메뉴 건너뛰기




Volumn 80, Issue 6, 2012, Pages 1003-1008

Evaluation of Structurally Diverse Benzoazepines Clubbed with Coumarins as Mycobacterium tuberculosis Agents

Author keywords

Benzodiazepines; Benzothiazepines; Coumarins; H37Rv; Microplate alamar blue assay; Mtb

Indexed keywords

BENZODIAZEPINE DERIVATIVE; COUMARIN DERIVATIVE; DIBENZOTHIAZEPINE DERIVATIVE;

EID: 84868139977     PISSN: 17470277     EISSN: 17470285     Source Type: Journal    
DOI: 10.1111/j.1747-0285.2012.01436.x     Document Type: Letter
Times cited : (27)

References (38)
  • 1
    • 0038519673 scopus 로고    scopus 로고
    • Progress in TB drug development and what is still needed
    • Duncan K. (2003) Progress in TB drug development and what is still needed. Tuberculosis;83:201-207.
    • (2003) Tuberculosis , vol.83 , pp. 201-207
    • Duncan, K.1
  • 2
    • 33847704942 scopus 로고    scopus 로고
    • Challenges in tuberculosis drug research and development
    • Ginsberg A.M., Spigelman M. (2007) Challenges in tuberculosis drug research and development. Nat Med;13:290-294.
    • (2007) Nat Med , vol.13 , pp. 290-294
    • Ginsberg, A.M.1    Spigelman, M.2
  • 3
    • 84863421391 scopus 로고    scopus 로고
    • Developments in chemical approaches to treat tuberculosis in the last decade
    • Tripathi R.P., Bisht S.S., Ajay A., Sharma A., Misra M., Gupt M.Pd. (2012) Developments in chemical approaches to treat tuberculosis in the last decade. Curr Med Chem;30:488-517.
    • (2012) Curr Med Chem , vol.30 , pp. 488-517
    • Tripathi, R.P.1    Bisht, S.S.2    Ajay, A.3    Sharma, A.4    Misra, M.5    Gupt, MP.6
  • 4
    • 77952542701 scopus 로고    scopus 로고
    • Multidrug-resistant and extensively drug-resistant tuberculosis: a threat to global control of tuberculosis
    • Gandhi N.R., Nunn P., Dheda K., Schaaf H.S., Zignol M., Van Soolingen D., Jensen P., Bayona J. (2010) Multidrug-resistant and extensively drug-resistant tuberculosis: a threat to global control of tuberculosis. Lancet;375:1830-1843.
    • (2010) Lancet , vol.375 , pp. 1830-1843
    • Gandhi, N.R.1    Nunn, P.2    Dheda, K.3    Schaaf, H.S.4    Zignol, M.5    Van Soolingen, D.6    Jensen, P.7    Bayona, J.8
  • 5
  • 6
    • 33847681052 scopus 로고    scopus 로고
    • Antituberculosis drugs: ten years of research
    • Janin Y.L. (2007) Antituberculosis drugs: ten years of research. Bioorg Med Chem;15:2479-2513.
    • (2007) Bioorg Med Chem , vol.15 , pp. 2479-2513
    • Janin, Y.L.1
  • 7
    • 84881377750 scopus 로고    scopus 로고
    • Current approaches to tuberculosis drug discovery and development, Series No. 14, Chapter 9
    • Cambridge, UK: RSC publishing.
    • Mitton-Fry M.J., Hanna D. (2012) Current approaches to tuberculosis drug discovery and development, Series No. 14, Chapter 9. Neglected Disease and Drug Discovery. Cambridge, UK: RSC publishing.
    • (2012) Neglected Disease and Drug Discovery
    • Mitton-Fry, M.J.1    Hanna, D.2
  • 8
    • 33846995990 scopus 로고    scopus 로고
    • XDR Tuberculosis-implications for global public health
    • Raviglione M.C., Smith I.M. (2007) XDR Tuberculosis-implications for global public health. N Engl J Med;356:656-659.
    • (2007) N Engl J Med , vol.356 , pp. 656-659
    • Raviglione, M.C.1    Smith, I.M.2
  • 9
    • 79959225741 scopus 로고    scopus 로고
    • Advent of imidazo[1,2-a]pyridine-3-carboxamides with potent multi- and extended drug resistant antituberculosis activity
    • Moraski G.C., Markley L.D., Hipskind P.A., Boshoff H., Cho S., Franzblau S.G., Miller M.J. (2011) Advent of imidazo[1, 2-a]pyridine-3-carboxamides with potent multi- and extended drug resistant antituberculosis activity. ACS Med Chem Lett;2:466-470.
    • (2011) ACS Med Chem Lett , vol.2 , pp. 466-470
    • Moraski, G.C.1    Markley, L.D.2    Hipskind, P.A.3    Boshoff, H.4    Cho, S.5    Franzblau, S.G.6    Miller, M.J.7
  • 10
    • 80052814263 scopus 로고    scopus 로고
    • Current status and research strategies in tuberculosis drug development
    • Dover L.G., Coxon G.D. (2011) Current status and research strategies in tuberculosis drug development. J Med Chem;54:6157-6165.
    • (2011) J Med Chem , vol.54 , pp. 6157-6165
    • Dover, L.G.1    Coxon, G.D.2
  • 11
    • 79251511858 scopus 로고    scopus 로고
    • Treatment of tuberculosis: update 2010
    • Yew W.W., Lange C., Leung C.C. (2011) Treatment of tuberculosis: update 2010. Eur Respir J;37:441-462.
    • (2011) Eur Respir J , vol.37 , pp. 441-462
    • Yew, W.W.1    Lange, C.2    Leung, C.C.3
  • 12
    • 22544449537 scopus 로고    scopus 로고
    • Recent advances in new structural classes of anti-tuberculosis agents
    • Nayyar A., Jain R. (2005) Recent advances in new structural classes of anti-tuberculosis agents. Curr Med Chem;12:1873-1886.
    • (2005) Curr Med Chem , vol.12 , pp. 1873-1886
    • Nayyar, A.1    Jain, R.2
  • 13
    • 79958784137 scopus 로고    scopus 로고
    • Molecular basis and mechanisms of drug resistance in Mycobacterium tuberculosis: classical and new drugs
    • Da Silva P.E.A., Palomino J.C. (2011) Molecular basis and mechanisms of drug resistance in Mycobacterium tuberculosis: classical and new drugs. J Antimicrob Chemother;66:1417-1430.
    • (2011) J Antimicrob Chemother , vol.66 , pp. 1417-1430
    • Da Silva, P.E.A.1    Palomino, J.C.2
  • 19
    • 0037168055 scopus 로고    scopus 로고
    • Three-dimensional quantitative structure-activity relationship of 1,4-dihydropyridines as antitubercular agents
    • Kharkar P.S., Desai B., Gaveria H., Varu B., Loriya R., Naliapara Y., Shah A., Kulkarni V.M. (2002) Three-dimensional quantitative structure-activity relationship of 1, 4-dihydropyridines as antitubercular agents. J Med Chem;45:4858-4867.
    • (2002) J Med Chem , vol.45 , pp. 4858-4867
    • Kharkar, P.S.1    Desai, B.2    Gaveria, H.3    Varu, B.4    Loriya, R.5    Naliapara, Y.6    Shah, A.7    Kulkarni, V.M.8
  • 20
    • 0034561776 scopus 로고    scopus 로고
    • Synthesis and antitubercular activity of some substituted 3-nitro and 3-bromo-4-hydroxy-2-quinolones
    • Dodia N., Shah A. (2000) Synthesis and antitubercular activity of some substituted 3-nitro and 3-bromo-4-hydroxy-2-quinolones. Indian J Heterocy Ch;10:69-70.
    • (2000) Indian J Heterocy Ch , vol.10 , pp. 69-70
    • Dodia, N.1    Shah, A.2
  • 21
    • 53149115626 scopus 로고    scopus 로고
    • Synthesis, screening for antitubercular activity and 3D-QSAR studies of substituted N-phenyl-6-methyl-2-oxo-4-phenyl-1,2,3,4-tetrahydro-pyrimidine-5-carboxamides
    • Virsodia V., Pissurlenkar R.R.S., Manvar D., Dholakia C., Adlakha P., Shah A., Coutinho E.C. (2008) Synthesis, screening for antitubercular activity and 3D-QSAR studies of substituted N-phenyl-6-methyl-2-oxo-4-phenyl-1, 2, 3, 4-tetrahydro-pyrimidine-5-carboxamides. Eur J Med Chem;43:2103-2115.
    • (2008) Eur J Med Chem , vol.43 , pp. 2103-2115
    • Virsodia, V.1    Pissurlenkar, R.R.S.2    Manvar, D.3    Dholakia, C.4    Adlakha, P.5    Shah, A.6    Coutinho, E.C.7
  • 22
    • 84868101028 scopus 로고    scopus 로고
    • 1,6-Methyl-4-phenyl-5-(phenyl or cycloalkyl) carbamoyl-1,2,3,4-tetrahydropyrimidin-2-one derivatives as antitubercular agents. PCT Int Appl, WO 2011/151701 A1 20111208.
    • Sarkar D., Sarkar S., Joshi R.R., Khedkar V.M., Pissurlenkar R.R., Coutinho E.C., Shah A.K. (2011) 1, 6-Methyl-4-phenyl-5-(phenyl or cycloalkyl) carbamoyl-1, 2, 3, 4-tetrahydropyrimidin-2-one derivatives as antitubercular agents. PCT Int Appl, WO 2011/151701 A1 20111208.
    • (2011)
    • Sarkar, D.1    Sarkar, S.2    Joshi, R.R.3    Khedkar, V.M.4    Pissurlenkar, R.R.5    Coutinho, E.C.6    Shah, A.K.7
  • 23
    • 84868120283 scopus 로고    scopus 로고
    • Preparation of 6-methyl-4-phenyl-5-(phenyl or cyclohexyl)carbamoyl-1,2,3,4-tetrahydropyrimidin-2-one derivatives as antitubercular agents. Indian Pat Appl IN2010DE01244A20120302.
    • Sarkar D., Sarkar S., Joshi R.R., Khedkar V.M., Pissurlenkar R.R., Coutinho E.C., Shah A.K. (2012) Preparation of 6-methyl-4-phenyl-5-(phenyl or cyclohexyl)carbamoyl-1, 2, 3, 4-tetrahydropyrimidin-2-one derivatives as antitubercular agents. Indian Pat Appl IN2010DE01244A20120302.
    • (2012)
    • Sarkar, D.1    Sarkar, S.2    Joshi, R.R.3    Khedkar, V.M.4    Pissurlenkar, R.R.5    Coutinho, E.C.6    Shah, A.K.7
  • 26
    • 2442480580 scopus 로고    scopus 로고
    • Facile one pot microwave induced solvent-free synthesis and antifungal, antitubercular screening of spiro[1,5]-benzothiazepin-2,3'[3'H]indol-2[1'H]-ones
    • Dandia A., Sati M., Arya K., Sharma R., Loupyb A. (2003) Facile one pot microwave induced solvent-free synthesis and antifungal, antitubercular screening of spiro[1, 5]-benzothiazepin-2, 3'[3'H]indol-2[1'H]-ones. Chem Pharm Bull;51:1137-1141.
    • (2003) Chem Pharm Bull , vol.51 , pp. 1137-1141
    • Dandia, A.1    Sati, M.2    Arya, K.3    Sharma, R.4    Loupyb, A.5
  • 27
    • 0032493995 scopus 로고    scopus 로고
    • Synthesis and antimicrobial evaluation of some new fluorinated spiro[[1,5]-benzothiazepin-2,3'[3'H]-indol]-2'(1'H)-ones
    • Dandia A., Upreti M., Rani B., Pant U.C., Gupta I.J. (1998) Synthesis and antimicrobial evaluation of some new fluorinated spiro[[1, 5]-benzothiazepin-2, 3'[3'H]-indol]-2'(1'H)-ones. J Fluorine Chem;91:171-174.
    • (1998) J Fluorine Chem , vol.91 , pp. 171-174
    • Dandia, A.1    Upreti, M.2    Rani, B.3    Pant, U.C.4    Gupta, I.J.5
  • 28
    • 33846641698 scopus 로고    scopus 로고
    • Solid-phase synthesis of a library of pyrrolo[2,1-c][1,4]benzodiazepine-5,11-diones with potential antitubercular activity
    • Kamal A., Reddy K.L., Devaiah V., Shankaraiah N., Reddy G.S.K., Raghvan S. (2007) Solid-phase synthesis of a library of pyrrolo[2, 1-c][1, 4]benzodiazepine-5, 11-diones with potential antitubercular activity. J Comb Chem;9:29-42.
    • (2007) J Comb Chem , vol.9 , pp. 29-42
    • Kamal, A.1    Reddy, K.L.2    Devaiah, V.3    Shankaraiah, N.4    Reddy, G.S.K.5    Raghvan, S.6
  • 31
    • 8944259902 scopus 로고    scopus 로고
    • Cardiovascular characterization of pyrrolo[2,1-d][1,5]benzothiazepines derivatives binding selectively to the peripheral-type benzodiazepine receptor (PBR): from dual PBR affinity and calcium antagonist activity to novel and selective calcium entry blockers
    • Campiani G., Fiorini I., De Filippis M.P., Ciani S.M., Garofalo A., Nacci V., Giorgi G., Sega A., Botta M., Chiarini A., Budriesi R., Bruni G., Romeo M.R., Manzoni C., Mennini T. (1996) Cardiovascular characterization of pyrrolo[2, 1-d][1, 5]benzothiazepines derivatives binding selectively to the peripheral-type benzodiazepine receptor (PBR): from dual PBR affinity and calcium antagonist activity to novel and selective calcium entry blockers. J Med Chem;39:2933-2938.
    • (1996) J Med Chem , vol.39 , pp. 2933-2938
    • Campiani, G.1    Fiorini, I.2    De Filippis, M.P.3    Ciani, S.M.4    Garofalo, A.5    Nacci, V.6    Giorgi, G.7    Sega, A.8    Botta, M.9    Chiarini, A.10    Budriesi, R.11    Bruni, G.12    Romeo, M.R.13    Manzoni, C.14    Mennini, T.15
  • 34
    • 0037368532 scopus 로고    scopus 로고
    • Synthesis of pyrazoline, pyrimidine and 1,5-benzodiazepine derivatives of 1,8-naphthyridine and evaluation of antibacterial activity
    • Mogilaih K., Sudhakar G.R. (2003) Synthesis of pyrazoline, pyrimidine and 1, 5-benzodiazepine derivatives of 1, 8-naphthyridine and evaluation of antibacterial activity. Indian J Chem;42B:636-640.
    • (2003) Indian J Chem , vol.42 B , pp. 636-640
    • Mogilaih, K.1    Sudhakar, G.R.2
  • 35
    • 77952773228 scopus 로고    scopus 로고
    • Synthesis of pyrazoline, pyrimidine and 1,5-benzodiazepine derivatives of 1,8-naphthyridine and evaluation of antibacterial activity
    • Kumar P.V., Rao V.R. (2008) Synthesis of pyrazoline, pyrimidine and 1, 5-benzodiazepine derivatives of 1, 8-naphthyridine and evaluation of antibacterial activity. Indian J Chem;47B:106-111.
    • (2008) Indian J Chem , vol.47 B , pp. 106-111
    • Kumar, P.V.1    Rao, V.R.2
  • 36
    • 82955178707 scopus 로고    scopus 로고
    • Synthesis and in vitro antimycobacterial activity of fluoroquinolone derivatives containing a coumarin moiety
    • Guo Q., Liu M.-L., Feng L.-S., Lv K., Guan G., Guo H.-Y., Xiao C.-L. (2011) Synthesis and in vitro antimycobacterial activity of fluoroquinolone derivatives containing a coumarin moiety. Arch Pharm Chem Life Sci;344:802-809.
    • (2011) Arch Pharm Chem Life Sci , vol.344 , pp. 802-809
    • Guo, Q.1    Liu, M.-L.2    Feng, L.-S.3    Lv, K.4    Guan, G.5    Guo, H.-Y.6    Xiao, C.-L.7
  • 38
    • 33846096215 scopus 로고
    • The reaction of 3-acyl-4-hydroxycoumarins with ammonium salts
    • Kloss R.A., Wiener C. (1963) The reaction of 3-acyl-4-hydroxycoumarins with ammonium salts. J Org Chem;28:1671-1673.
    • (1963) J Org Chem , vol.28 , pp. 1671-1673
    • Kloss, R.A.1    Wiener, C.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.