메뉴 건너뛰기




Volumn 18, Issue 4, 2013, Pages 834-843

Preparation and characterization of microemulsion formulations of nicotinic acid and its prodrugs for transdermal delivery

Author keywords

Dodecyl nicotinate; Microemulsion; Myristyl nicotinate; Nicotinic acid; Transdermal delivery

Indexed keywords

DODECYL NICOTINATE; LABRASOL; MYRISTIC ACID ISOPROPYL ESTER; MYRISTYL NICOTINATE; NICOTINIC ACID; NICOTINIC ACID DERIVATIVE; PRODRUG; UNCLASSIFIED DRUG;

EID: 84877850297     PISSN: 10837450     EISSN: 10979867     Source Type: Journal    
DOI: 10.3109/10837450.2012.727003     Document Type: Article
Times cited : (21)

References (42)
  • 2
    • 0025804094 scopus 로고
    • Structuremetabolism relationships in the hydrolysis of nicotinate esters by rat liver and brain subcellular fractions
    • Durrer A, Walther B, Racciatti A, Boss G, Testa B. Structuremetabolism relationships in the hydrolysis of nicotinate esters by rat liver and brain subcellular fractions. Pharm Res 1991;8:832-839.
    • (1991) Pharm Res , vol.8 , pp. 832-839
    • Durrer, A.1    Walther, B.2    Racciatti, A.3    Boss, G.4    Testa, B.5
  • 3
    • 0019474574 scopus 로고
    • Influence of nicotinic acid on metabolism of cholesterol and triglycerides in man
    • Grundy SM, Mok HY, Zech L, Berman M. Influence of nicotinic acid on metabolism of cholesterol and triglycerides in man. J Lipid Res 1981;22:24-36.
    • (1981) J Lipid Res , vol.22 , pp. 24-36
    • Grundy, S.M.1    Mok, H.Y.2    Zech, L.3    Berman, M.4
  • 5
    • 0037352280 scopus 로고    scopus 로고
    • PUMA-G and HM74 are receptors for nicotinic acid and mediate its anti-lipolytic effect
    • Tunaru S, Kero J, Schaub A, Wufka C, Blaukat A, Pfeffer K et al. PUMA-G and HM74 are receptors for nicotinic acid and mediate its anti-lipolytic effect. Nat Med 2003;9:352-355.
    • (2003) Nat Med , vol.9 , pp. 352-355
    • Tunaru, S.1    Kero, J.2    Schaub, A.3    Wufka, C.4    Blaukat, A.5    Pfeffer, K.6
  • 7
    • 67649372666 scopus 로고    scopus 로고
    • Flushing profile of extended-release niacin/laropiprant versus gradually titrated niacin extendedrelease in patients with dyslipidemia with and without ischemic cardiovascular disease
    • Maccubbin D, Koren MJ, Davidson M, Gavish D, Pasternak RC, Macdonell G et al. Flushing profile of extended-release niacin/laropiprant versus gradually titrated niacin extendedrelease in patients with dyslipidemia with and without ischemic cardiovascular disease. Am J Cardiol 2009;104:74-81.
    • (2009) Am J Cardiol , vol.104 , pp. 74-81
    • Maccubbin, D.1    Koren, M.J.2    Davidson, M.3    Gavish, D.4    Pasternak, R.C.5    Macdonell, G.6
  • 9
    • 84877853963 scopus 로고    scopus 로고
    • Opinion of the Scientific Committee on Food on the Tolerable Upper Intake Levels of Nicotinic Acid and Nicotinamide (Niacin)
    • Opinion of the Scientific Committee on Food on the Tolerable Upper Intake Levels of Nicotinic Acid and Nicotinamide (Niacin). Scientific committee on food SCF/CS/NUT/UPPLEV/39 Final. 2002:1-20.
    • (2002) Scientific Committee on Food SCF/CS/NUT/UPPLEV/39 Final , pp. 1-20
  • 10
    • 0035213058 scopus 로고    scopus 로고
    • Cholesterol and glycemic effects of Niaspan in patients with type 2 diabetes
    • Kane MP, Hamilton RA, Addesse E, Busch RS, Bakst G. Cholesterol and glycemic effects of Niaspan in patients with type 2 diabetes. Pharmacotherapy 2001;21:1473-1478.
    • (2001) Pharmacotherapy , vol.21 , pp. 1473-1478
    • Kane, M.P.1    Hamilton, R.A.2    Addesse, E.3    Busch, R.S.4    Bakst, G.5
  • 11
    • 0642344305 scopus 로고    scopus 로고
    • Overview of niacin formulations: Differences in pharmacokinetics, efficacy, and safety
    • quiz S25
    • Pieper JA. Overview of niacin formulations: Differences in pharmacokinetics, efficacy, and safety. Am J Health Syst Pharm 2003;60:S9-14; quiz S25.
    • (2003) Am J Health Syst Pharm , vol.60
    • Pieper, J.A.1
  • 12
    • 0036737714 scopus 로고    scopus 로고
    • Understanding niacin formulations
    • Pieper JA. Understanding niacin formulations. Am J Manag Care 2002;8:S308-S314.
    • (2002) Am J Manag Care , vol.8
    • Pieper, J.A.1
  • 13
    • 84877862808 scopus 로고    scopus 로고
    • National Drugs Poisons Schedule Committee June
    • National Drugs and Poisons Schedule Committee. Record of Reasons of Meeting 53. June 2008;206-207.
    • (2008) Record of Reasons of Meeting 53 , pp. 206-207
  • 14
    • 84877853229 scopus 로고    scopus 로고
    • University of Arizona: Southwest Environmental Health Sciences Center Accessed on: March 2010
    • University of Arizona: Southwest Environmental Health Sciences Center. Available at: http://swehsc.pharmacy.arizona.edu. Accessed on: March 2010.
  • 15
    • 0018621689 scopus 로고
    • Clinical pharmacology and pharmacokinetics of nicotinic acid
    • Weiner M. Clinical pharmacology and pharmacokinetics of nicotinic acid. Drug Metab Rev 1979;9:99-106.
    • (1979) Drug Metab Rev , vol.9 , pp. 99-106
    • Weiner, M.1
  • 16
    • 84890000723 scopus 로고    scopus 로고
    • Developing topical prodrugs for skin cancer prevention
    • Alberts DS, Hess LM, eds. Verlag Berlin Heidelberg: Springer
    • Jacobson EL, Kim H, Kim M, Wondrak GT, Jacobson MK. (2008). Developing topical prodrugs for skin cancer prevention. In: Alberts DS, Hess LM, eds. Fundamentals of Cancer Prevention. Verlag Berlin Heidelberg: Springer, 215-237.
    • (2008) Fundamentals of Cancer Prevention , pp. 215-237
    • Jacobson, E.L.1    Kim, H.2    Kim, M.3    Wondrak, G.T.4    Jacobson, M.K.5
  • 17
    • 28844436909 scopus 로고    scopus 로고
    • Simultaneous determination of myristyl nicotinate, nicotinic acid, and nicotinamide in rabbit plasma by liquid chromatographytandem mass spectrometry using methyl ethyl ketone as a deproteinization solvent
    • Catz P, Shinn W, Kapetanovic IM, Kim H, Kim M, Jacobson EL et al. Simultaneous determination of myristyl nicotinate, nicotinic acid, and nicotinamide in rabbit plasma by liquid chromatographytandem mass spectrometry using methyl ethyl ketone as a deproteinization solvent. J Chromatogr B Analyt Technol Biomed Life Sci 2005;829:123-135.
    • (2005) J Chromatogr B Analyt Technol Biomed Life Sci , vol.829 , pp. 123-135
    • Catz, P.1    Shinn, W.2    Kapetanovic, I.M.3    Kim, H.4    Kim, M.5    Jacobson, E.L.6
  • 19
    • 33750507126 scopus 로고    scopus 로고
    • Microemulsions as transdermal drug delivery vehicles
    • Kogan A, Garti N. Microemulsions as transdermal drug delivery vehicles. Adv Colloid Interface Sci 2006;123-126:369-385.
    • (2006) Adv Colloid Interface Sci , vol.123-126 , pp. 369-385
    • Kogan, A.1    Garti, N.2
  • 20
    • 36249019156 scopus 로고    scopus 로고
    • Role of novel delivery systems in developing topical antioxidants as therapeutics to combat photoageing
    • Kaur IP, Kapila M, Agrawal R. Role of novel delivery systems in developing topical antioxidants as therapeutics to combat photoageing. Ageing Res Rev 2007;6:271-288.
    • (2007) Ageing Res Rev , vol.6 , pp. 271-288
    • Kaur, I.P.1    Kapila, M.2    Agrawal, R.3
  • 21
    • 39749176475 scopus 로고    scopus 로고
    • Microemulsions-modern colloidal carrier for dermal and transdermal drug delivery
    • Heuschkel S, Goebel A, Neubert RH. Microemulsions-modern colloidal carrier for dermal and transdermal drug delivery. J Pharm Sci 2008;97:603-631.
    • (2008) J Pharm Sci , vol.97 , pp. 603-631
    • Heuschkel, S.1    Goebel, A.2    Neubert, R.H.3
  • 22
    • 80155173443 scopus 로고    scopus 로고
    • Microemulsions in topical drug delivery
    • Smith EW, Maibach HI, eds. 2nd edition. Boca Raton: CRC Press, Taylor & Francis Group
    • Pappinen S, Urtti A. (2006). Microemulsions in topical drug delivery. In: Smith EW, Maibach HI, eds. Percutaneous Penetration Enhancers. 2nd edition. Boca Raton: CRC Press, Taylor & Francis Group, 109-116.
    • (2006) Percutaneous Penetration Enhancers , pp. 109-116
    • Pappinen, S.1    Urtti, A.2
  • 23
    • 18844450421 scopus 로고    scopus 로고
    • In vitro release of diclofenac diethylamine from caprylocaproyl macrogolglycerides based microemulsions
    • Djordjevic L, Primorac M, Stupar M. In vitro release of diclofenac diethylamine from caprylocaproyl macrogolglycerides based microemulsions. Int J Pharm 2005;296:73-79.
    • (2005) Int J Pharm , vol.296 , pp. 73-79
    • Djordjevic, L.1    Primorac, M.2    Stupar, M.3
  • 26
    • 0036851496 scopus 로고    scopus 로고
    • Influence of microemulsions on cutaneous drug delivery
    • Kreilgaard M. Influence of microemulsions on cutaneous drug delivery. Adv Drug Deliv Rev 2002;54 Suppl 1:S77-S98.
    • (2002) Adv Drug Deliv Rev , vol.54 , Issue.SUPPL. 1
    • Kreilgaard, M.1
  • 27
    • 39649112861 scopus 로고    scopus 로고
    • The influence of cosurfactants and oils on the formation of pharmaceutical microemulsions based on PEG-8 caprylic/capric glycerides
    • Djekic L, Primorac M. The influence of cosurfactants and oils on the formation of pharmaceutical microemulsions based on PEG-8 caprylic/capric glycerides. Int J Pharm 2008;352:231-239.
    • (2008) Int J Pharm , vol.352 , pp. 231-239
    • Djekic, L.1    Primorac, M.2
  • 28
    • 0347385190 scopus 로고    scopus 로고
    • Dermatological formulation and transdermal systems
    • Walters KA, ed. New York: Marcel Dekker Inc
    • Walters KA, Brain KR. (2002). Dermatological formulation and transdermal systems. In: Walters KA, ed. Dermatological and Transdermal Formulations. New York: Marcel Dekker Inc, 349-432.
    • (2002) Dermatological and Transdermal Formulations , pp. 349-432
    • Walters, K.A.1    Brain, K.R.2
  • 29
    • 35348882182 scopus 로고    scopus 로고
    • Comparison of stratum corneum penetration and localization of a lipophilic model drug applied in an o/w microemulsion and an amphiphilic cream
    • Teichmann A, Heuschkel S, Jacobi U, Presse G, Neubert RH, Sterry W et al. Comparison of stratum corneum penetration and localization of a lipophilic model drug applied in an o/w microemulsion and an amphiphilic cream. Eur J Pharm Biopharm 2007;67:699-706.
    • (2007) Eur J Pharm Biopharm , vol.67 , pp. 699-706
    • Teichmann, A.1    Heuschkel, S.2    Jacobi, U.3    Presse, G.4    Neubert, R.H.5    Sterry, W.6
  • 30
    • 33747334666 scopus 로고    scopus 로고
    • Investigation of microemulsion system for transdermal delivery of meloxicam
    • Yuan Y, Li SM, Mo FK, Zhong DF. Investigation of microemulsion system for transdermal delivery of meloxicam. Int J Pharm 2006;321:117-123.
    • (2006) Int J Pharm , vol.321 , pp. 117-123
    • Yuan, Y.1    Li, S.M.2    Mo, F.K.3    Zhong, D.F.4
  • 31
    • 28544451387 scopus 로고    scopus 로고
    • Formulation and physicochemical characterization of microemulsion system using isopropyl myristate, medium-chain glyceride, polysorbate 80 and water
    • Subramanian N, Ghosal SK, Acharya A, Moulik SP. Formulation and physicochemical characterization of microemulsion system using isopropyl myristate, medium-chain glyceride, polysorbate 80 and water. Chem Pharm Bull 2005;53:1530-1535.
    • (2005) Chem Pharm Bull , vol.53 , pp. 1530-1535
    • Subramanian, N.1    Ghosal, S.K.2    Acharya, A.3    Moulik, S.P.4
  • 32
    • 48149109605 scopus 로고    scopus 로고
    • A study of the properties of mixed nonionic surfactants microemulsions by NMR, SAXS, viscosity and conductivity
    • Fanun M. A study of the properties of mixed nonionic surfactants microemulsions by NMR, SAXS, viscosity and conductivity. J Mol Liq 2008;142:103-110.
    • (2008) J Mol Liq , vol.142 , pp. 103-110
    • Fanun, M.1
  • 33
    • 15044355680 scopus 로고    scopus 로고
    • Ketorolac amide prodrugs for transdermal delivery: Stability and in vitro rat skin permeation studies
    • Kim BY, Doh HJ, Le TN, Cho WJ, Yong CS, Choi HG et al. Ketorolac amide prodrugs for transdermal delivery: Stability and in vitro rat skin permeation studies. Int J Pharm 2005;293:193-202.
    • (2005) Int J Pharm , vol.293 , pp. 193-202
    • Kim, B.Y.1    Doh, H.J.2    Le, T.N.3    Cho, W.J.4    Yong, C.S.5    Choi, H.G.6
  • 34
    • 0141447812 scopus 로고    scopus 로고
    • Permeation, metabolism and site of action concentration of nicotinic acid derivatives in human skin. Correlation with topical pharmacological effect
    • Muller B, Kasper M, Surber C, Imanidis G. Permeation, metabolism and site of action concentration of nicotinic acid derivatives in human skin. Correlation with topical pharmacological effect. Eur J Pharm Sci 2003;20:181-195.
    • (2003) Eur J Pharm Sci , vol.20 , pp. 181-195
    • Muller, B.1    Kasper, M.2    Surber, C.3    Imanidis, G.4
  • 35
    • 16244376796 scopus 로고    scopus 로고
    • Characterisation of the water-isopropyl myristate system
    • Abraham MH, Acree WE Jr. Characterisation of the water-isopropyl myristate system. Int J Pharm 2005;294:121-128.
    • (2005) Int J Pharm , vol.294 , pp. 121-128
    • Abraham, M.H.1    Acree Jr., W.E.2
  • 37
    • 0033752983 scopus 로고    scopus 로고
    • Permeation enhancers for transdermal drug delivery
    • Sinha VR, Kaur MP. Permeation enhancers for transdermal drug delivery. Drug Dev Ind Pharm 2000;26:1131-1140.
    • (2000) Drug Dev Ind Pharm , vol.26 , pp. 1131-1140
    • Sinha, V.R.1    Kaur, M.P.2
  • 38
    • 69249084491 scopus 로고    scopus 로고
    • Chemical penetration enhancers for transdermal drug delivery systems
    • Pathan IB, Setty CM. Chemical penetration enhancers for transdermal drug delivery systems. Trop J Pharmaceut Res 2009;8:173-179.
    • (2009) Trop J Pharmaceut Res , vol.8 , pp. 173-179
    • Pathan, I.B.1    Setty, C.M.2
  • 42
    • 0036001399 scopus 로고    scopus 로고
    • Transdermal delivery of highly lipophilic drugs. in vitro fluxes of antiestrogens, permeation enhancers, and solvents from liquid formulations
    • Funke AP, Schiller R, Motzkus HW, Gunther C, Muller RH, Lipp R. Transdermal delivery of highly lipophilic drugs: In vitro fluxes of antiestrogens, permeation enhancers, and solvents from liquid formulations. Pharm Res 2002;19:661-668.
    • (2002) Pharm Res , vol.19 , pp. 661-668
    • Funke, A.P.1    Schiller, R.2    Motzkus, H.W.3    Gunther, C.4    Muller, R.H.5    Lipp, R.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.