Comparative efficacy of HgCl2 with candidate aquaporin-1 inhibitors DMSO, gold, TEA+ and acetazolamide

FEBS Letters

Volumn 580, Issue 28-29, 2006, Pages 6679-6684

  Yang, Baoxue ^a   Kim, Jung Kyung ^a   Verkman, A S ^a  

^a UNIVERSITY OF CALIFORNIA   (United States)

Author keywords

AQP1; Drug discovery; Inhibitor; Water channel; Water transport

Indexed keywords

ACETAZOLAMIDE; AQUAPORIN 1; DIMETHYL SULFOXIDE; GOLD; MERCURIC CHLORIDE; PROTEIN INHIBITOR; TETRYLAMMONIUM; WATER;

ANIMAL CELL; ARTICLE; CONTROLLED STUDY; DILUTION; EPITHELIUM CELL; ERYTHROCYTE; HUMAN; HUMAN CELL; IC 50; LIGHT SCATTERING; MOUSE; NONHUMAN; OSMOSIS; PRIORITY JOURNAL; RAT; WATER PERMEABILITY; ANIMAL; CELL MEMBRANE PERMEABILITY; COMPARATIVE STUDY; DRUG ANTAGONISM; DRUG EFFECT; FISCHER 344 RAT; RADIATION SCATTERING; TRANSPORT AT THE CELLULAR LEVEL;

ACETAZOLAMIDE; ANIMALS; AQUAPORIN 1; BIOLOGICAL TRANSPORT; CELL MEMBRANE PERMEABILITY; DIMETHYL SULFOXIDE; EPITHELIAL CELLS; GOLD; HUMANS; MERCURIC CHLORIDE; MICE; OSMOSIS; RATS; RATS, INBRED F344; SCATTERING, RADIATION; TETRAETHYLAMMONIUM; WATER;

EID: 33751502148     PISSN: 00145793     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.febslet.2006.11.025     Document Type: Article

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