Development of inhibitors of the PAS-B domain of the HIF-2α transcription factor

Journal of Medicinal Chemistry

Volumn 56, Issue 4, 2013, Pages 1739-1747

  Rogers, Jamie L ^a   Bayeh, Liela ^a   Scheuermann, Thomas H ^a   Longgood, Jamie ^a   Key, Jason ^a   Naidoo, Jacinth ^a   Melito, Lisa ^a   Shokri, Cameron ^a   Frantz, Doug E ^a   Bruick, Richard K ^a   Gardner, Kevin H ^a   MacMillan, John B ^a   Tambar, Uttam K ^a  

^a UNIVERSITY OF TEXAS SOUTHWESTERN MEDICAL CENTER   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

HYPOXIA INDUCIBLE FACTOR 2ALPHA; HYPOXIA INDUCIBLE FACTOR 2ALPHA INHIBITOR; PROTEIN INHIBITOR; UNCLASSIFIED DRUG;

ARTICLE; DIMERIZATION; HETERODIMERIZATION; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; PAS B DOMAIN; PROTEIN DOMAIN; PROTEIN INTERACTION; STRUCTURE ACTIVITY RELATION; X RAY CRYSTALLOGRAPHY;

EID: 84874605449     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm301847z     Document Type: Article

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