Kinetic characterization of a slow-binding inhibitor of Bla2: Thiomaltol

Journal of Enzyme Inhibition and Medicinal Chemistry

Volumn 28, Issue 1, 2013, Pages 137-142

  Schlesinger, Sara R ^a   Bruner, Britain ^a   Farmer, Patrick J ^a   Kim, Sung Kun ^a  

^a BAYLOR UNIVERSITY   (United States)

Author keywords

Bacillus anthracis; Drug resistance; Htma; Metallo lactamase; Time dependent inhibition

Indexed keywords

ANTIINFECTIVE AGENT; HYDROLASE INHIBITOR; NITROCEFIN; THIOMALTOL; UNCLASSIFIED DRUG;

ANTIBACTERIAL ACTIVITY; ARTICLE; BACILLUS ANTHRACIS; BINDING KINETICS; COMPETITIVE INHIBITION; COMPUTER MODEL; CONTROLLED STUDY; DRUG SCREENING; IC 50; NONHUMAN; PRIORITY JOURNAL;

ANTI-BACTERIAL AGENTS; BACILLUS ANTHRACIS; BETA-LACTAMASES; CEPHALOSPORINS; COMPUTER SIMULATION; ENZYME INHIBITORS; INHIBITORY CONCENTRATION 50; KINETICS; MOLECULAR DOCKING SIMULATION; MOLECULAR STRUCTURE; PYRANS; THIONES;

EID: 84874147380     PISSN: 14756366     EISSN: 14756374     Source Type: Journal    
DOI: 10.3109/14756366.2011.640632     Document Type: Article

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