFGksrc%3D
    • Serajuddin ATM. Salt formation to improve drug solubility. Adv Drug Deliv Rev. 2007;59:603-16.
    • (2007) Adv Drug Deliv Rev , vol.59 , pp. 603-616
    • Serajuddin, A.T.M.1
  • 7
  • 8
    • 51949100375 scopus 로고    scopus 로고
    • Preparation and characterization of salt forms of enalapril
    • 18720234 10.1080/10837450802244686 1:CAS:528:DC%2BD1cXhtFaisrzE
    • Kumar L, Amin A, Bansal AK. Preparation and characterization of salt forms of enalapril. Pharm Dev Technol. 2008;13:345-57.
    • (2008) Pharm Dev Technol , vol.13 , pp. 345-357
    • Kumar, L.1    Amin, A.2    Bansal, A.K.3
  • 9
    • 0028219710 scopus 로고
    • An integrated approach to the selection of optimal salt form for a new drug candidate
    • 10.1016/0378-5173(94)90104-X 1:CAS:528:DyaK2cXjtlSqurw%3D
    • Morris KR, Fakes MG, Thakur AB, Newman AW, Singh AK, Venit JJ, et al. An integrated approach to the selection of optimal salt form for a new drug candidate. Int J Pharm. 1994;105:209-17.
    • (1994) Int J Pharm , vol.105 , pp. 209-217
    • Morris, K.R.1    Fakes, M.G.2    Thakur, A.B.3    Newman, A.W.4    Singh, A.K.5    Venit, J.J.6
  • 11
    • 80053378054 scopus 로고
    • Adrenergic receptor blocking agents
    • B.G. Katzung (eds) Lange Medical Los Altos
    • Hofmann BB. Adrenergic receptor blocking agents. In: Katzung BG, editor. Basic and clinical pharmacology. Los Altos: Lange Medical; 1984. p. 97-107.
    • (1984) Basic and Clinical Pharmacology , pp. 97-107
    • Hofmann, B.B.1
  • 12
    • 84912073430 scopus 로고
    • Polar and nonpolar interactions in adhesion
    • 10.1080/00218467308078437 1:CAS:528:DyaE3sXhsVyhtbw%3D
    • Wu S. Polar and nonpolar interactions in adhesion. J Adhes. 1973;5:39-55.
    • (1973) J Adhes , vol.5 , pp. 39-55
    • Wu, S.1
  • 14
    • 77956922967 scopus 로고
    • Prazosin hydrochloride
    • Brittain HG, editor Amsterdam: Elsevier
    • Kostek LJ. Prazosin hydrochloride. In: Brittain HG, editor. Analytical profile of drug substances and excipients, vol. 18. Amsterdam: Elsevier; 1989. p. 351-81.
    • (1989) Analytical Profile of Drug Substances and Excipients , vol.18 , pp. 351-381
    • Kostek, L.J.1
  • 15
    • 0036179239 scopus 로고    scopus 로고
    • Experimental and computational screening models for prediction of aqueous drug solubility
    • 11885560 10.1023/A:1014224900524
    • Bergström CAS, Norinder U, Luthman K, Artursson P. Experimental and computational screening models for prediction of aqueous drug solubility. Pharm Res. 2002;19:182-8.
    • (2002) Pharm Res , vol.19 , pp. 182-188
    • Bergström, C.A.S.1    Norinder, U.2    Luthman, K.3    Artursson, P.4
  • 17
    • 84878546315 scopus 로고    scopus 로고
    • Accessed 1 May 2012
    • Prazosin permeability. http://www.cyprotex.com/cloescreen/in-vitro- permeability/mdr1-mdck-permeability/. Accessed 1 May 2012.
    • Prazosin Permeability
  • 19
    • 80053345313 scopus 로고    scopus 로고
    • Effect of humidity on the hydration behaviour of prazosin hydrochloride polyhydrate: Thermal, sorption and crystallographic study
    • 10.1016/j.tca.2011.08.006
    • Kumar L, Bansal AK. Effect of humidity on the hydration behaviour of prazosin hydrochloride polyhydrate: thermal, sorption and crystallographic study. Thermochim Acta. 2012;525:206-10.
    • (2012) Thermochim Acta , vol.525 , pp. 206-210
    • Kumar, L.1    Bansal, A.K.2
  • 20
  • 23
    • 0019992394 scopus 로고
    • Common ion equilibria of hydrochloride salts and the Setschenow equation
    • 7097509 10.1002/jps.2600710527 1:CAS:528:DyaL38Xit1eit7k%3D
    • Bogardus JB. Common ion equilibria of hydrochloride salts and the Setschenow equation. J Pharm Sci. 1982;71:588-90.
    • (1982) J Pharm Sci , vol.71 , pp. 588-590
    • Bogardus, J.B.1
  • 24
    • 0034607382 scopus 로고    scopus 로고
    • Salt form selection and characterization of LY333531 mesylate monohydrate
    • 10767572 10.1016/S0378-5173(00)00350-1 1:CAS:528:DC%2BD3cXitlelu7w%3D
    • Engel GL, Farid NA, Faul MM, Richardson LA, Winneroski LL. Salt form selection and characterization of LY333531 mesylate monohydrate. Int J Pharm. 2000;198:239-47.
    • (2000) Int J Pharm , vol.198 , pp. 239-247
    • Engel, G.L.1    Farid, N.A.2    Faul, M.M.3    Richardson, L.A.4    Winneroski, L.L.5
  • 25
    • 0019513805 scopus 로고
    • Precaution on use of hydrochloride salts in pharmaceutical formulation
    • 7252797 10.1002/jps.2600700604 1:CAS:528:DyaL3MXksV2gs7w%3D
    • Miyazaki S, Oshiba M, Nadai T. Precaution on use of hydrochloride salts in pharmaceutical formulation. J Pharm Sci. 1981;70:594-6.
    • (1981) J Pharm Sci , vol.70 , pp. 594-596
    • Miyazaki, S.1    Oshiba, M.2    Nadai, T.3
  • 26
    • 84873525097 scopus 로고    scopus 로고
    • Preparation of water-soluble compounds through salt formation
    • C.G. Wermuth (eds) Academic London
    • Bowker MJ, Stahl PH. Preparation of water-soluble compounds through salt formation. In: Wermuth CG, editor. The practice of medicinal chemistry. London: Academic; 2008. p. 749-66.
    • (2008) The Practice of Medicinal Chemistry , pp. 749-766
    • Bowker, M.J.1    Stahl, P.H.2
  • 27
    • 0017158036 scopus 로고
    • Enhancement of solubility of drug salts by hydrophilic counterions: Properties of organic salts of an antimalarial drug
    • 932950 10.1002/jps.2600650533 1:CAS:528:DyaE28Xkt1Ggsbo%3D
    • Agharkar S, Lindenbaum S, Higuchi T. Enhancement of solubility of drug salts by hydrophilic counterions: properties of organic salts of an antimalarial drug. J Pharm Sci. 1976;65:747-9.
    • (1976) J Pharm Sci , vol.65 , pp. 747-749
    • Agharkar, S.1    Lindenbaum, S.2    Higuchi, T.3
  • 28
    • 0023253722 scopus 로고
    • Preformulation salt selection - Physical property comparison of the tris(hydroxymethyl)aminomethane salts of four analgesic/antiinflammatory agents with the sodium salts and the free acids
    • 3509292 10.1023/A:1016420514689 1:CAS:528:DyaL2sXls1Wmsrw%3D
    • Gu L, Strickley RL. Preformulation salt selection - physical property comparison of the tris(hydroxymethyl)aminomethane salts of four analgesic/antiinflammatory agents with the sodium salts and the free acids. Pharm Res. 1987;4:255-7.
    • (1987) Pharm Res , vol.4 , pp. 255-257
    • Gu, L.1    Strickley, R.L.2
  • 29
    • 0021876419 scopus 로고
    • Predictive relationships in the water solubility of salts of a nonsteroidal anti-inflammatory drug
    • 4032262 10.1002/jps.2600740803 1:CAS:528:DyaL2MXlt1yqtr0%3D
    • Anderson BD, Conradi RA. Predictive relationships in the water solubility of salts of a nonsteroidal anti-inflammatory drug. J Pharm Sci. 1985;74:815-20.
    • (1985) J Pharm Sci , vol.74 , pp. 815-820
    • Anderson, B.D.1    Conradi, R.A.2
  • 30
    • 0018145767 scopus 로고
    • PH-solubility profiles of organic carboxylic acids and their salts
    • 29115 10.1002/jps.2600670918 1:CAS:528:DyaE1cXlvVGqu78%3D
    • Chowhan JT. pH-solubility profiles of organic carboxylic acids and their salts. J Pharm Sci. 1978;67:1257-60.
    • (1978) J Pharm Sci , vol.67 , pp. 1257-1260
    • Chowhan, J.T.1
  • 31
    • 78649903986 scopus 로고    scopus 로고
    • Analysis of relationships between solid-state properties, counterion, and developability of pharmaceutical salts
    • 20680707 10.1208/s12249-010-9499-4 1:CAS:528:DC%2BC3cXhsFemsLfJ
    • Guerrieri P, Rumondor ACF, Li T, Taylor LS. Analysis of relationships between solid-state properties, counterion, and developability of pharmaceutical salts. AAPS PharmSciTech. 2010;11:1212-22.
    • (2010) AAPS PharmSciTech , vol.11 , pp. 1212-1222
    • Guerrieri, P.1    Rumondor, A.C.F.2    Li, T.3    Taylor, L.S.4
  • 32
    • 0024949425 scopus 로고
    • Solubility and solid state properties of the sodium salts of drugs
    • 2760824 10.1002/jps.2600780614 1:CAS:528:DyaL1MXlt1Sksrc%3D
    • Rubino JT. Solubility and solid state properties of the sodium salts of drugs. J Pharm Sci. 1989;78:485-9.
    • (1989) J Pharm Sci , vol.78 , pp. 485-489
    • Rubino, J.T.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.