Discovery of novel human aquaporin-1 blockers

ACS Chemical Biology

Volumn 8, Issue 1, 2013, Pages 249-256

  Seeliger, Daniel ^a   Zapater, Cinta ^b   Krenc, Dawid ^c   Haddoub, Rose ^d   Flitsch, Sabine ^d   Beitz, Eric ^c   Cerdà, Joan ^b   De Groot, Bert L ^a  

^a MAX PLANCK INSTITUTE FOR BIOPHYSICAL CHEMISTRY   (Germany)

^b CSIC   (Spain)

^c UNIVERSITY OF KIEL   (Germany)

^d UNIVERSITY OF MANCHESTER   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

ACETAZOLAMIDE; AQUAPORIN 1; AQUAPORIN 1 INHIBITOR; PROTEIN INHIBITOR; PROTEIN INHIBITOR CPD1; PROTEIN INHIBITOR CPD2; PROTEIN INHIBITOR CPD3; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CONCENTRATION (PARAMETERS); CONTROLLED STUDY; DRUG BINDING; DRUG IDENTIFICATION; DRUG SCREENING; DRUG STRUCTURE; IC 50; MOLECULAR DOCKING; MOLECULAR DYNAMICS; NONHUMAN; OOCYTE; PRIORITY JOURNAL; WATER PERMEABILITY; XENOPUS LAEVIS;

ACETAZOLAMIDE; ANIMALS; AQUAPORIN 1; BINDING SITES; DRUG DISCOVERY; HUMANS; MODELS, MOLECULAR; MOLECULAR DYNAMICS SIMULATION; XENOPUS;

XENOPUS LAEVIS;

EID: 84872550207     PISSN: 15548929     EISSN: 15548937     Source Type: Journal    
DOI: 10.1021/cb300153z     Document Type: Article

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