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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 10, 2013, Pages 2880-2882

Novel racemic tetrahydrocurcuminoid dihydropyrimidinone analogues as potent acetylcholinesterase inhibitors

(5) Arunkhamkaew, Sarawalee a Athipornchai, Anan a Apiratikul, Nuttapon a Suksamrarn, Apichart a Ajavakom, Vachiraporn a

a RAMKHAMHAENG UNIVERSITY (Thailand)

Author keywords

Alzheimer's disease Acetylcholinesterase inhibitor Curcumin Dihydropyrimidinone

Indexed keywords

CHOLINESTERASE INHIBITOR; COPPER SULFATE; DIHYDROPYRIMIDINONE; GALANTAMINE; TETRAHYDROBISDEMETHOXYCURCUMIN; TETRAHYDROCURCUMIN; TETRAHYDRODEMETHOXYCURCUMIN; UNCLASSIFIED DRUG;

ALZHEIMER DISEASE; ARTICLE; BIGINELLI REACTION; CATALYST; DRUG ACTIVITY; DRUG POTENCY; DRUG SCREENING; DRUG SYNTHESIS; IC 50; STRUCTURE ACTIVITY RELATION;

ACETYLCHOLINESTERASE; CHOLINESTERASE INHIBITORS; CURCUMIN; DOSE-RESPONSE RELATIONSHIP, DRUG; HUMANS; MOLECULAR STRUCTURE; PYRIMIDINES; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84876677228 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.03.069 Document Type: Article

Times cited : (40)

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