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Volumn 5, Issue 9, 2010, Pages 1609-1615

Bidentate zinc chelators for α-carbonic anhydrases that produce a trigonal bipyramidal coordination geometry

(8) Wischeler, Johannes Schulze a Innocenti, Alessio b Vullo, Daniela b Agrawal, Arpita c Cohen, Seth M c Heine, Andreas a Supuran, Claudiu T b Klebe, Gerhard a

a PHILIPPS UNIVERSITY MARBURG (Germany)

b UNIVERSITY OF FLORENCE (Italy)

c UNIVERSITY OF CALIFORNIA (United States)

Author keywords

Carbonic anhydrase; Crystal structures; Drug discovery; Inhibitors; Metalloenzymes; Zinc binding groups

Indexed keywords

CARBONATE DEHYDRATASE; CARBONATE DEHYDRATASE INHIBITOR;

ARTICLE; BINDING AFFINITY; CRYSTAL STRUCTURE; DRUG DESIGN; DRUG STRUCTURE; ENZYME INHIBITION; PRIORITY JOURNAL; X RAY CRYSTALLOGRAPHY;

BINDING SITES; CARBONIC ANHYDRASE INHIBITORS; CARBONIC ANHYDRASES; CHELATING AGENTS; CRYSTALLOGRAPHY, X-RAY; HUMANS; PROTEIN BINDING; PROTEIN ISOFORMS; PROTEIN STRUCTURE, TERTIARY; ZINC;

EID: 77956419023 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201000200 Document Type: Article

Times cited : (24)

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