Effect of humidity on the hydration behaviour of prazosin hydrochloride polyhydrate: Thermal, sorption and crystallographic study

Thermochimica Acta

Volumn 525, Issue 1-2, 2011, Pages 206-210

  Kumar, Lokesh ^a   Bansal, Arvind K ^a  

^a NATIONAL INSTITUTE OF PHARMACEUTICAL EDUCATION AND RESEARCH NIPER   (India)

Author keywords

Dynamic vapour sorption; Polyhydrate; Powder X ray diffraction; Prazosin

Indexed keywords

AMBIENT CONDITIONS; CRYSTALLOGRAPHIC DATA; CRYSTALLOGRAPHIC STUDIES; DIFFRACTION PEAKS; DIHYDRATES; INTERSTITIAL WATER; LATTICE WATER; POLYHYDRATE; POWDER X-RAY DIFFRACTION; PRAZOSIN; SINGLE-STEP; SORPTION ISOTHERMS; WATER LOSS;

BEHAVIORAL RESEARCH; DIFFERENTIAL SCANNING CALORIMETRY; DIFFRACTION; HEATING; HEATING RATE; HYDRATES; HYDRATION; SORPTION; X RAY DIFFRACTION; X RAY DIFFRACTION ANALYSIS;

THERMOGRAVIMETRIC ANALYSIS;

EID: 80053345313     PISSN: 00406031     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tca.2011.08.006     Document Type: Article

References (22)

1. U.J. Griesser The importance of solvates R. Hilfiker, Polymorphism in the Pharmaceutical Industry 2006 Wiley-VCH Verlag GmbH Weinheim 211 257
2. K.R. Morris, and N. Rodriguez-Hornedo Hydrates J. Swarbrick, J.C. Boylan, Encyclopedia of Pharmaceutical Technology vol. 7 1993 Marcel Dekker Inc. New York, NY 393 440
3. L.R. Chen Solid state behaviour of cromolyn sodium hydrates J. Pharm. Sci. 88 1999 1191 1200 (Pubitemid 29526306)
4. K. Kawakami Effect of salt type on hygroscopicity of a new cephalosporin Pharm. Res. 22 2005 1365 1373 (Pubitemid 41176041)
5. F.G. Vogt, P.C. Dell'Orco, A.M. Diederich, Q. Su, J.L. Wood, G.E. Zuber, L.M. Katrincic, R.L. Mueller, D.J. Busby, and C.W. DeBrosse A study of variable hydration states in topotecan hydrochloride J. Pharmaceut. Biomed. Anal. 40 2006 1080 1088 (Pubitemid 43247444)
6. B.B. Hofmann Adrenergic receptor blocking agents B.G. Katzung, Basic and Clinical Pharmacology 1984 Lange Medical Publications Los Altos 97 107
7. L.J. Kostek Prazosin hydrochloride H.G. Brittain, Analytical Profile of Drug Substances and Excipients vol. 18 1989 Elsevier, Inc. 351 381
8. J. Vincent, P.A. Meredith, J.L. Reid, H.L. Elliot, and P.C. Rubin Clinical pharmacokinetics of prazosin Clin. Pharmacokin. 10 1985 144 154
9. R.F. Westermen, J.A. Schouten, and W.A. Hengeveld Prazosin once or twice daily? Eur. J. Clin. Pharmacol. 28 1985 11 15 (Pubitemid 15126521)
10. E.J. Bianco, Novel crystalline forms of prazosin hydrochloride, US Patent, US4092315, 1978.
11. V.V. Chernyshev, P.W. Stephens, A.V. Yatsenko, O.B. Ryabova, and V.A. Makarov Structural characterization of prazosin hydrochloride and prazosin free base J. Pharm. Sci. 93 2004 3090 3095 (Pubitemid 39657812)
12. S.O.E. Lindholm, A process for the preparation of anhydrous, stable, crystalline delta-form of prazosin hydrochloride, US Patent, US4873330, 1989.
13. Y. Niimoto, S. Yoshida, Preparation of prazosin hydrochloride anhydrous epsilon-type crystals, JP Patent, JP03206088, 1991.
14. R. Roteman, 1-(4-Amino-6,7-dimethoxy-2-quinazolinyl)-4-(2- tetrahydrofuroyl)piperazine hydrochloride dihydrate, US Patent, US4251532, 1981.
15. H. Schickaneder, I. Grafe, K.H. Ahrens, Crystalline anhydrous sigma form of 2-(4-(2-furoyl)-(2-piperazin)-1-yl)-4-amino-6,7-dimethoxy-quinazoline hydrochloride and a process for its preparation, US Patent, US4816455, 1989.
16. F.G. Vogt, P.C. Dell'Orco, A.M. Diederich, Q. Su, J.L. Wood, G.E. Zuber, L.M. Katrincic, R.L. Mueller, D.J. Busby, and C.W. DeBrosse A study of variable hydration states in topotecan hydrochloride J. Pharm. Biomed. Anal. 40 2006 1080 1088 (Pubitemid 43247444)
17. K.R. Morris Structural aspects of hydrates and solvates H.G. Brittain, Polymorphism in Pharmaceutical Solids 1999 Marcel Dekker Inc. New York, NY 125 182
18. K.R. Morris, A.W. Newman, D.E. Bugay, S.A. Ranadive, A.K. Singh, M. Szyper, S.A. Varia, H.G. Brittain, and A.T.M. Serajuddin Characterization of humidity dependent changes in crystal properties of a new HMG-CoA reductase inhibitor in support of its dosage form development Int. J. Pharm. 108 1994 195 206 (Pubitemid 24223174)
19. J. Baronsky, S. Bongaerts, M. Traeubel, H.-C. Weiss, and N. Urbanetz The study of different solid forms of Emodepside Eur. J. Pharm. Biopharm. 71 2009 88 99
20. J.S.G. Cox, G.D. Woodard, and W.C. McCrone Solid-state chemistry of cromolyn sodium (disodium cromoglycate) J. Pharm. Sci. 60 1971 1458 1465
21. J.R. Authelin Thermodynamics of non-stoichiometric pharmaceutical hydrates Int. J. Pharm. 303 2005 37 53
22. F.G. Vogt, J. Brum, L.M. Katrincic, A. Flanch, and J.M. Socha Physical, crystallographic, and spectroscopic characterization of a crystalline pharmaceutical hydrate: understanding the role of water Cryst. Growth Des. 6 2006 2333 2354 (Pubitemid 44629543)