Heterobivalent dual-target probe for targeting GRP and Y1 receptors on tumor cells

Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 3, 2013, Pages 687-692

  Shrivastava, Ajay ^a   Wang, Shu Huei ^a   Raju, Natarajan ^a   Gierach, Izabela ^a   Ding, Haiming ^a   Tweedle, Michael F ^a  

^a OHIO STATE UNIVERSITY   (United States)

Author keywords

AMBA; Bombesin; Breast cancer; BVD15; DO3A; Gastrin releasing peptide receptor; Heterobivalent dual target probe; Hormone peptide; Imaging probe; Neuromedin B; Neuropeptide Y; Prostate cancer; Y1 receptor

Indexed keywords

BOMBESIN DERIVATIVE; GASTRIN RELEASING PEPTIDE RECEPTOR; HETEROBIVALENT LIGAND; NEUROPEPTIDE Y1 RECEPTOR; RADIOISOTOPE; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; DRUG BINDING; DRUG TARGETING; HUMAN; HUMAN CELL; HUMAN TISSUE; IC 50; PROTEIN BINDING; PROTEIN EXPRESSION; TUMOR CELL;

AMINO ACID SEQUENCE; ANIMALS; BREAST NEOPLASMS; CELL LINE, TUMOR; CHEMISTRY TECHNIQUES, SYNTHETIC; DRUG DELIVERY SYSTEMS; FEMALE; HUMANS; INHIBITORY CONCENTRATION 50; LIGANDS; MOLECULAR SEQUENCE DATA; PEPTIDES; PROTEIN BINDING; RECEPTORS, BOMBESIN; RECEPTORS, NEUROPEPTIDE Y; SWINE;

SUS;

EID: 84872344965     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2012.11.110     Document Type: Article

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