SCOPUS 정보 검색 플랫폼

Volumn 3, Issue 9, 2012, Pages 1164-1169

A matched molecular pair analysis of in vitro human microsomal metabolic stability measurements for heterocyclic replacements of di-substituted benzene containing compounds - Identification of those isosteres more likely to have beneficial effects

(3) Dossetter, Alexander G a Douglas, Adam a O'Donnell, Charles a

a ASTRAZENECA (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

1,2,4 OXADIAZOLE DERIVATIVE; 1,3,4 OXADIAZOLE DERIVATIVE; BENZENE DERIVATIVE; FURAN DERIVATIVE; HETEROCYCLIC COMPOUND; IMIDAZOLE DERIVATIVE; ISOSTERE DERIVATIVE; ISOXAZOLE DERIVATIVE; OXAZOLE DERIVATIVE; PIPERAZINE DERIVATIVE; PYRAZINE DERIVATIVE; PYRAZOLE DERIVATIVE; PYRIDINE DERIVATIVE; PYRIMIDINE DERIVATIVE; THIAZOLE DERIVATIVE; THIOPHENE DERIVATIVE; TRIAZINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL ANALYSIS; CHEMICAL STRUCTURE; CHEMISTRY; CONTROLLED STUDY; HUMAN; IN VITRO STUDY; MEDICINAL CHEMISTRY; METABOLISM; MICROSOME; PRIORITY JOURNAL;

EID: 84865518339 PISSN: 20402503 EISSN: 20402511 Source Type: Journal
DOI: 10.1039/c2md20155k Document Type: Article

Times cited : (18)

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