Targeting the DNA-binding activity of the human ERG transcription factor using new heterocyclic dithiophene diamidines

Nucleic Acids Research

Volumn 41, Issue 1, 2013, Pages 125-138

  Nhili, Raja ^a   Peixoto, Paul ^a   Depauw, Sabine ^a   Flajollet, Sébastien ^a   Dezitter, Xavier ^a   Munde, Manoj M ^b   Ismail, Mohamed A ^b   Kumar, Arvind ^b   Farahat, Abdelbasset A ^b   Stephens, Chad E ^b   Duterque Coquillaud, Martine ^a   David Wilson, W ^b   Boykin, David W ^b   David Cordonnier, Marie Hélène ^a  

^a UNIV LILLE   (France)

^b GEORGIA STATE UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

DIAMIDINE DERIVATIVE; HETROCYCLIC DITHIOPHENE DIAMIDINE DERIVATIVE; LUCIFERASE; OSTEOPONTIN; TRANSCRIPTION FACTOR ERG; UNCLASSIFIED DRUG;

ARTICLE; BINDING SITE; BIOSENSOR; COMPLEX FORMATION; CONTROLLED STUDY; DNA FOOTPRINTING; DNA SEQUENCE; GEL MOBILITY SHIFT ASSAY; HUMAN; HUMAN CELL; IN VITRO STUDY; PRIORITY JOURNAL; PROMOTER REGION; PROTEIN DNA INTERACTION; PROTEIN TARGETING; REPORTER GENE; SPECTROMETRY; STRUCTURE ACTIVITY RELATION; SURFACE PLASMON RESONANCE; TRANSCRIPTION REGULATION;

AMIDINES; ANTINEOPLASTIC AGENTS; BINDING SITES; CELL LINE, TUMOR; DNA; DRUG EVALUATION, PRECLINICAL; HUMANS; THIOPHENES; TRANS-ACTIVATORS; TRANSCRIPTIONAL ACTIVATION;

EID: 84871748962     PISSN: 03051048     EISSN: 13624962     Source Type: Journal    
DOI: 10.1093/nar/gks971     Document Type: Article

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