Ex vivo permeation characteristics of venlafaxine through sheep nasal mucosa

European Journal of Pharmaceutical Sciences

Volumn 48, Issue 1-2, 2013, Pages 195-201

  Pund, Swati ^a   Rasve, Ganesh ^a   Borade, Ganesh ^a  

^a Sinhgad Institute of Pharmacy   (India)

Author keywords

Ex vivo permeation; In situ gel; Venlafaxine

Indexed keywords

POLYMER; VENLAFAXINE;

ANIMAL EXPERIMENT; ARTICLE; CONTROLLED STUDY; DRUG DELIVERY SYSTEM; DRUG DIFFUSION; DRUG PENETRATION; DRUG RELEASE; DRUG TRANSPORT; EX VIVO STUDY; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; HISTOPATHOLOGY; MUCOADHESION; NONHUMAN; NOSE MUCOSA; PRIORITY JOURNAL; STEADY STATE;

ADHESIVENESS; ANIMALS; ANTIDEPRESSIVE AGENTS, SECOND-GENERATION; CYCLOHEXANOLS; NASAL MUCOSA; PERMEABILITY; SHEEP;

EID: 84870359903     PISSN: 09280987     EISSN: 18790720     Source Type: Journal    
DOI: 10.1016/j.ejps.2012.10.029     Document Type: Article

References (32)

1. R. Asasutjarit, S. Thanasanchokpibull, A. Fuongfuchat, and S. Veeranondha Optimization and evaluation of thermoresponsive diclofenac sodium ophthalmic in situ gels Int. J. Pharm. 411 2011 128 135
2. S. Basu, and A.K. Bandyopadhyay Development and characterization of mucoadhesive in situ nasal gel of midazolam prepared with Ficus carica mucilage AAPS PharmSciTechnol. 11 2010 1223 1231
3. U. Bonnet, D. Bingmann, J. Wiltfang, N. Scherbaum, and M. Wiemann Modulatory effects of neuropsychopharmaca on intracellular pH of hippocampal neurones in vitro Br. J. Pharmacol. 159 2 2010 474 483
4. Z. Cai, X. Song, F. Sun, Z. Yang, S. Hou, and Z. Liu Formulation and evaluation of in situ gelling systems for intranasal administration of gastrodin AAPS PharmSciTechnol. 12 4 2011 1102 1109
5. H.R. Costantino, L. Illum, G. Brandt, P.H. Johnson, and S.C. Quay Intranasal delivery: physicochemical and therapeutic aspects Int. J. Pharm. 337 2007 1 24
6. A.H. El-Kamel In vitro and in vivo evaluation of Pluronic F127-based ocular delivery system for timolol maleate Int. J. Pharm. 241 2002 47 55
7. F. Fawaz, A. Koffi, M. Guyot, and P. Millet Comparative in vitro-in vivo study of two quinine rectal gel formulations Int. J. Pharm. 280 2004 151 162
8. Q. Gardiner, M. Oluwole, L. Tan, and P.S. White An animal model for training in endoscopic nasal and sinus surgery J. Laryngol. Otol. 110 1996 425 428
9. L.I. Giannola, V.D. Caro, G. Giandalia, M.G. Siragusa, C. Tripodo, A.M. Florena, and G. Campisi Release of naltrexone on buccal mucosa: permeation studies, histological aspects and matrix system design Eur. J. Pharm. Biopharm. 67 2007 425 433
10. J.C. Gilbert, J.L. Richardson, M.C. Davies, K.J. Palin, and J. Hadgraft The effect of solutes and polymers on the gelation properties of Pluronic F-127 solutions for controlled drug delivery J. Controlled Release 5 1987 113 118
11. A.M. Gutierrez, L.G. Stimmel, and Y.J. Aiso Venlafaxine: a 2003 update Clin. Ther. 25 2003 2138 2154
12. S. Haque, S. Md, M. Fazil, M. Kumar, J.K. Sahni, J. Ali, and S. Baboota Venlafaxine loaded chitosan NPs for brain targeting: pharmacokinetic and pharmacodynamic evaluation Carbohydr. Polym. 89 2012 72 79
13. A.A. Heda, A.R. Sonawane, G.H. Naranje, V.G. Somani, and P.K. Puranik Development and in vitro evaluation of betahistine adhesive-type transdermal delivery system Topical J. Pharm. Res. 9 6 2010 516 524
14. L. Illum Nasal delivery. The use of animal models to predict performance in man J. Drug Targeting 3 1996 427 442
15. L. Illum Nasal drug delivery - recent developments and future prospects J. Controlled Release 161 2012 254 263
16. H.Y. Karasulu, Z.E. Sanal, S. Sözer, T. Güneri, and G. Ertan Permeation studies of indomethacin from different emulsions for nasal delivery and their possible anti-inflammatory effects AAPS PharmSciTechnol. 9 2 2008 342 348
17. L. Karlsson, U. Schmitt, M. Josefsson, B. Carlsson, J. Ahlner, F. Bengtsson, F.C. Kugelberg, and C. Hiemke Blood-brain barrier penetration of the enantiomers of venlafaxine and its metabolites in mice lacking P-glycoprotein Eur. Neuropsychopharmacol. 20 2010 632 640
18. C.D. Kilts Potential new drug delivery system for antidepressants: an overview J. Clin. Psychiatry 64 2003 31 33
19. Majithiya, R.J.; Ghosh, P.K.; Umrethia, M.L.; Murthy, R.S.R.; 2006. Thermoreversible-mucoadhesive gel for nasal delivery of sumatriptan. AAPS PharmSciTechnol. 7(3) Article 67, E1-E7.
20. C.D. Mathers, and D. Loncar Projections of global mortality and burden of disease from 2002 to 2030 PLoS Med. 3 11 2006 2011 2030
21. Y.J. Park, C.S. Yong, H.M. Kim, J.D. Rhee, Y.K. Oh, C.K. Kim, and H.G. Choi Effect of sodium chloride on the release, absorption and safety of diclofenac sodium delivered by poloxamer gel Int. J. Pharm. 263 2003 105 111
22. A. Pires, A. Fortuna, G. Alves, and A. Falcão Intranasal drug delivery: how, why and what for? J. Pharm. Pharm. Sci. 12 3 2009 288 311
23. G. Rathnam, N. Narayanan, and R. Ilavarasan Carbopol-based gels for nasal delivery of progesterone AAPS PharmSciTechnol. 9 4 2008 E1 E9
24. T. Rehman, S. Tavelin, and G. Gröbner Chitosan in situ gelation for improved drug loading and retention in poloxamer 407 gels Int. J. Pharm. 409 2011 19 29
25. G. Samson, A.G. Calera, S.D. Girod, F. Faure, E. Decullier, G. Paintaud, C. Vignault, J.Y. Scoazec, C. Pivot, H. Plauchu, and F. Pirot Ex vivo study of bevacizumab transport through porcine nasal mucosa Eur. J. Pharm. Biopharm. 80 2012 465 469
26. I.R. Schmolka Artificial skin. I. Preparation and properties of Pluronic F-127 gels for the treatment of burns J. Biomed. Mater. Res. 6 1972 571 582
27. G. Singh, B. Ghosh, D. Kaushalkumar, and V. Somsekhar Screening of venlafaxine hydrochloride for transdermal delivery: passive diffusion and iontophoresis AAPS PharmSciTechnol. 9 3 2008 791 797
28. S.M. Stahl, M.M. Grady, C. Moret, and M. Briley SNRIs: their pharmacology, clinical efficacy and tolerability in comparison with other classes of antidepressants CNS Spectrosc. 10 2005 732 747
29. S.M. Troy, V.D. Parekar, R.J. Fruncillo, and S.T. Chiang The pharmacokinetics of venlafaxine when given in a twice daily regimen J. Clin. Pharmacol. 35 1995 404 409
30. M.I. Ugwoke, G. Kaufmann, N. Verbeke, and R. Kinget Intranasal bioavailability of apomorphine from carboxymethylcellulose-based drug delivery systems Int. J. Pharm. 202 2000 125 131
31. N.M. Zaki, G.A. Awad, N.D. Mortada, and S.S. Abd El Hady Enhanced bioavailability of metoclopramide HCl by intranasal administration of a mucoadhesive in situ gel with modulated rheological and mucociliary transport properties Eur. J. Pharm. Sci. 32 2007 296 307
32. M. Zhou, and M.D. Donovan Intranasal mucociliary clearance of putative bioadhesive polymer gels Int. J. Pharm. 135 1996 115 125