Differential regulation of drug transporter expression by all-trans retinoic acid in hepatoma HepaRG cells and human hepatocytes

European Journal of Pharmaceutical Sciences

Volumn 48, Issue 4-5, 2013, Pages 767-774

  Le Vee, Marc ^a   Jouan, Elodie ^a   Stieger, Bruno ^b   Fardel, Olivier ^a,c  

^a UNIVERSITÉ DE RENNES 1   (France)

^b UNIVERSITY HOSPITAL ZURICH   (Switzerland)

^c PONTCHAILLOU UNIVERSITY HOSPITAL   (France)

Author keywords

Drug transporters; Hepatocytes; RAR; Regulation; Retinoic acid; RXR

Indexed keywords

BREAST CANCER RESISTANCE PROTEIN; CHOLESTEROL 7ALPHA MONOOXYGENASE; CYTOCHROME P450 26A1; MESSENGER RNA; ORGANIC ANION TRANSPORTER 2; ORGANIC ANION TRANSPORTING POLYPEPTIDE 1B1; ORGANIC ANION TRANSPORTING POLYPEPTIDE 2B1; ORGANIC CATION TRANSPORTER 1; RETINOIC ACID; RETINOIC ACID RECEPTOR ALPHA; RETINOID X RECEPTOR ALPHA; SMALL INTERFERING RNA; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; DRUG ACTIVITY; ENZYME ACTIVITY; GENETIC TRANSFECTION; HUMAN; HUMAN CELL; HUMAN TISSUE; IN VITRO STUDY; LIVER CELL CARCINOMA; PRIORITY JOURNAL; PROTEIN EXPRESSION;

AGED; CELL LINE, TUMOR; CELLS, CULTURED; FEMALE; HEPATOCYTES; HUMANS; MALE; MEMBRANE TRANSPORT PROTEINS; MIDDLE AGED; RECEPTORS, RETINOIC ACID; RETINOID X RECEPTOR ALPHA; RNA, MESSENGER; TRETINOIN;

EID: 84873744673     PISSN: 09280987     EISSN: 18790720     Source Type: Journal    
DOI: 10.1016/j.ejps.2013.01.005     Document Type: Article

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