Fetal muscle-type nicotinic acetylcholine receptor activation in TE-671 cells and inhibition of fetal movement in a day 40 pregnant goat model by optical isomers of the piperidine alkaloid coniine

Journal of Pharmacology and Experimental Therapeutics

Volumn 344, Issue 1, 2013, Pages 295-307

  Green, Benedict T ^a   Lee, Stephen T ^a   Welch, Kevin D ^a   Pfister, James A ^a   Panter, Kip E ^a  

^a AGRICULTURAL RESEARCH SERVICE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ALPHA CONOTOXIN EI; ALPHA CONOTOXIN GI; CONIINE; MANDELIC ACID; NICOTINE; NICOTINIC RECEPTOR; NICOTINIC RECEPTOR BLOCKING AGENT; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ARTICLE; BINDING SITE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG ANTAGONISM; DRUG RECEPTOR BINDING; DRUG SPECIFICITY; FEMALE; FETUS MOVEMENT; GESTATIONAL AGE; GOAT; HUMAN; HUMAN CELL; IN VITRO STUDY; IN VIVO STUDY; ISOMER; LIGAND BINDING; MUSCLE FIBER MEMBRANE POTENTIAL; NONHUMAN; PRIORITY JOURNAL; PROTEIN EXPRESSION; PROTEIN FUNCTION; PROTEIN INDUCTION; PROTEIN STRUCTURE; STEREOCHEMISTRY; STRUCTURE ACTIVITY RELATION;

ACETYLCHOLINE; ALKALOIDS; ANIMALS; CALCIUM CHANNEL BLOCKERS; CELL LINE; CELL LINE, TUMOR; CONOTOXINS; CRYSTALLIZATION; DOSE-RESPONSE RELATIONSHIP, DRUG; FEMALE; FETAL MOVEMENT; GOATS; HUMANS; MANDELIC ACIDS; MUSCLE, SKELETAL; PIPERIDINES; PREGNANCY; RECEPTORS, NICOTINIC; STEREOISOMERISM;

EID: 84871706848     PISSN: 00223565     EISSN: 15210103     Source Type: Journal    
DOI: 10.1124/jpet.112.199588     Document Type: Article

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