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Volumn 3, Issue 5, 2012, Pages 600-604

Oxadiazole isomers: All bioisosteres are not created equal

(10) Goldberg, Kristin a Groombridge, Sam a Hudson, Julian a Leach, Andrew G a MacFaul, Philip A a Pickup, Adrian a Poultney, Ruth a Scott, James S a Svensson, Per H b,c Sweeney, Joseph d

a ASTRAZENECA (United Kingdom)

b ASTRAZENECA R AND D (Sweden)

c ROYAL INSTITUTE OF TECHNOLOGY (Sweden)

d UNIVERSITY OF HUDDERSFIELD (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

1,2,4 OXADIAZOLE DERIVATIVE; 1,3,4 OXADIAZOLE DERIVATIVE;

ARTICLE; DRUG HALF LIFE; DRUG PROTEIN BINDING; DRUG SOLUBILITY; DRUG STABILITY; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN; HYDROGEN BOND; ISOMER; LIPOPHILICITY; MOUSE; NONHUMAN; PLASMA PROTEIN BINDING; PRIORITY JOURNAL; RAT; STRUCTURE ANALYSIS; SUBSTITUTION REACTION;

EID: 84860429692 PISSN: 20402503 EISSN: 20402511 Source Type: Journal
DOI: 10.1039/c2md20054f Document Type: Article

Times cited : (34)

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