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Volumn 30, Issue 2, 2013, Pages 116-123

Long-acting formulation of a new muscarinic receptor antagonist for the treatment of overactive bladder

Author keywords

5 hydroxymethyl tolterodine; Biodegradable polymer; Microsphere; Pharmacodynamics; Pharmacokinetics

Indexed keywords

CARBACHOL; MICROSPHERE; POLYGLACTIN; TOLTERODINE;

EID: 84873047884     PISSN: 02652048     EISSN: 14645246     Source Type: Journal    
DOI: 10.3109/02652048.2012.704950     Document Type: Article
Times cited : (3)

References (24)
  • 1
    • 0031809695 scopus 로고    scopus 로고
    • Tolterodine, a new antimuscarinic agent: As effective but better tolerated than oxybutynin in patients with an overactive bladder
    • Abrams P, Freeman R, Anderstrom C, Mattiasson A. Tolterodine, a new antimuscarinic agent: As effective but better tolerated than oxybutynin in patients with an overactive bladder. Br J Urol, 1998;81:801-10.
    • (1998) Br J Urol , vol.81 , pp. 801-810
    • Abrams, P.1    Freeman, R.2    Anderstrom, C.3    Mattiasson, A.4
  • 2
    • 0031471714 scopus 로고    scopus 로고
    • Clinical efficacy and safety of tolterodine in the treatment of overactive bladder: A pooled analysis
    • Appell RA. Clinical efficacy and safety of tolterodine in the treatment of overactive bladder: A pooled analysis. Urology, 1997;50:90-6.
    • (1997) Urology , vol.50 , pp. 90-96
    • Appell, R.A.1
  • 3
    • 34147092491 scopus 로고    scopus 로고
    • Poly(lactic-co-glycolic acid)microspheres for the controlled release of huperzine A In vitro and in vivo studies and the application in the treatment of the impaired memory of mice
    • Chu DF, Tian JW, Liu WH, Li Z, Li YX. Poly(lactic-co-glycolic acid)microspheres for the controlled release of huperzine A: In vitro and in vivo studies and the application in the treatment of the impaired memory of mice. Chem Pharm Bull, 2007;55:625-8.
    • (2007) Chem Pharm Bull , vol.55 , pp. 625-628
    • Chu, D.F.1    Tian, J.W.2    Liu, W.H.3    Li, Z.4    Li, Y.X.5
  • 4
    • 33748454642 scopus 로고    scopus 로고
    • Biodegradable PLGA microspheres as a sustained release system for a new luteinizing hormonereleasing hormone (LHRH) antagonist
    • Du L, Cheng JP, Chi Q, Qie JK, Liu Y, Mei XG. Biodegradable PLGA microspheres as a sustained release system for a new luteinizing hormonereleasing hormone (LHRH) antagonist. Chem Pharm Bull, 2006;54:1259-65.
    • (2006) Chem Pharm Bull , vol.54 , pp. 1259-1265
    • Du, L.1    Cheng, J.P.2    Chi, Q.3    Qie, J.K.4    Liu, Y.5    Mei, X.G.6
  • 5
    • 0003428585 scopus 로고    scopus 로고
    • Guidance for industry: Dissolution testing of immediate release solid oral dosage forms
    • FDA.
    • FDA. 1997. Guidance for industry: Dissolution testing of immediate release solid oral dosage forms. Silver Spring, MD: Center for Drug Evaluation and Research, USA, p. 9.
    • (1997) Silver Spring, MD: Center for Drug Evaluation and Research, USA , pp. 9
  • 6
    • 11844259383 scopus 로고    scopus 로고
    • Microencapsulation by solvent extraction/evaporation: Reviewing the state of the art of microsphere preparation process technology
    • Freitas S, Merkle HP, Gander BJ. Microencapsulation by solvent extraction/evaporation: Reviewing the state of the art of microsphere preparation process technology. J Control Release, 2005;102:313-32.
    • (2005) J Control Release , vol.102 , pp. 313-332
    • Freitas, S.1    Merkle, H.P.2    Gander, B.J.3
  • 7
    • 37549018549 scopus 로고    scopus 로고
    • Preparation and characterization of PLGA particles for subcutaneous controlled drug release by membrane emulsification
    • Gasparini G, Kosvintsev SR, Stillwell MT, Holdich RG. Preparation and characterization of PLGA particles for subcutaneous controlled drug release by membrane emulsification. Colloids Surf B, 2008;61:199-207.
    • (2008) Colloids Surf B , vol.61 , pp. 199-207
    • Gasparini, G.1    Kosvintsev, S.R.2    Stillwell, M.T.3    Holdich, R.G.4
  • 8
    • 0026068802 scopus 로고
    • Preparation of poly (l-lactide) microspheres of different crystalline morphology and effect of crystalline morphology on drug release rate
    • Izumikawa S, Yoshioka S, Aso Y, Takeda Y. Preparation of poly (l-lactide) microspheres of different crystalline morphology and effect of crystalline morphology on drug release rate. J Controlled Release, 1991;15:133-40.
    • (1991) J Controlled Release , vol.15 , pp. 133-140
    • Izumikawa, S.1    Yoshioka, S.2    Aso, Y.3    Takeda, Y.4
  • 9
    • 84873029534 scopus 로고    scopus 로고
    • Transdermally administered tolterodine as anti-muscarinic agent for the treatment of overactive bladder
    • Jacobsen LO, Kreilgard B, Hoeck U, Kristensen H. 2003. Transdermally administered tolterodine as anti-muscarinic agent for the treatment of overactive bladder, US Patent 6,517,864.
    • (2003) US Patent 6 , vol.517 , pp. 864
    • Jacobsen, L.O.1    Kreilgard, B.2    Hoeck, U.3    Kristensen, H.4
  • 10
    • 80052339250 scopus 로고    scopus 로고
    • Biodegradable PLGA microsphere for the controlled release of tolterodine derivative
    • Jiang CJ, Teng LS, Teng LR, Li CM, Li YX. Biodegradable PLGA microsphere for the controlled release of tolterodine derivative. J Biotechnol, 2008;136:S416-7.
    • (2008) J Biotechnol , vol.136
    • Jiang, C.J.1    Teng, L.S.2    Teng, L.R.3    Li, C.M.4    Li, Y.X.5
  • 11
    • 0035126767 scopus 로고    scopus 로고
    • Tolterodine oncedaily: Superior efficacy and tolerability in the treatment of the overactive bladder
    • Kerrebroeck PV, Kreder K, Jonas U, Zinner N, Wein AN. Tolterodine oncedaily: Superior efficacy and tolerability in the treatment of the overactive bladder. Urology, 2001;57:414-21.
    • (2001) Urology , vol.57 , pp. 414-421
    • Kerrebroeck, P.V.1    Kreder, K.2    Jonas, U.3    Zinner, N.4    Wein, A.N.5
  • 12
    • 14844364327 scopus 로고    scopus 로고
    • Clinical review of a long-acting, injectable formulation of risperidone
    • Knox ED, Stimmel GL. Clinical review of a long-acting, injectable formulation of risperidone. Clin Ther, 2004;26:1994-2002.
    • (2004) Clin Ther , vol.26 , pp. 1994-2002
    • Knox, E.D.1    Stimmel, G.L.2
  • 13
    • 25844439321 scopus 로고    scopus 로고
    • Preparation and in vitro and in vivo release studies of Huperzine A loaded microspheres for the treatment of Alzheimer's disease
    • Liu WH, Song JL, Liu K, Chu DF, Li YX. Preparation and in vitro and in vivo release studies of Huperzine A loaded microspheres for the treatment of Alzheimer's disease. J Control Release, 2005;107:417-27.
    • (2005) J Control Release , vol.107 , pp. 417-427
    • Liu, W.H.1    Song, J.L.2    Liu, K.3    Chu, D.F.4    Li, Y.X.5
  • 14
    • 33947188787 scopus 로고    scopus 로고
    • Effect of WOW process parameters on morphology and burst release of FITC-dextran loaded PLGA microspheres
    • Mao SR, Xu J, Cai CF. Effect of WOW process parameters on morphology and burst release of FITC-dextran loaded PLGA microspheres. Int J Pharm, 2007;334:137-48.
    • (2007) Int J Pharm , vol.334 , pp. 137-148
    • Mao, S.R.1    Xu, J.2    Cai, C.F.3
  • 15
    • 49049101138 scopus 로고    scopus 로고
    • Optimization of formulation variables for the development of long acting microsphere based depot injection of olanzapine
    • Nahata T, Saini TR. Optimization of formulation variables for the development of long acting microsphere based depot injection of olanzapine. J Microencapsul, 2008;25:426-33.
    • (2008) J Microencapsul , vol.25 , pp. 426-433
    • Nahata, T.1    Saini, T.R.2
  • 16
    • 0030903463 scopus 로고    scopus 로고
    • Tolterodine, a new bladder selective muscarinic receptor antagonist: Preclinical pharmacological and clinical data
    • Nilvebrant L, Hallen B, Larsson G. Tolterodine, a new bladder selective muscarinic receptor antagonist: Preclinical pharmacological and clinical data. Life Sci, 1997;60:1129-36.
    • (1997) Life Sci , vol.60 , pp. 1129-1136
    • Nilvebrant, L.1    Hallen, B.2    Larsson, G.3
  • 17
    • 0028787412 scopus 로고
    • Biodegradable microspheres in drug delivery
    • Okada H, Toguchi H. Biodegradable microspheres in drug delivery. Crit Rev Ther Drug, 1995;12:1-99.
    • (1995) Crit Rev Ther Drug , vol.12 , pp. 1-99
    • Okada, H.1    Toguchi, H.2
  • 18
    • 0344267753 scopus 로고    scopus 로고
    • Serum protein binding of tolterodine and its major metabolites in humans and several animal species
    • Pahlman Z, Gozzi P. Serum protein binding of tolterodine and its major metabolites in humans and several animal species. Biopharm Drug Dispos, 1999;20:91-9.
    • (1999) Biopharm Drug Dispos , vol.20 , pp. 91-9
    • Pahlman, Z.1    Gozzi, P.2
  • 19
    • 55849152841 scopus 로고    scopus 로고
    • Microencapsulation of doxycycline into poly(lactide-co-glycolide) by spray drying technique: Effect of polymer molecular weight on process parameters
    • Patel P, Mundargi RC, Babu VR, Jain D, Rangaswamy V, Aminabhavi TM. Microencapsulation of doxycycline into poly(lactide-co-glycolide) by spray drying technique: Effect of polymer molecular weight on process parameters. J Appl Polym Sci, 2008;108:4038-46.
    • (2008) J Appl Polym Sci , vol.108 , pp. 4038-4046
    • Patel, P.1    Mundargi, R.C.2    Babu, V.R.3    Jain, D.4    Rangaswamy, V.5    Aminabhavi, T.M.6
  • 20
    • 0031918465 scopus 로고    scopus 로고
    • A new muscarinic receptor antagonist is metabolized by cytochromes P450 2D6 and 3A in human liver microsomes
    • Postlind H, Danielson A, Lindgren A, Andersson SH. A new muscarinic receptor antagonist is metabolized by cytochromes P450 2D6 and 3A in human liver microsomes. Drug Metab Dispos, 1998;26:289-93.
    • (1998) Drug Metab Dispos , vol.26 , pp. 289-293
    • Postlind, H.1    Danielson, A.2    Lindgren, A.3    Andersson, S.H.4
  • 21
    • 0242351950 scopus 로고    scopus 로고
    • Biodegradable microparticles for sustained release of a new GnRH antagonist Y Part I: Screening commercial PLGA and formulation technologies
    • Schwach G, Oudry N, Delhomme S, Luck M, Lindner H, Gurny R. Biodegradable microparticles for sustained release of a new GnRH antagonist Y Part I: Screening commercial PLGA and formulation technologies. Eur J Pharm Biopharm, 2003;56:327-36.
    • (2003) Eur J Pharm Biopharm , vol.56 , pp. 327-336
    • Schwach, G.1    Oudry, N.2    Delhomme, S.3    Luck, M.4    Lindner, H.5    Gurny, R.6
  • 22
    • 55649104973 scopus 로고    scopus 로고
    • Principles of encapsulating hydrophobic drugs in PLA/PLGA microparticles
    • Wischke C, Schwendeman SP. Principles of encapsulating hydrophobic drugs in PLA/PLGA microparticles. Int J Pharm, 2008;364:298-327.
    • (2008) Int J Pharm , vol.364 , pp. 298-327
    • Wischke, C.1    Schwendeman, S.P.2
  • 23
    • 0035255916 scopus 로고    scopus 로고
    • Morphology, drug distribution, and in vitro release profiles of biodegradable polymeric microspheres containing protein fabricated by double emulsion solvent extraction/evaporation method
    • Yang YY, Chung TS, Ng NP. Morphology, drug distribution, and in vitro release profiles of biodegradable polymeric microspheres containing protein fabricated by double emulsion solvent extraction/evaporation method. Biomaterials, 2001;22:231-41.
    • (2001) Biomaterials , vol.22 , pp. 231-241
    • Yang, Y.Y.1    Chung, T.S.2    Ng, N.P.3
  • 24
    • 41249098853 scopus 로고    scopus 로고
    • Evaluation of in vivo-in vitro release of dexamethasone from PLGA microspheres
    • Zolnik BS, Burgess DJ. Evaluation of in vivo-in vitro release of dexamethasone from PLGA microspheres. J Controlled Release, 2008;127:137-45.
    • (2008) J Controlled Release , vol.127 , pp. 137-145
    • Zolnik, B.S.1    Burgess, D.J.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.