The development of highly potent inhibitors for porcupine

Journal of Medicinal Chemistry

Volumn 56, Issue 6, 2013, Pages 2700-2704

  Wang, Xiaolei ^a   Moon, Jesung ^a   Dodge, Michael E ^b   Pan, Xinchao ^a   Zhang, Lishu ^b   Hanson, Jordan M ^a   Tuladhar, Rubina ^b   Ma, Zhiqiang ^a   Shi, Heping ^a   Williams, Noelle S ^a   Amatruda, James F ^a   Carroll, Thomas J ^a   Lum, Lawrence ^b   Chen, Chuo ^a  

^a UNIVERSITY OF TEXAS SOUTHWESTERN MEDICAL CENTER   (United States)

^b UNIVERSITY OF TEXAS SOUTHWESTERN MEDICAL CENTER   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ACYLTRANSFERASE; ACYLTRANSFERASE INHIBITOR; PROTEIN PORCUPINE; UNCLASSIFIED DRUG; WNT PROTEIN;

ANTERIOR POSTERIOR AXIS; ARTICLE; KIDNEY TUBULE; NONHUMAN; PALMITOYLATION; STRUCTURE ACTIVITY RELATION; ZEBRA FISH;

DRUG DISCOVERY; ENZYME INHIBITORS; MEMBRANE PROTEINS; SMALL MOLECULE LIBRARIES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84875709096     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm400159c     Document Type: Article

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