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Volumn 8, Issue 5, 2013, Pages

Identification of Adiponectin Receptor Agonist Utilizing a Fluorescence Polarization Based High Throughput Assay

Author keywords

[No Author keywords available]

Indexed keywords

ADIPONECTIN RECEPTOR; ADIPONECTIN RECEPTOR 1 AGONIST; ADIPONECTIN RECEPTOR 2 AGONIST; ADIPONECTIN RECEPTOR AGONIST; ARCTIGENIN; ARCTIIN; DEOXYSCHIZANDRIN; GRAMINE; HORMONE RECEPTOR STIMULATING AGENT; LIGAND; MATAIRESINOL; PARTHENOLIDE; SYRINGIN; TAXIFOLIOL; UNCLASSIFIED DRUG;

EID: 84877771919     PISSN: None     EISSN: 19326203     Source Type: Journal    
DOI: 10.1371/journal.pone.0063354     Document Type: Article
Times cited : (51)

References (38)
  • 3
    • 9444285912 scopus 로고    scopus 로고
    • Induction of adiponectin in skeletal muscle by inflammatory cytokines: in vivo and in vitro studies
    • Delaigle AM, Jonas JC, Bauche IB, Cornu O, Brichard SM, (2004) Induction of adiponectin in skeletal muscle by inflammatory cytokines: in vivo and in vitro studies. Endocrinology 145: 5589-5597.
    • (2004) Endocrinology , vol.145 , pp. 5589-5597
    • Delaigle, A.M.1    Jonas, J.C.2    Bauche, I.B.3    Cornu, O.4    Brichard, S.M.5
  • 4
    • 10844220730 scopus 로고    scopus 로고
    • Adiponectin and its receptors in non-alcoholic steatohepatitis
    • Kaser S, Moschen A, Cayon A, Kaser A, Crespo J, et al. (2005) Adiponectin and its receptors in non-alcoholic steatohepatitis. Gut 54: 117-121.
    • (2005) Gut , vol.54 , pp. 117-121
    • Kaser, S.1    Moschen, A.2    Cayon, A.3    Kaser, A.4    Crespo, J.5
  • 5
    • 33847065560 scopus 로고    scopus 로고
    • Adiponectin deficiency protects mice from chemically induced colonic inflammation
    • Fayad R, Pini M, Sennello JA, Cabay RJ, Chan L, et al. (2007) Adiponectin deficiency protects mice from chemically induced colonic inflammation. Gastroenterology 132: 601-614.
    • (2007) Gastroenterology , vol.132 , pp. 601-614
    • Fayad, R.1    Pini, M.2    Sennello, J.A.3    Cabay, R.J.4    Chan, L.5
  • 6
    • 24944532986 scopus 로고    scopus 로고
    • Adiponectin is synthesized and secreted by human and murine cardiomyocytes
    • Pineiro R, Iglesias MJ, Gallego R, Raghay K, Eiras S, et al. (2005) Adiponectin is synthesized and secreted by human and murine cardiomyocytes. FEBS Lett 579: 5163-5169.
    • (2005) FEBS Lett , vol.579 , pp. 5163-5169
    • Pineiro, R.1    Iglesias, M.J.2    Gallego, R.3    Raghay, K.4    Eiras, S.5
  • 7
    • 33745895901 scopus 로고    scopus 로고
    • Salivary gland epithelial cells: a new source of the immunoregulatory hormone adiponectin
    • Katsiougiannis S, Kapsogeorgou EK, Manoussakis MN, Skopouli FN, (2006) Salivary gland epithelial cells: a new source of the immunoregulatory hormone adiponectin. Arthritis Rheum 54: 2295-2299.
    • (2006) Arthritis Rheum , vol.54 , pp. 2295-2299
    • Katsiougiannis, S.1    Kapsogeorgou, E.K.2    Manoussakis, M.N.3    Skopouli, F.N.4
  • 9
    • 18844432308 scopus 로고    scopus 로고
    • Adiponectin and adiponectin receptors
    • Kadowaki T, Yamauchi T, (2005) Adiponectin and adiponectin receptors. Endocr Rev 26: 439-451.
    • (2005) Endocr Rev , vol.26 , pp. 439-451
    • Kadowaki, T.1    Yamauchi, T.2
  • 10
    • 33847733103 scopus 로고    scopus 로고
    • Targeted disruption of AdipoR1 and AdipoR2 causes abrogation of adiponectin binding and metabolic actions
    • Yamauchi T, Nio Y, Maki T, Kobayashi M, Takazawa T, et al. (2007) Targeted disruption of AdipoR1 and AdipoR2 causes abrogation of adiponectin binding and metabolic actions. Nat Med 13: 332-339.
    • (2007) Nat Med , vol.13 , pp. 332-339
    • Yamauchi, T.1    Nio, Y.2    Maki, T.3    Kobayashi, M.4    Takazawa, T.5
  • 11
    • 3142701401 scopus 로고    scopus 로고
    • Insulin/Foxo1 pathway regulates expression levels of adiponectin receptors and adiponectin sensitivity
    • Tsuchida A, Yamauchi T, Ito Y, Hada Y, Maki T, et al. (2004) Insulin/Foxo1 pathway regulates expression levels of adiponectin receptors and adiponectin sensitivity. J Biol Chem 279: 30817-30822.
    • (2004) J Biol Chem , vol.279 , pp. 30817-30822
    • Tsuchida, A.1    Yamauchi, T.2    Ito, Y.3    Hada, Y.4    Maki, T.5
  • 13
    • 33744972277 scopus 로고    scopus 로고
    • APPL1 binds to adiponectin receptors and mediates adiponectin signalling and function
    • Mao X, Kikani CK, Riojas RA, Langlais P, Wang L, et al. (2006) APPL1 binds to adiponectin receptors and mediates adiponectin signalling and function. Nat Cell Biol 8: 516-523.
    • (2006) Nat Cell Biol , vol.8 , pp. 516-523
    • Mao, X.1    Kikani, C.K.2    Riojas, R.A.3    Langlais, P.4    Wang, L.5
  • 14
    • 54949140363 scopus 로고    scopus 로고
    • Adiponectin mediates an antiproliferative response in human MDA-MB 231 breast cancer cells
    • Dos Santos E, Benaitreau D, Dieudonne MN, Leneveu MC, Serazin V, et al. (2008) Adiponectin mediates an antiproliferative response in human MDA-MB 231 breast cancer cells. Oncol Rep 20: 971-977.
    • (2008) Oncol Rep , vol.20 , pp. 971-977
    • Dos Santos, E.1    Benaitreau, D.2    Dieudonne, M.N.3    Leneveu, M.C.4    Serazin, V.5
  • 15
    • 0034641647 scopus 로고    scopus 로고
    • Adiponectin, an adipocyte-derived plasma protein, inhibits endothelial NF-kappaB signaling through a cAMP-dependent pathway
    • Ouchi N, Kihara S, Arita Y, Okamoto Y, Maeda K, et al. (2000) Adiponectin, an adipocyte-derived plasma protein, inhibits endothelial NF-kappaB signaling through a cAMP-dependent pathway. Circulation 102: 1296-1301.
    • (2000) Circulation , vol.102 , pp. 1296-1301
    • Ouchi, N.1    Kihara, S.2    Arita, Y.3    Okamoto, Y.4    Maeda, K.5
  • 16
    • 40349108448 scopus 로고    scopus 로고
    • Adiponectin in relation to malignancies: a review of existing basic research and clinical evidence
    • Barb D, Williams CJ, Neuwirth AK, Mantzoros CS, (2007) Adiponectin in relation to malignancies: a review of existing basic research and clinical evidence. Am J Clin Nutr 86: s858-866.
    • (2007) Am J Clin Nutr , vol.86
    • Barb, D.1    Williams, C.J.2    Neuwirth, A.K.3    Mantzoros, C.S.4
  • 17
    • 74049157079 scopus 로고    scopus 로고
    • Adiponectin in insulin resistance: lessons from translational research
    • Ziemke F, Mantzoros CS, (2010) Adiponectin in insulin resistance: lessons from translational research. Am J Clin Nutr 91: 258S-261S.
    • (2010) Am J Clin Nutr , vol.91
    • Ziemke, F.1    Mantzoros, C.S.2
  • 18
    • 77955759804 scopus 로고    scopus 로고
    • Effect of adiponectin on apoptosis: proapoptosis or antiapoptosis
    • Sun Y, Chen X, (2010) Effect of adiponectin on apoptosis: proapoptosis or antiapoptosis? BioFactors 36: 179-186.
    • (2010) BioFactors , vol.36 , pp. 179-186
    • Sun, Y.1    Chen, X.2
  • 19
  • 21
    • 0034999667 scopus 로고    scopus 로고
    • Hypoadiponectinemia in obesity and type 2 diabetes: close association with insulin resistance and hyperinsulinemia
    • Weyer C, Funahashi T, Tanaka S, Hotta K, Matsuzawa Y, et al. (2001) Hypoadiponectinemia in obesity and type 2 diabetes: close association with insulin resistance and hyperinsulinemia. J Clin Endocrinol Metab 86: 1930-1935.
    • (2001) J Clin Endocrinol Metab , vol.86 , pp. 1930-1935
    • Weyer, C.1    Funahashi, T.2    Tanaka, S.3    Hotta, K.4    Matsuzawa, Y.5
  • 22
    • 0034096988 scopus 로고    scopus 로고
    • Plasma concentrations of a novel, adipose-specific protein, adiponectin, in type 2 diabetic patients
    • Hotta K, Funahashi T, Arita Y, Takahashi M, Matsuda M, et al. (2000) Plasma concentrations of a novel, adipose-specific protein, adiponectin, in type 2 diabetic patients. Arterioscler Thromb Vasc Biol 20: 1595-1599.
    • (2000) Arterioscler Thromb Vasc Biol , vol.20 , pp. 1595-1599
    • Hotta, K.1    Funahashi, T.2    Arita, Y.3    Takahashi, M.4    Matsuda, M.5
  • 23
    • 80053478017 scopus 로고    scopus 로고
    • Design and development of a peptide-based adiponectin receptor agonist for cancer treatment
    • Otvos L Jr, Haspinger E, La Russa F, Maspero F, Graziano P, et al. (2011) Design and development of a peptide-based adiponectin receptor agonist for cancer treatment. BMC Biotechnol 11: 90.
    • (2011) BMC Biotechnol , vol.11 , pp. 90
    • Otvos Jr., L.1    Haspinger, E.2    La Russa, F.3    Maspero, F.4    Graziano, P.5
  • 24
    • 70349085370 scopus 로고    scopus 로고
    • A systematic review of the anticancer properties of berberine, a natural product from Chinese herbs
    • Sun Y, Xun K, Wang Y, Chen X, (2009) A systematic review of the anticancer properties of berberine, a natural product from Chinese herbs. Anti-cancer drugs 20: 757-769.
    • (2009) Anti-Cancer Drugs , vol.20 , pp. 757-769
    • Sun, Y.1    Xun, K.2    Wang, Y.3    Chen, X.4
  • 25
    • 78651099528 scopus 로고    scopus 로고
    • Experimental investigation of the immunoregulatory and anti-inflammatory effects of the traditional Chinese medicine "Li-Yan Zhi-Ke Granule" for relieving chronic pharyngitis in rats
    • Sun Y, Zang Z, Xu X, Zhang Z, Zhong L, et al. (2011) Experimental investigation of the immunoregulatory and anti-inflammatory effects of the traditional Chinese medicine "Li-Yan Zhi-Ke Granule" for relieving chronic pharyngitis in rats. Molecular biology reports 38: 199-203.
    • (2011) Molecular Biology Reports , vol.38 , pp. 199-203
    • Sun, Y.1    Zang, Z.2    Xu, X.3    Zhang, Z.4    Zhong, L.5
  • 26
    • 40249106432 scopus 로고    scopus 로고
    • Adiponectin effects on human breast cancer cells are dependent on 17-beta estradiol
    • Pfeiler GH, Buechler C, Neumeier M, Schaffler A, Schmitz G, et al. (2008) Adiponectin effects on human breast cancer cells are dependent on 17-beta estradiol. Oncol Rep 19: 787-793.
    • (2008) Oncol Rep , vol.19 , pp. 787-793
    • Pfeiler, G.H.1    Buechler, C.2    Neumeier, M.3    Schaffler, A.4    Schmitz, G.5
  • 27
    • 67649935011 scopus 로고    scopus 로고
    • Effects of adiponectin and leptin co-treatment on human breast cancer cell growth
    • Nkhata KJ, Ray A, Schuster TF, Grossmann ME, Cleary MP, (2009) Effects of adiponectin and leptin co-treatment on human breast cancer cell growth. Oncol Rep 21: 1611-1619.
    • (2009) Oncol Rep , vol.21 , pp. 1611-1619
    • Nkhata, K.J.1    Ray, A.2    Schuster, T.F.3    Grossmann, M.E.4    Cleary, M.P.5
  • 29
    • 36849020464 scopus 로고    scopus 로고
    • The chemopreventive effects of Saussurea salicifolia through induction of apoptosis and phase II detoxification enzyme
    • Kang K, Lee HJ, Kim CY, Lee SB, Tunsag J, et al. (2007) The chemopreventive effects of Saussurea salicifolia through induction of apoptosis and phase II detoxification enzyme. Biol Pharm Bull 30: 2352-2359.
    • (2007) Biol Pharm Bull , vol.30 , pp. 2352-2359
    • Kang, K.1    Lee, H.J.2    Kim, C.Y.3    Lee, S.B.4    Tunsag, J.5
  • 30
    • 33749520448 scopus 로고    scopus 로고
    • Americanin, a bioactive dibenzylbutyrolactone lignan, from the seeds of Centaurea americana
    • Shoeb M, MacManus SM, Kumarasamy Y, Jaspars M, Nahar L, et al. (2006) Americanin, a bioactive dibenzylbutyrolactone lignan, from the seeds of Centaurea americana. Phytochemistry 67: 2370-2375.
    • (2006) Phytochemistry , vol.67 , pp. 2370-2375
    • Shoeb, M.1    MacManus, S.M.2    Kumarasamy, Y.3    Jaspars, M.4    Nahar, L.5
  • 32
    • 40849118099 scopus 로고    scopus 로고
    • Release of acetylcholine by syringin, an active principle of Eleutherococcus senticosus, to raise insulin secretion in Wistar rats
    • Liu KY, Wu YC, Liu IM, Yu WC, Cheng JT, (2008) Release of acetylcholine by syringin, an active principle of Eleutherococcus senticosus, to raise insulin secretion in Wistar rats. Neurosci Lett 434: 195-199.
    • (2008) Neurosci Lett , vol.434 , pp. 195-199
    • Liu, K.Y.1    Wu, Y.C.2    Liu, I.M.3    Yu, W.C.4    Cheng, J.T.5
  • 33
    • 40349094851 scopus 로고    scopus 로고
    • Hypoglycemic effect of syringin from Eleutherococcus senticosus in streptozotocin-induced diabetic rats
    • Niu HS, Liu IM, Cheng JT, Lin CL, Hsu FL, (2008) Hypoglycemic effect of syringin from Eleutherococcus senticosus in streptozotocin-induced diabetic rats. Planta Med 74: 109-113.
    • (2008) Planta Med , vol.74 , pp. 109-113
    • Niu, H.S.1    Liu, I.M.2    Cheng, J.T.3    Lin, C.L.4    Hsu, F.L.5
  • 34
    • 77957897103 scopus 로고    scopus 로고
    • [Therapeutic effect of syringin on adjuvant arthritis in rats and its mechanisms]
    • Song YY, Li Y, Zhang HQ, (2010) [Therapeutic effect of syringin on adjuvant arthritis in rats and its mechanisms]. Yao Xue Xue Bao 45: 1006-1011.
    • (2010) Yao Xue Xue Bao , vol.45 , pp. 1006-1011
    • Song, Y.Y.1    Li, Y.2    Zhang, H.Q.3
  • 35
    • 84873877188 scopus 로고    scopus 로고
    • Parthenolide induces caspase-independent and AIF-mediated cell death in human osteosarcoma and melanoma cells
    • D'Anneo A, Carlisi D, Lauricella M, Emanuele S, Di Fiore R,et al. (2012) Parthenolide induces caspase-independent and AIF-mediated cell death in human osteosarcoma and melanoma cells. J Cell Physiol.
    • (2012) J Cell Physiol
    • D'Anneo, A.1    Carlisi, D.2    Lauricella, M.3    Emanuele, S.4    Di Fiore, R.5
  • 36
    • 84866480747 scopus 로고    scopus 로고
    • Parthenolide suppresses tumor growth in a xenograft model of colorectal cancer cells by inducing mitochondrial dysfunction and apoptosis
    • Kim SL, Trang KT, Kim SH, Kim IH, Lee SO,et al. (2012) Parthenolide suppresses tumor growth in a xenograft model of colorectal cancer cells by inducing mitochondrial dysfunction and apoptosis. Int J Oncol.
    • (2012) Int J Oncol
    • Kim, S.L.1    Trang, K.T.2    Kim, S.H.3    Kim, I.H.4    Lee, S.O.5
  • 37
    • 58649091086 scopus 로고    scopus 로고
    • Gramine-induced growth inhibition, oxidative damage and antioxidant responses in freshwater cyanobacterium Microcystis aeruginosa
    • Hong Y, Hu HY, Xie X, Sakoda A, Sagehashi M, et al. (2009) Gramine-induced growth inhibition, oxidative damage and antioxidant responses in freshwater cyanobacterium Microcystis aeruginosa. Aquat Toxicol 91: 262-269.
    • (2009) Aquat Toxicol , vol.91 , pp. 262-269
    • Hong, Y.1    Hu, H.Y.2    Xie, X.3    Sakoda, A.4    Sagehashi, M.5
  • 38
    • 84864408367 scopus 로고    scopus 로고
    • Heterocycle-functional gramine analogues: Solvent- and catalyst-free synthesis and their inhibition activities against cell proliferation
    • Ke S, Shi L, Cao X, Yang Q, Liang Y, et al. (2012) Heterocycle-functional gramine analogues: Solvent- and catalyst-free synthesis and their inhibition activities against cell proliferation. Eur J Med Chem 54: 248-254.
    • (2012) Eur J Med Chem , vol.54 , pp. 248-254
    • Ke, S.1    Shi, L.2    Cao, X.3    Yang, Q.4    Liang, Y.5


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.