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Volumn 5, Issue , 2012, Pages

SU11652 inhibits tyrosine kinase activity of FLT3 and growth of MV-4-11 cells

Author keywords

Acute myeloid leukemia; FLT3; Inhibitor screening; SU11652; Tyrosine kinase

Indexed keywords

CD135 ANTIGEN; MITOGEN ACTIVATED PROTEIN KINASE; PROTEIN KINASE B; PROTEIN TYROSINE KINASE INHIBITOR; STAT PROTEIN; SU 11652; UNCLASSIFIED DRUG;

EID: 84870405511     PISSN: None     EISSN: 17568722     Source Type: Journal    
DOI: 10.1186/1756-8722-5-72     Document Type: Article
Times cited : (14)

References (26)
  • 1
    • 33751267902 scopus 로고    scopus 로고
    • Acute myeloid leukaemia
    • DOI 10.1016/S0140-6736(06)69780-8, PII S0140673606697808
    • Acute myeloid leukaemia. Estey E, Döhner H, Lancet 2006 368 1894 1907 10.1016/S0140-6736(06)69780-8 17126723 (Pubitemid 44794525)
    • (2006) Lancet , vol.368 , Issue.9550 , pp. 1894-1907
    • Estey, E.1    Dohner, H.2
  • 3
    • 84055218304 scopus 로고    scopus 로고
    • Acute myeloid leukemia: 2012 update on diagnosis, risk stratification, and management
    • 10.1002/ajh.22246 22180162
    • Acute myeloid leukemia: 2012 update on diagnosis, risk stratification, and management. Estey EH, Am J Hematol 2012 87 89 99 10.1002/ajh.22246 22180162
    • (2012) Am J Hematol , vol.87 , pp. 89-99
    • Estey, E.H.1
  • 4
    • 80052836966 scopus 로고    scopus 로고
    • Current findings for recurring mutations in acute myeloid leukemia
    • 10.1186/1756-8722-4-36 21917154
    • Current findings for recurring mutations in acute myeloid leukemia. Takahashi S, J Hematol Oncol 2011 4 36 10.1186/1756-8722-4-36 21917154
    • (2011) J Hematol Oncol , vol.4 , pp. 36
    • Takahashi, S.1
  • 5
    • 84867396974 scopus 로고    scopus 로고
    • Targeting the FMS-like tyrosine kinase 3 in acute myeloid leukemia
    • 10.1038/leu.2012.114 22614177
    • Targeting the FMS-like tyrosine kinase 3 in acute myeloid leukemia. Swords R, Freeman C, Giles F, Leukemia 2012 26 2176 2185 10.1038/leu.2012.114 22614177
    • (2012) Leukemia , vol.26 , pp. 2176-2185
    • Swords, R.1    Freeman, C.2    Giles, F.3
  • 6
    • 84873569249 scopus 로고    scopus 로고
    • FLT3 inhibition-A moving and evolving target in acute myeloid leukaemia
    • 10.1038/leu.2012.195
    • FLT3 inhibition-a moving and evolving target in acute myeloid leukaemia. Leung AY, Man CH, Kwong YL, Leukemia 2012 10.1038/leu.2012.195
    • (2012) Leukemia
    • Leung, A.Y.1    Man, C.H.2    Kwong, Y.L.3
  • 7
    • 0141465061 scopus 로고    scopus 로고
    • The role of FLT3 in haematopoietic malignancies
    • The role of FLT3 in haematopoietic malignancies. Stirewalt DL, Radich JP, Nat Rev Cancer 2003 3 650 665 10.1038/nrc1169 12951584 (Pubitemid 37328820)
    • (2003) Nature Reviews Cancer , vol.3 , Issue.9 , pp. 650-665
    • Stirewalt, D.L.1    Radich, J.P.2
  • 8
    • 73249135797 scopus 로고    scopus 로고
    • Molecular prognostic markers for adult acute myeloid leukemia with normal cytogenetics
    • 10.1186/1756-8722-2-23 19490647
    • Molecular prognostic markers for adult acute myeloid leukemia with normal cytogenetics. Gregory TK, Wald D, Chen Y, Vermaat JM, Xiong Y, Tse W, J Hematol Oncol 2009 2 23 10.1186/1756-8722-2-23 19490647
    • (2009) J Hematol Oncol , vol.2 , pp. 23
    • Gregory, T.K.1    Wald, D.2    Chen, Y.3    Vermaat, J.M.4    Xiong, Y.5    Tse, W.6
  • 9
    • 79953244064 scopus 로고    scopus 로고
    • Downstream molecular pathways of FLT3 in the pathogenesis of acute myeloid leukemia: Biology and therapeutic implications
    • 10.1186/1756-8722-4-13 21453545
    • Downstream molecular pathways of FLT3 in the pathogenesis of acute myeloid leukemia: biology and therapeutic implications. Takahashi S, J Hematol Oncol 2011 4 13 10.1186/1756-8722-4-13 21453545
    • (2011) J Hematol Oncol , vol.4 , pp. 13
    • Takahashi, S.1
  • 12
    • 77951111333 scopus 로고    scopus 로고
    • Novel agents and regimens for acute myeloid leukemia: 2009 ASH annual meeting highlights
    • 10.1186/1756-8722-3-17 20416083
    • Novel agents and regimens for acute myeloid leukemia: 2009 ASH annual meeting highlights. Zhu X, Ma Y, Liu D, J Hematol Oncol 2010 3 17 10.1186/1756-8722-3-17 20416083
    • (2010) J Hematol Oncol , vol.3 , pp. 17
    • Zhu, X.1    Ma, Y.2    Liu, D.3
  • 17
    • 78650073854 scopus 로고    scopus 로고
    • FLT3 as a therapeutic target in AML: Still challenging after all these years
    • 10.1182/blood-2010-04-261867 20705759
    • FLT3 as a therapeutic target in AML: still challenging after all these years. Kindler T, Lipka DB, Fischer T, Blood 2010 116 5089 5102 10.1182/blood-2010-04-261867 20705759
    • (2010) Blood , vol.116 , pp. 5089-5102
    • Kindler, T.1    Lipka, D.B.2    Fischer, T.3
  • 18
    • 77954750384 scopus 로고    scopus 로고
    • Bench to Bedside Targeting of FLT3 in Acute Leukemia
    • 10.2174/138945010791320782 20370649
    • Bench to Bedside Targeting of FLT3 in Acute Leukemia. Pratz KW, Levis MJ, Curr Drug Targets 2010 11 781 789 10.2174/138945010791320782 20370649
    • (2010) Curr Drug Targets , vol.11 , pp. 781-789
    • Pratz, K.W.1    Levis, M.J.2
  • 19
    • 84865229701 scopus 로고    scopus 로고
    • Generation and characterization of a highly effective protein substrate for analysis of FLT3 activity
    • 10.1186/1756-8722-5-39 22800464
    • Generation and characterization of a highly effective protein substrate for analysis of FLT3 activity. Chen Y, Guo Y, Han J, Ho WT, Li S, Fu X, Zhao Z, J Hematol Oncol 2012 5 39 10.1186/1756-8722-5-39 22800464
    • (2012) J Hematol Oncol , vol.5 , pp. 39
    • Chen, Y.1    Guo, Y.2    Han, J.3    Ho, W.T.4    Li, S.5    Fu, X.6    Zhao, Z.7
  • 20
    • 0037100281 scopus 로고    scopus 로고
    • Inhibition of constitutively active forms of mutant kit by multitargeted indolinone tyrosine kinase inhibitors
    • DOI 10.1182/blood-2001-12-0350
    • Inhibition of constitutively active forms of mutant kit by multitargeted indolinone tyrosine kinase inhibitors. Liao AT, Chien MB, Shenoy N, Mendel DB, McMahon G, Cherrington JM, London CA, Blood 2002 100 585 593 10.1182/blood-2001-12-0350 12091352 (Pubitemid 34761123)
    • (2002) Blood , vol.100 , Issue.2 , pp. 585-593
    • Liao, A.T.1    Chien, M.B.2    Shenoy, N.3    Mendel, D.B.4    McMahon, G.5    Cherrington, J.M.6    London, C.A.7
  • 21
    • 0037468875 scopus 로고    scopus 로고
    • Discovery of 5-[5-fluoro-2-oxo-1,2-dihydroindol-(3Z)-ylidenemethyl]-2, 4-dimethyl-1H-pyrrole-3-carboxylic acid (2-diethylaminoethyl)amide, a novel tyrosine kinase inhibitor targeting vascular endothelial and platelet-derived growth factor receptor tyrosine kinase
    • DOI 10.1021/jm0204183
    • Discovery of 5-[5-fluoro-2-oxo-1,2- dihydroindol-(3Z)-ylidenemethyl]-2,4- dimethyl-1H-pyrrole-3-carboxylic acid (2-diethylaminoethyl)amide, a novel tyrosine kinase inhibitor targeting vascular endothelial and platelet-derived growth factor receptor tyrosine kinase. Sun L, Liang C, Shirazian S, Zhou Y, Miller T, Cui J, Fukuda JY, Chu JY, Nematalla A, Wang X, Chen H, Sistla A, Luu TC, Tang F, Wei J, Tang C, J Med Chem 2003 46 1116 1119 10.1021/jm0204183 12646019 (Pubitemid 36428215)
    • (2003) Journal of Medicinal Chemistry , vol.46 , Issue.7 , pp. 1116-1119
    • Sun, L.1    Liang, C.2    Shirazian, S.3    Zhou, Y.4    Miller, T.5    Cui, J.6    Fukuda, J.Y.7    Chu, J.-Y.8    Nematalla, A.9    Wang, X.10    Chen, H.11    Sistla, A.12    Luu, T.C.13    Tang, F.14    Wei, J.15    Tang, C.16
  • 22
    • 0037265645 scopus 로고    scopus 로고
    • FLT3 mutations in acute myeloid leukemia cell lines
    • DOI 10.1038/sj.leu.2402740
    • FLT3 mutations in acute myeloid leukemia cell lines. Quentmeier H, Reinhardt J, Zaborski M, Drexler HG, Leukemia 2003 17 120 124 10.1038/sj.leu.2402740 12529668 (Pubitemid 36175896)
    • (2003) Leukemia , vol.17 , Issue.1 , pp. 120-124
    • Quentmeier, H.1    Reinhardt, J.2    Zaborski, M.3    Drexler, H.G.4
  • 23
    • 33749489416 scopus 로고    scopus 로고
    • The expression of CD30 in anaplastic large cell lymphoma is regulated by nucleophosmin-anaplastic lymphoma kinase-mediated JunB level in a cell type-specific manner
    • DOI 10.1158/0008-5472.CAN-05-4101
    • The Expression of CD30 in Anaplastic Large Cell Lymphoma Is Regulated by Nucleophosmin-Anaplastic Lymphoma Kinase-Mediated JunB Level in a Cell Type-Specific Manner. Hsu FY, Johnston PB, Burke KA, Zhao Y, Cancer Res 2006 66 9002 9008 10.1158/0008-5472.CAN-05-4101 16982741 (Pubitemid 44521118)
    • (2006) Cancer Research , vol.66 , Issue.18 , pp. 9002-9008
    • Hsu, F.Y.-Y.1    Johnston, P.B.2    Burke, K.A.3    Zhao, Y.4
  • 24
    • 84872264689 scopus 로고    scopus 로고
    • JAK2V617F and p53 mutations coexist in erythroleukemia and megakaryoblastic leukemic cell lines
    • 10.1186/2162-3619-1-15 23242571
    • JAK2V617F and p53 mutations coexist in erythroleukemia and megakaryoblastic leukemic cell lines. Zhao W, Du Y, Ho WT, Fu X, Zhao ZJ, Experimental Hematology & Oncology 2012 1 15 10.1186/2162-3619-1-15 23242571
    • (2012) Experimental Hematology & Oncology , vol.1 , pp. 15
    • Zhao, W.1    Du, Y.2    Ho, W.T.3    Fu, X.4    Zhao, Z.J.5
  • 26
    • 35448951230 scopus 로고    scopus 로고
    • V617F Activity
    • DOI 10.1016/j.exphem.2007.07.003, PII S0301472X07004262
    • Characterization of a highly effective protein substrate for analysis of JAK2(V617F) Activity. Li Z, Xing S, Wang S, Ho WT, Zhao ZJ, Exp Hematol 2007 35 1624 1632 10.1016/j.exphem.2007.07.003 17764811 (Pubitemid 47633769)
    • (2007) Experimental Hematology , vol.35 , Issue.11 , pp. 1624-1632
    • Li, Z.1    Xing, S.2    Wang, S.3    Ho, W.T.4    Zhao, Z.J.5


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.