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Volumn 112, Issue 2, 2013, Pages 124-131

The Effect of Paracetamol and Tropisetron on Pain: Experimental Studies and a Review of Published Data

Author keywords

[No Author keywords available]

Indexed keywords

GRANISETRON; ONDANSETRON; PARACETAMOL; PLACEBO; TROPISETRON;

EID: 84872167481     PISSN: 17427835     EISSN: 17427843     Source Type: Journal    
DOI: 10.1111/j.1742-7843.2012.00935.x     Document Type: Article
Times cited : (22)

References (46)
  • 1
    • 55049106413 scopus 로고    scopus 로고
    • Single dose oral paracetamol (acetaminophen) for postoperative pain in adults
    • Oct 8(4):CD004602.
    • Toms L, McQuay HJ, Derry S, Moore RA. Single dose oral paracetamol (acetaminophen) for postoperative pain in adults. Coch Database Sys Rev 2008; Oct 8(4):CD004602.
    • (2008) Coch Database Sys Rev
    • Toms, L.1    McQuay, H.J.2    Derry, S.3    Moore, R.A.4
  • 2
    • 0026653542 scopus 로고
    • Plasma and cerebrospinal fluid concentrations of paracetamol after a single intravenous dose of propacetamol
    • Bannwarth B, Netter P, Lapicque F, Gillet P, Péré P, Boccard E et al. Plasma and cerebrospinal fluid concentrations of paracetamol after a single intravenous dose of propacetamol. Br J Clin Pharmac 1992;34:79-81.
    • (1992) Br J Clin Pharmac , vol.34 , pp. 79-81
    • Bannwarth, B.1    Netter, P.2    Lapicque, F.3    Gillet, P.4    Péré, P.5    Boccard, E.6
  • 4
    • 25644445318 scopus 로고    scopus 로고
    • Paracetamol and the Cyclooxygenase-3 puzzle: sorting out facts, fictions and uncertainties
    • Kis B, Snipes JA, Busija DW. Paracetamol and the Cyclooxygenase-3 puzzle: sorting out facts, fictions and uncertainties. J Pharmacol Exp Ther 2005;315:1-7.
    • (2005) J Pharmacol Exp Ther , vol.315 , pp. 1-7
    • Kis, B.1    Snipes, J.A.2    Busija, D.W.3
  • 5
    • 38949136999 scopus 로고    scopus 로고
    • Paracetamol (acetaminophen) is a selective cyclooxygenase-2 inhibitor in man
    • Hinz B, Cheremina O, Brune K. Paracetamol (acetaminophen) is a selective cyclooxygenase-2 inhibitor in man. FASEB J 2008;22:383-90.
    • (2008) FASEB J , vol.22 , pp. 383-390
    • Hinz, B.1    Cheremina, O.2    Brune, K.3
  • 6
    • 34248563753 scopus 로고    scopus 로고
    • Paracetamol selectively suppresses peripheral prostaglandin E2 release and increases COX-2 gene expression in a clinical model of acute inflammation
    • Lee Y-S, Kim H, Brahim JS, Rowan J, Lee G, Dionne RA. Paracetamol selectively suppresses peripheral prostaglandin E2 release and increases COX-2 gene expression in a clinical model of acute inflammation. Pain 2007;129:279-86.
    • (2007) Pain , vol.129 , pp. 279-286
    • Lee, Y.-S.1    Kim, H.2    Brahim, J.S.3    Rowan, J.4    Lee, G.5    Dionne, R.A.6
  • 7
    • 39449100661 scopus 로고    scopus 로고
    • Different mechanisms underlie the analgesic actions of paracetamol and dipyrone in a rat model of inflammatory pain
    • Rezende RM, França DS, Menezes GB, dos Reis WGP, Bakhle YS, Francischi JN. Different mechanisms underlie the analgesic actions of paracetamol and dipyrone in a rat model of inflammatory pain. Br J Pharmacol 2007;153:760-8.
    • (2007) Br J Pharmacol , vol.153 , pp. 760-768
    • Rezende, R.M.1    França, D.S.2    Menezes, G.B.3    dos Reis, W.G.P.4    Bakhle, Y.S.5    Francischi, J.N.6
  • 8
    • 17144408419 scopus 로고    scopus 로고
    • Mechanism of action of paracetamol
    • Graham GG, Scott KF. Mechanism of action of paracetamol. Am J Ther 2005;12:46-55.
    • (2005) Am J Ther , vol.12 , pp. 46-55
    • Graham, G.G.1    Scott, K.F.2
  • 10
    • 32044453549 scopus 로고    scopus 로고
    • The analgesic activity of paracetamol is prevented by the blockade of cannabinoid CB1 receptors
    • Ottani A, Leone S, Sandrini M, Ferrari A, Bertolini A. The analgesic activity of paracetamol is prevented by the blockade of cannabinoid CB1 receptors. Eur J Pharmacol 2006;531:280-1.
    • (2006) Eur J Pharmacol , vol.531 , pp. 280-281
    • Ottani, A.1    Leone, S.2    Sandrini, M.3    Ferrari, A.4    Bertolini, A.5
  • 11
    • 51749108193 scopus 로고    scopus 로고
    • Endocannabinoid and serotonergic systems are needed for paracetamol-induced analgesia
    • Mallet C, Daulhac L, Bonnefont J, Ledent C, Etienne M, Chapuy E, et al. Endocannabinoid and serotonergic systems are needed for paracetamol-induced analgesia. Pain 2008;139:190-200.
    • (2008) Pain , vol.139 , pp. 190-200
    • Mallet, C.1    Daulhac, L.2    Bonnefont, J.3    Ledent, C.4    Etienne, M.5    Chapuy, E.6
  • 12
    • 82555196604 scopus 로고    scopus 로고
    • TRPA1 mediates spinal antinociception induced by acetaminophen and the cannabinoid Δ(9)-tetrahydrocannabiorcol
    • Andersson DA, Gentry C, Alenmyr L, Killander D, Lewis SE, Andersson A et al. TRPA1 mediates spinal antinociception induced by acetaminophen and the cannabinoid Δ(9)-tetrahydrocannabiorcol. Nat Commun 2011;2:551.
    • (2011) Nat Commun , vol.2 , pp. 551
    • Andersson, D.A.1    Gentry, C.2    Alenmyr, L.3    Killander, D.4    Lewis, S.E.5    Andersson, A.6
  • 13
    • 0030426275 scopus 로고    scopus 로고
    • Paracetamol exerts a spinal antinociceptive effect involving an indirect interaction with 5-hydroxytryptamine3-receptors: in vivo and in vitro evidence
    • Pelissier T, Alloui A, Caussade F, Dubray C, Cloarec A, Lavarenne J et al. Paracetamol exerts a spinal antinociceptive effect involving an indirect interaction with 5-hydroxytryptamine3-receptors: in vivo and in vitro evidence. J Pharmacol Exp Ther 1996;278:8-14.
    • (1996) J Pharmacol Exp Ther , vol.278 , pp. 8-14
    • Pelissier, T.1    Alloui, A.2    Caussade, F.3    Dubray, C.4    Cloarec, A.5    Lavarenne, J.6
  • 14
    • 0029741730 scopus 로고    scopus 로고
    • Tropisetron inhibits the antinociceptive effect of intrathecally administered paracetamol and serotonin
    • Alloui A, Pelissier T, Dubray C, Lavarenne J, Eschalier A. Tropisetron inhibits the antinociceptive effect of intrathecally administered paracetamol and serotonin. Fundam Clin Pharmacol 1996;10:406-7.
    • (1996) Fundam Clin Pharmacol , vol.10 , pp. 406-407
    • Alloui, A.1    Pelissier, T.2    Dubray, C.3    Lavarenne, J.4    Eschalier, A.5
  • 15
    • 4944239125 scopus 로고    scopus 로고
    • Paracetamol: a central analgesic drug that involves a spinal tropisetron-sensitive, non-5-HT3 receptor-mediated effect
    • Libert F, Bonnefont J, Bourinet E, Doucet E, Alloui A, Hamon M et al. Paracetamol: a central analgesic drug that involves a spinal tropisetron-sensitive, non-5-HT3 receptor-mediated effect. Mol Pharmacol 2004;66:728-34.
    • (2004) Mol Pharmacol , vol.66 , pp. 728-734
    • Libert, F.1    Bonnefont, J.2    Bourinet, E.3    Doucet, E.4    Alloui, A.5    Hamon, M.6
  • 16
    • 61449108148 scopus 로고    scopus 로고
    • Modulation of paracetamol and nefopam antinociception by serotonin 5-HT3 receptor antagonists in mice
    • Girard P, Pansart Y, Coppé M-C, Niedergang B, Gillardin J-M. Modulation of paracetamol and nefopam antinociception by serotonin 5-HT3 receptor antagonists in mice. Pharmacology 2009;83:243-6.
    • (2009) Pharmacology , vol.83 , pp. 243-246
    • Girard, P.1    Pansart, Y.2    Coppé, M.-C.3    Niedergang, B.4    Gillardin, J.-M.5
  • 17
    • 79952198242 scopus 로고    scopus 로고
    • Ondansetron does not block paracetamol-induced analgesia in a mouse model of fracture pain
    • Minville V, Fourcade O, Mazoit JX, Girolami JP, Tack I. Ondansetron does not block paracetamol-induced analgesia in a mouse model of fracture pain. Br J Anaesth 2011;106:112-8.
    • (2011) Br J Anaesth , vol.106 , pp. 112-118
    • Minville, V.1    Fourcade, O.2    Mazoit, J.X.3    Girolami, J.P.4    Tack, I.5
  • 20
    • 77952583915 scopus 로고    scopus 로고
    • The influence of ondansetron on the analgesic effect of paracetamol after laparoscopic hysterectomy
    • Jokela R, Ahonen J, Seitsonen E, Marjakangas P, Korttila K. The influence of ondansetron on the analgesic effect of paracetamol after laparoscopic hysterectomy. Clin Pharmacol Ther 2010;87:672-8.
    • (2010) Clin Pharmacol Ther , vol.87 , pp. 672-678
    • Jokela, R.1    Ahonen, J.2    Seitsonen, E.3    Marjakangas, P.4    Korttila, K.5
  • 22
    • 84859876148 scopus 로고    scopus 로고
    • Effect of pain on autonomic nervous system indices derived from photoplethysmography in healthy volunteers
    • Feb 26
    • Hamunen K, Kontinen V, Hakala E, Talke P, Paloheimo M, Kalso E. Effect of pain on autonomic nervous system indices derived from photoplethysmography in healthy volunteers. Br J Anesth 2012; Feb 26:1-7.
    • (2012) Br J Anesth , pp. 1-7
    • Hamunen, K.1    Kontinen, V.2    Hakala, E.3    Talke, P.4    Paloheimo, M.5    Kalso, E.6
  • 25
    • 0036292398 scopus 로고    scopus 로고
    • A new highly reliable instrument for the assessment of pre- and postoperative gynecological pain
    • Stener-Victorin E, Kowalski J, Lundeberg T. A new highly reliable instrument for the assessment of pre- and postoperative gynecological pain. Anesth Analg 2002;95:151-7.
    • (2002) Anesth Analg , vol.95 , pp. 151-157
    • Stener-Victorin, E.1    Kowalski, J.2    Lundeberg, T.3
  • 28
    • 0034534187 scopus 로고    scopus 로고
    • Efficacy and tolerability of tropisetron in primary fibromyalgia - a highly selective and competitive 5-HT3 receptor antagonist. German Fibromyalgia Study Group
    • Färber L, Stratz T, Brückle W, Späth M, Pongratz D, Lautenschläger J et al. Efficacy and tolerability of tropisetron in primary fibromyalgia - a highly selective and competitive 5-HT3 receptor antagonist. German Fibromyalgia Study Group. Scand J Rheumatol Suppl 2000;113:49-54.
    • (2000) Scand J Rheumatol Suppl , vol.113 , pp. 49-54
    • Färber, L.1    Stratz, T.2    Brückle, W.3    Späth, M.4    Pongratz, D.5    Lautenschläger, J.6
  • 29
    • 4444313622 scopus 로고    scopus 로고
    • Treatment of chronic low back pain with tropisetron
    • Stratz T, Müller W. Treatment of chronic low back pain with tropisetron. Scand J Rheumatol, Suppl 2004;119:76-78.
    • (2004) Scand J Rheumatol, Suppl , vol.119 , pp. 76-78
    • Stratz, T.1    Müller, W.2
  • 30
    • 4444254988 scopus 로고    scopus 로고
    • Intra-articular treatment of arthritides and activated osteoarthritis with the 5-HT3 receptor antagonist. A double-blind study compared with methylprednisolone
    • Samborski W, Stratz T, Mackiewitz S, Müller W. Intra-articular treatment of arthritides and activated osteoarthritis with the 5-HT3 receptor antagonist. A double-blind study compared with methylprednisolone. Scand J Rheumatol, Suppl 2004;119:51-54.
    • (2004) Scand J Rheumatol, Suppl , vol.119 , pp. 51-54
    • Samborski, W.1    Stratz, T.2    Mackiewitz, S.3    Müller, W.4
  • 31
    • 69949128268 scopus 로고    scopus 로고
    • Assessing efficacy of non-opioid analgesics in experimental pain models in healthy volunteers: an updated review
    • Staahl C, Olesen A, Andresen T, Arendt-Nielsen L, Drewes A. Assessing efficacy of non-opioid analgesics in experimental pain models in healthy volunteers: an updated review. Br J Clin Pharmacol 2009;68:322-41.
    • (2009) Br J Clin Pharmacol , vol.68 , pp. 322-341
    • Staahl, C.1    Olesen, A.2    Andresen, T.3    Arendt-Nielsen, L.4    Drewes, A.5
  • 32
    • 84930478017 scopus 로고    scopus 로고
    • Human experimental pain models for assessing the therapeutic efficacy of analgesic drugs
    • Olesen AE, Andresen T, Staahl C, Drewes AM. Human experimental pain models for assessing the therapeutic efficacy of analgesic drugs. Pharmacol Rev 2012;64:722-79.
    • (2012) Pharmacol Rev , vol.64 , pp. 722-779
    • Olesen, A.E.1    Andresen, T.2    Staahl, C.3    Drewes, A.M.4
  • 33
    • 0026646143 scopus 로고
    • Effects of paracetamol and antipyrine on non-inflammatory pain and EEG activity
    • Bromm B, Forth W, Richter E, Scharein E. Effects of paracetamol and antipyrine on non-inflammatory pain and EEG activity. Pain 1992;50:213-21.
    • (1992) Pain , vol.50 , pp. 213-221
    • Bromm, B.1    Forth, W.2    Richter, E.3    Scharein, E.4
  • 34
    • 0031919614 scopus 로고    scopus 로고
    • Dose-related effects of oral paracetamol on cold-induced pain: A double-blind, randomized, placebo-controlled trial
    • Yuan C-S, Karrison T, Wu JA, Lowell T, Lynch J, Foss J. Dose-related effects of oral paracetamol on cold-induced pain: A double-blind, randomized, placebo-controlled trial. Clin Pharmacol Ther 1998;63:379-83.
    • (1998) Clin Pharmacol Ther , vol.63 , pp. 379-383
    • Yuan, C.-S.1    Karrison, T.2    Wu, J.A.3    Lowell, T.4    Lynch, J.5    Foss, J.6
  • 35
    • 70149116337 scopus 로고    scopus 로고
    • Randomized double-blind placebo controlled crossover study of paracetamol, ibuprofen, paracetamol/hydrocodone, and placebo for the relief of pain from a standard painful stimulus
    • Miner J. Randomized double-blind placebo controlled crossover study of paracetamol, ibuprofen, paracetamol/hydrocodone, and placebo for the relief of pain from a standard painful stimulus. Acad Emerg Med 2009;16:911-4.
    • (2009) Acad Emerg Med , vol.16 , pp. 911-914
    • Miner, J.1
  • 37
    • 0026013315 scopus 로고
    • A comparison of the hypoalgesic effect of paracetamol in slow-release and plain tablets on laser-induced pain
    • Nielsen JC, Bjerring P, Arendt-Nielsen L. A comparison of the hypoalgesic effect of paracetamol in slow-release and plain tablets on laser-induced pain. Br J Clin Pharmacol 1991;31:267-70.
    • (1991) Br J Clin Pharmacol , vol.31 , pp. 267-270
    • Nielsen, J.C.1    Bjerring, P.2    Arendt-Nielsen, L.3
  • 38
    • 0026546980 scopus 로고
    • Analgesic efficacy of immediate and sustained release paracetamol and plasma concentration of paracetamol. Double blind, placebo-controlled evaluation using painful laser stimulation
    • Nielsen JC, Bjerring P, Arendt-Nielsen L, Petterson KJ. Analgesic efficacy of immediate and sustained release paracetamol and plasma concentration of paracetamol. Double blind, placebo-controlled evaluation using painful laser stimulation. Eur J Clin Pharmacol 1992;42:261-4.
    • (1992) Eur J Clin Pharmacol , vol.42 , pp. 261-264
    • Nielsen, J.C.1    Bjerring, P.2    Arendt-Nielsen, L.3    Petterson, K.J.4
  • 40
    • 32844473613 scopus 로고    scopus 로고
    • Adding propacetamol to ketorolac increases the tolerance to painful pressure
    • Romundstad L, Stubhaug A, Niemi G, Rosseland LA, Breivik H. Adding propacetamol to ketorolac increases the tolerance to painful pressure. Eur J Pain 2006;10:177-83.
    • (2006) Eur J Pain , vol.10 , pp. 177-183
    • Romundstad, L.1    Stubhaug, A.2    Niemi, G.3    Rosseland, L.A.4    Breivik, H.5
  • 41
    • 34249094123 scopus 로고    scopus 로고
    • Caffeine accelerates absorption and enhances the analgesic effect of paracetamol
    • Renner B, Clarke G, Grattan T, Beisel A, Mueller C, Werner U et al. Caffeine accelerates absorption and enhances the analgesic effect of paracetamol. J Clin Pharmacol 2007;47:715-26.
    • (2007) J Clin Pharmacol , vol.47 , pp. 715-726
    • Renner, B.1    Clarke, G.2    Grattan, T.3    Beisel, A.4    Mueller, C.5    Werner, U.6
  • 42
    • 1342342982 scopus 로고    scopus 로고
    • The cyclooxygenase isozyme inhibitors parecoxib and paracetamol reduce central hyperalgesia in humans
    • Koppert W, Wehrfritz A, Korber N, Sittl R, Albrecht S, Schuttler J et al. The cyclooxygenase isozyme inhibitors parecoxib and paracetamol reduce central hyperalgesia in humans. Pain 2004;108:148-53.
    • (2004) Pain , vol.108 , pp. 148-153
    • Koppert, W.1    Wehrfritz, A.2    Korber, N.3    Sittl, R.4    Albrecht, S.5    Schuttler, J.6
  • 43
    • 43549096159 scopus 로고    scopus 로고
    • Supra-additive effects of tramadol and paracetamol in a human pain model
    • Filitz J, Ihmsen H, Gunther W, Troster A, Schwilden H, Schuttler J et al. Supra-additive effects of tramadol and paracetamol in a human pain model. Pain 2008;136:262-70.
    • (2008) Pain , vol.136 , pp. 262-270
    • Filitz, J.1    Ihmsen, H.2    Gunther, W.3    Troster, A.4    Schwilden, H.5    Schuttler, J.6
  • 45
    • 33645025625 scopus 로고    scopus 로고
    • Hyperalgesia induced by cutaneous freeze injury for testing analgesics in healthy volunteers
    • Chassaing C, Schmidt J, Eschalier A, Cardot JM, Dubray C. Hyperalgesia induced by cutaneous freeze injury for testing analgesics in healthy volunteers. Br J Clin Pharmacol 2006;61:389-97.
    • (2006) Br J Clin Pharmacol , vol.61 , pp. 389-397
    • Chassaing, C.1    Schmidt, J.2    Eschalier, A.3    Cardot, J.M.4    Dubray, C.5
  • 46
    • 79956064862 scopus 로고    scopus 로고
    • Tropisetron blocks analgesic action of paracetamol: a human pain model study
    • Bandschapp O, Filitz J, Urwyler A, Koppert W, Ruppen W. Tropisetron blocks analgesic action of paracetamol: a human pain model study. Pain 2011;152:1304-10.
    • (2011) Pain , vol.152 , pp. 1304-1310
    • Bandschapp, O.1    Filitz, J.2    Urwyler, A.3    Koppert, W.4    Ruppen, W.5


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