-
1
-
-
38949173868
-
Novel application of multicellular layers culture for in situ evaluation of cytotoxicity and penetration of paclitaxel
-
18271941 10.1111/j.1349-7006.2007.00700.x 1:CAS:528:DC%2BD1MXjs1ygu78%3D
-
Al-Abd AM, Lee JH, Kim SY, Kun N, Kuh HJ (2008) Novel application of multicellular layers culture for in situ evaluation of cytotoxicity and penetration of paclitaxel. Cancer Sci 99:423-431
-
(2008)
Cancer Sci
, vol.99
, pp. 423-431
-
-
Al-Abd, A.M.1
Lee, J.H.2
Kim, S.Y.3
Kun, N.4
Kuh, H.J.5
-
2
-
-
79959908726
-
Synthesis of some new 1,3,5-trisubstituted pyrazolines bearing benzene sulfonamide as anticancer and anti-inflammatory agents
-
21664130 10.1016/j.bmcl.2011.05.061 1:CAS:528:DC%2BC3MXosFWrsLc%3D
-
Bashir R, Ovais S, Yaseen S, Hamid H, Alam MS, Samim M, Singh S, Javed K (2011) Synthesis of some new 1,3,5-trisubstituted pyrazolines bearing benzene sulfonamide as anticancer and anti-inflammatory agents. Bioorg Med Chem Lett 21:4301-4305
-
(2011)
Bioorg Med Chem Lett
, vol.21
, pp. 4301-4305
-
-
Bashir, R.1
Ovais, S.2
Yaseen, S.3
Hamid, H.4
Alam, M.S.5
Samim, M.6
Singh, S.7
Javed, K.8
-
3
-
-
0035834057
-
Photochemically enhanced binding of small molecules to the tumor necrosis factor receptor-1 inhibits the binding of TNF-α
-
11592999 10.1073/pnas.211178398 1:CAS:528:DC%2BD3MXns1equrc%3D
-
Carter PH, Scherle PA, Muckelbauer JA, Voss ME, Liu R-Q, Thompson LA, Tebben AJ, Solomon KA, Lo YC, Li Z, Strzemienski P, Yang G, Falahatpisheh N, Xu M, Wu Z, Farrow NA, Ramnarayan K, Wang J, Rideout D, Yalamoori V, Domaille P, Underwood DJ, Trzaskos JM, Friedman SM, Newton RC, Decicco CP (2001) Photochemically enhanced binding of small molecules to the tumor necrosis factor receptor-1 inhibits the binding of TNF-α. Proc Natl Acad Sci USA 98:11879-11884
-
(2001)
Proc Natl Acad Sci USA
, vol.98
, pp. 11879-11884
-
-
Carter, P.H.1
Scherle, P.A.2
Muckelbauer, J.A.3
Voss, M.E.4
Liu, R.-Q.5
Thompson, L.A.6
Tebben, A.J.7
Solomon, K.A.8
Lo, Y.C.9
Li, Z.10
Strzemienski, P.11
Yang, G.12
Falahatpisheh, N.13
Xu, M.14
Wu, Z.15
Farrow, N.A.16
Ramnarayan, K.17
Wang, J.18
Rideout, D.19
Yalamoori, V.20
Domaille, P.21
Underwood, D.J.22
Trzaskos, J.M.23
Friedman, S.M.24
Newton, R.C.25
Decicco, C.P.26
more..
-
4
-
-
38949192547
-
Targeted cancer therapy: Conferring specificity to cytotoxic drugs
-
17705444 10.1021/ar700108g 1:CAS:528:DC%2BD2sXpt12isLo%3D
-
Chari RV (2008) Targeted cancer therapy: conferring specificity to cytotoxic drugs. Acc Chem Res 41:98-107
-
(2008)
Acc Chem Res
, vol.41
, pp. 98-107
-
-
Chari, R.V.1
-
5
-
-
73549097080
-
Synthesis and inhibitory activity against human monoamine oxidase of N1-thiocarbamoyl-3,5-di(hetero)aryl-4,5-dihydro-(1H)-pyrazole derivatives
-
19926363 10.1016/j.ejmech.2009.11.003 1:CAS:528:DC%2BC3cXos1Smtg%3D%3D
-
Chimenti F, Carradori S, Secci D, Bolasco A, Bizzarri B, Chimenti P, Granese A, Yanez M, Orallo F (2010) Synthesis and inhibitory activity against human monoamine oxidase of N1-thiocarbamoyl-3,5-di(hetero)aryl-4,5-dihydro-(1H)- pyrazole derivatives. Eur J Med Chem 45:800-804
-
(2010)
Eur J Med Chem
, vol.45
, pp. 800-804
-
-
Chimenti, F.1
Carradori, S.2
Secci, D.3
Bolasco, A.4
Bizzarri, B.5
Chimenti, P.6
Granese, A.7
Yanez, M.8
Orallo, F.9
-
6
-
-
77955981424
-
Synthesis and in vitro antitumor activity of new 4,5-dihydropyrazole derivatives
-
20702096 10.1016/j.bmc.2010.07.037 1:CAS:528:DC%2BC3cXhtVKgsLbM
-
Congiu C, Onnis V, Vesci L, Castorina M, Pisano C (2010) Synthesis and in vitro antitumor activity of new 4,5-dihydropyrazole derivatives. Bioorg Med Chem 18:6238-6248
-
(2010)
Bioorg Med Chem
, vol.18
, pp. 6238-6248
-
-
Congiu, C.1
Onnis, V.2
Vesci, L.3
Castorina, M.4
Pisano, C.5
-
7
-
-
20644458125
-
Rhodanine derivatives as inhibitors of JSP-1
-
15961311 10.1016/j.bmcl.2005.05.034 1:CAS:528:DC%2BD2MXlsVCmu7o%3D
-
Cutshall NS, O'Day C, Prerzhdo M (2005) Rhodanine derivatives as inhibitors of JSP-1. Bioorg Med Chem Lett 15:3374-3379
-
(2005)
Bioorg Med Chem Lett
, vol.15
, pp. 3374-3379
-
-
Cutshall, N.S.1
O'Day, C.2
Prerzhdo, M.3
-
8
-
-
37049045930
-
Chalcones and related compounds. Part I. Preparation of nitro-, amino-, and halogeno-chalcones
-
Davey W, Gwilt JR (1953) Chalcones and related compounds. Part I. Preparation of nitro-, amino-, and halogeno-chalcones. J Chem Soc 1008-1014
-
(1953)
J Chem Soc
, pp. 1008-1014
-
-
Davey, W.1
Gwilt, J.R.2
-
9
-
-
33746763743
-
Discovery of small molecule integrin alpha-beta3 antagonists as novel anticancer agents
-
16854058 10.1021/jm051296s 1:CAS:528:DC%2BD28XmsVKmsb4%3D
-
Dayam R, Aiello F, Deng J, Wu Y, Garofalo A, Chen X, Neamati N (2006) Discovery of small molecule integrin alpha-beta3 antagonists as novel anticancer agents. J Med Chem 49:4526-4534
-
(2006)
J Med Chem
, vol.49
, pp. 4526-4534
-
-
Dayam, R.1
Aiello, F.2
Deng, J.3
Wu, Y.4
Garofalo, A.5
Chen, X.6
Neamati, N.7
-
10
-
-
0035150803
-
Identification of small-molecule inhibitors of interaction between the BH3 domain and Bcl-xL
-
11175750 10.1038/35055085 1:CAS:528:DC%2BD3MXht1KmsLY%3D
-
Degterev A, Lugovskoy A, Cardone M, Mulley B, Wagner G, Mitchison T, Yuan J (2001) Identification of small-molecule inhibitors of interaction between the BH3 domain and Bcl-xL. Nat Cell Biol 3:173-182
-
(2001)
Nat Cell Biol
, vol.3
, pp. 173-182
-
-
Degterev, A.1
Lugovskoy, A.2
Cardone, M.3
Mulley, B.4
Wagner, G.5
Mitchison, T.6
Yuan, J.7
-
11
-
-
79751486350
-
Synthesis and antimicrobial activity of some 3,5-diaryl-4,5- dihydropyrazole derivatives
-
1:CAS:528:DC%2BC3MXhvFSksL0%3D
-
El-Enany MM, El-Meligie SEM, Abdou NA, El-Nassan HB (2010) Synthesis and antimicrobial activity of some 3,5-diaryl-4,5-dihydropyrazole derivatives. Orient J Chem 26:1265-1270
-
(2010)
Orient J Chem
, vol.26
, pp. 1265-1270
-
-
El-Enany, M.M.1
El-Meligie, S.E.M.2
Abdou, N.A.3
El-Nassan, H.B.4
-
12
-
-
79955573099
-
Synthesis and antitumor activity of novel pyrido[2,3d][1,2,4]triazolo[4, 3-a]pyrimidin-5-one derivatives
-
21429629 10.1016/j.ejmech.2011.02.055 1:CAS:528:DC%2BC3MXlsVCnsbs%3D
-
El-Nassan HB (2011) Synthesis and antitumor activity of novel pyrido[2,3d][1,2,4]triazolo[4,3-a]pyrimidin-5-one derivatives. Eur J Med Chem 46:2031-2036
-
(2011)
Eur J Med Chem
, vol.46
, pp. 2031-2036
-
-
El-Nassan, H.B.1
-
13
-
-
67649909614
-
Synthesis and antitumor activity of substituted triazolo[4,3-a]pyrimidin- 6-sulfonamide with an incorporated thiazolidinone moiety
-
19540114 10.1016/j.bmcl.2009.05.126 1:CAS:528:DC%2BD1MXosVGmtrk%3D
-
Hafez HN, El-Gazzar A (2009) Synthesis and antitumor activity of substituted triazolo[4,3-a]pyrimidin-6-sulfonamide with an incorporated thiazolidinone moiety. Bioorg Med Chem Lett 19:4143-4147
-
(2009)
Bioorg Med Chem Lett
, vol.19
, pp. 4143-4147
-
-
Hafez, H.N.1
El-Gazzar, A.2
-
14
-
-
77957844111
-
Synthesis and anticancer activity evaluation of 4-thiazolidinones containing benzothiazole moiety
-
20810193 10.1016/j.ejmech.2010.08.008 1:CAS:528:DC%2BC3cXht1KrtrjM
-
Havrylyuk D, Mosula L, Zimenkovsky B, Vasylenko O, Gzella A, Lesyk R (2010) Synthesis and anticancer activity evaluation of 4-thiazolidinones containing benzothiazole moiety. Eur J Med Chem 45:5012-5021
-
(2010)
Eur J Med Chem
, vol.45
, pp. 5012-5021
-
-
Havrylyuk, D.1
Mosula, L.2
Zimenkovsky, B.3
Vasylenko, O.4
Gzella, A.5
Lesyk, R.6
-
15
-
-
80051483748
-
Synthesis and anticancer activity of isatin-based pyrazolines and thiazolidines conjugates
-
10.1002/ardp.201100055
-
Havrylyuk D, Kovach N, Zimenkovsky B, Vasylenko O, Lesyk R (2011) Synthesis and anticancer activity of isatin-based pyrazolines and thiazolidines conjugates. Arch Pharm 344:1-9
-
(2011)
Arch Pharm
, vol.344
, pp. 1-9
-
-
Havrylyuk, D.1
Kovach, N.2
Zimenkovsky, B.3
Vasylenko, O.4
Lesyk, R.5
-
16
-
-
70349387855
-
Breast cancer: Beyond the cutting edge
-
19761355 10.1517/14656560903167957 1:CAS:528:DC%2BD1MXhtFCgsrnI
-
Higa GM (2009) Breast cancer: beyond the cutting edge. Expert Opin Pharmacother 10:2479-2498
-
(2009)
Expert Opin Pharmacother
, vol.10
, pp. 2479-2498
-
-
Higa, G.M.1
-
17
-
-
34548838284
-
Design, synthesis, and biological testing of pyrazoline derivatives of combretastatin-A4
-
17827004 10.1016/j.bmcl.2007.07.105 1:CAS:528:DC%2BD2sXhtFSit7fP
-
Johnson M, Younglove B, Lee L, LeBlanc R, Holt H, Hills P, Mackay H, Brown T, Mooberry SL, Lee M (2007) Design, synthesis, and biological testing of pyrazoline derivatives of combretastatin-A4. Bioorg Med Chem Lett 17:5897-5901
-
(2007)
Bioorg Med Chem Lett
, vol.17
, pp. 5897-5901
-
-
Johnson, M.1
Younglove, B.2
Lee, L.3
Leblanc, R.4
Holt, H.5
Hills, P.6
MacKay, H.7
Brown, T.8
Mooberry, S.L.9
Lee, M.10
-
18
-
-
77952569256
-
Excellent outcomes with adjuvant toremifene or tamoxifen in early stage breast cancer
-
20209619 10.1002/cncr.24962 1:CAS:528:DC%2BC3cXmsFyqsrk%3D
-
Lewis JD, Chagpar AB, Shaughnessy EA, Nurko J, McMasters K, Edwards MJ (2010) Excellent outcomes with adjuvant toremifene or tamoxifen in early stage breast cancer. Cancer 116:2307-2315
-
(2010)
Cancer
, vol.116
, pp. 2307-2315
-
-
Lewis, J.D.1
Chagpar, A.B.2
Shaughnessy, E.A.3
Nurko, J.4
McMasters, K.5
Edwards, M.J.6
-
19
-
-
72049095834
-
Design, synthesis and biological evaluation of thiazolidinone derivatives as potential EGFR and HER-2 kinase inhibitors
-
19914835 10.1016/j.bmc.2009.10.051 1:CAS:528:DC%2BD1MXhsFykurvF
-
Lv P-C, Zhou C-F, Chen J, Liu P-G, Wang K-R, Mao W-J, Li H-Q, Yang Y, Xiong J, Zhu H-L (2010) Design, synthesis and biological evaluation of thiazolidinone derivatives as potential EGFR and HER-2 kinase inhibitors. Bioorg Med Chem 18:314-319
-
(2010)
Bioorg Med Chem
, vol.18
, pp. 314-319
-
-
Lv, P.-C.1
Zhou, C.-F.2
Chen, J.3
Liu, P.-G.4
Wang, K.-R.5
Mao, W.-J.6
Li, H.-Q.7
Yang, Y.8
Xiong, J.9
Zhu, H.-L.10
-
20
-
-
80051931734
-
Synthesis, molecular docking and evaluation of thiazolyl-pyrazoline derivatives as EGFR TK inhibitors and potential anticancer agents
-
21802290 10.1016/j.bmcl.2011.07.010 1:CAS:528:DC%2BC3MXhtVKis73F
-
Lv P, Li D, Li Q, Lu X, Xiao Z, Zhu H (2011) Synthesis, molecular docking and evaluation of thiazolyl-pyrazoline derivatives as EGFR TK inhibitors and potential anticancer agents. Bioorg Med Chem Lett 21:5374-5377
-
(2011)
Bioorg Med Chem Lett
, vol.21
, pp. 5374-5377
-
-
Lv, P.1
Li, D.2
Li, Q.3
Lu, X.4
Xiao, Z.5
Zhu, H.6
-
21
-
-
72049105061
-
Pyrazoline bearing benzimidazoles: Search for anticancer agent
-
19883957 10.1016/j.ejmech.2009.09.032 1:CAS:528:DC%2BD1MXhsF2ju7%2FM
-
Shaharyar M, Abdullah MM, Bakht MA, Majeed J (2010) Pyrazoline bearing benzimidazoles: search for anticancer agent. Eur J Med Chem 45:114-119
-
(2010)
Eur J Med Chem
, vol.45
, pp. 114-119
-
-
Shaharyar, M.1
Abdullah, M.M.2
Bakht, M.A.3
Majeed, J.4
-
22
-
-
64849098639
-
Primary tumor resection improves the survival of younger patients with metastatic breast cancer
-
19212646
-
Shien T, Kinoshita T, Shimizu C, Hojo T, Taira N, Doihara H, Kashi-Tanaka S (2009) Primary tumor resection improves the survival of younger patients with metastatic breast cancer. Oncol Rep 21:827-832
-
(2009)
Oncol Rep
, vol.21
, pp. 827-832
-
-
Shien, T.1
Kinoshita, T.2
Shimizu, C.3
Hojo, T.4
Taira, N.5
Doihara, H.6
Kashi-Tanaka, S.7
-
23
-
-
0025341331
-
New colorimetric assay for anticancer-drug screening
-
2359136 10.1093/jnci/82.13.1107 1:CAS:528:DyaK3cXltVylsL8%3D
-
Skehan P, Storeng R, Scudiero D, Monks A, McMahon J, Vistica D, Warren JT, Bokesch H, Kenney S, Boyd MR (1990) New colorimetric assay for anticancer-drug screening. J Natl Cancer Inst 82:1107-1112
-
(1990)
J Natl Cancer Inst
, vol.82
, pp. 1107-1112
-
-
Skehan, P.1
Storeng, R.2
Scudiero, D.3
Monks, A.4
McMahon, J.5
Vistica, D.6
Warren, J.T.7
Bokesch, H.8
Kenney, S.9
Boyd, M.R.10
-
24
-
-
58849114609
-
Cancer screening in the United States, 2009: A review of current American Cancer Society guidelines and issues in cancer screening
-
19147867 10.3322/caac.20008
-
Smith RA, Cokkinides V, Brawley OW (2009) Cancer screening in the United States, 2009: a review of current American Cancer Society guidelines and issues in cancer screening. CA Cancer J Clin 59:27-41
-
(2009)
CA Cancer J Clin
, vol.59
, pp. 27-41
-
-
Smith, R.A.1
Cokkinides, V.2
Brawley, O.W.3
-
25
-
-
84873986517
-
Über das Ketochlorid und Chlorcarbinol des p,p-Dichlor- benzalacetophenons
-
Straus F, Ackermann A (1909) Über das Ketochlorid und Chlorcarbinol des p,p-Dichlor-benzalacetophenons. Ber Dtsch Chem Ges 42:1804-1823
-
(1909)
Ber Dtsch Chem Ges
, vol.42
, pp. 1804-1823
-
-
Straus, F.1
Ackermann, A.2
-
26
-
-
79953190384
-
Synthesis, characterization and cytotoxicity of the gold(III) complexes of 4,5-dihydropyrazole-1-carbothioamide derivatives
-
21392862 10.1016/j.ejmech.2011.02.031 1:CAS:528:DC%2BC3MXjvFSiurw%3D
-
Wang S, Shao W, Li H, Liu C, Wang K, Zhang J (2011) Synthesis, characterization and cytotoxicity of the gold(III) complexes of 4,5-dihydropyrazole-1-carbothioamide derivatives. Eur J Med Chem 46:1914-1918
-
(2011)
Eur J Med Chem
, vol.46
, pp. 1914-1918
-
-
Wang, S.1
Shao, W.2
Li, H.3
Liu, C.4
Wang, K.5
Zhang, J.6
|