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Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 18, 2012, Pages 5889-5892

Biologically active ester derivatives as potent inhibitors of the soluble epoxide hydrolase

(7) Kim, In Hae a,b Nishi, Kosuke a,b Kasagami, Takeo a,c Morisseau, Christophe a Liu, Jun Yan a Tsai, Hsing Ju a Hammock, Bruce D a

a UNIVERSITY OF CALIFORNIA (United States)

b EHIME UNIVERSITY (Japan)

c LSI MEDIENCE CORPORATION (Japan)

Author keywords

Metabolic stability; sEH; sEH inhibitors; Substituted urea ester derivatives

Indexed keywords

EPOXIDE HYDROLASE; ESTER DERIVATIVE;

ARTICLE; CHEMICAL MODIFICATION; DRUG ACTIVITY; DRUG POTENCY; DRUG SCREENING; DRUG STABILITY; DRUG SYNTHESIS; ENZYME INHIBITION; HUMAN; HUMAN CELL; IN VITRO STUDY; LIVER MICROSOME; PHYSICAL CHEMISTRY;

DOSE-RESPONSE RELATIONSHIP, DRUG; ENZYME INHIBITORS; EPOXIDE HYDROLASES; ESTERS; HUMANS; MICROSOMES, LIVER; MOLECULAR STRUCTURE; SOLUBILITY; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84865517379 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2012.07.074 Document Type: Article

Times cited : (10)

References (30)

1
- 0033993749
- J.H. Capdevila, J.R. Falck, and R.C. Harris J. Lipid Res. 41 2000 163
- (2000) J. Lipid Res. , vol.41 , pp. 163
- Capdevila, J.H.¹ Falck, J.R.² Harris, R.C.³

2
- 0034711488
- Z. Yu, F. Xu, L.M. Huse, C. Morisseau, A.J. Draper, J.W. Newman, C. Parker, L. Graham, M.M. Engler, B.D. Hammock, D.C. Zeldin, and D.L. Kroetz Circ. Res. 87 2000 992
- (2000) Circ. Res. , vol.87 , pp. 992
- Yu, Z.¹ Xu, F.² Huse, L.M.³ Morisseau, C.⁴ Draper, A.J.⁵ Newman, J.W.⁶ Parker, C.⁷ Graham, L.⁸ Engler, M.M.⁹ Hammock, B.D.¹⁰ Zeldin, D.C.¹¹ Kroetz, D.L.¹²

3
- 0036179501
- J.D. Imig, X. Zhao, J.H. Capdevila, C. Morisseau, and B.D. Hammock Hypertension 39 2002 690
- (2002) Hypertension , vol.39 , pp. 690
- Imig, J.D.¹ Zhao, X.² Capdevila, J.H.³ Morisseau, C.⁴ Hammock, B.D.⁵

4
- 11144356945
- X. Zhao, T. Yamamoto, J.W. Newman, I.-H. Kim, T. Watanabe, B.D. Hammock, J. Stewart, J.S. Pollock, D.M. Pollock, and J.D. Imig J. Am. Soc. Nephrol. 15 2004 1244
- (2004) J. Am. Soc. Nephrol. , vol.15 , pp. 1244
- Zhao, X.¹ Yamamoto, T.² Newman, J.W.³ Kim, I.-H.⁴ Watanabe, T.⁵ Hammock, B.D.⁶ Stewart, J.⁷ Pollock, J.S.⁸ Pollock, D.M.⁹ Imig, J.D.¹⁰

5
- 15744382006
- O. Jung, R.P. Brandes, I.H. Kim, F. Schweda, R. Schmidt, B.D. Hammock, R. Busse, and I. Fleming Hypertension 45 2005 759
- (2005) Hypertension , vol.45 , pp. 759
- Jung, O.¹ Brandes, R.P.² Kim, I.H.³ Schweda, F.⁴ Schmidt, R.⁵ Hammock, B.D.⁶ Busse, R.⁷ Fleming, I.⁸

6
- 33644654633
- J.D. Imig, X. Zhao, C.Z. Zaharis, J.J. Olearczyk, D.M. Pollock, J.W. Newman, I.H. Kim, T. Watanabe, and B.D. Hammock Hypertension 46 2006 975
- (2006) Hypertension , vol.46 , pp. 975
- Imig, J.D.¹ Zhao, X.² Zaharis, C.Z.³ Olearczyk, J.J.⁴ Pollock, D.M.⁵ Newman, J.W.⁶ Kim, I.H.⁷ Watanabe, T.⁸ Hammock, B.D.⁹

7
- 13844315294
- K.R. Smith, K.E. Pinkerton, T. Watanabe, T.L. Pedersen, S.J. Ma, and B.D. Hammock Proc. Natl. Acad. Sci. U.S.A. 102 2005 2186
- (2005) Proc. Natl. Acad. Sci. U.S.A. , vol.102 , pp. 2186
- Smith, K.R.¹ Pinkerton, K.E.² Watanabe, T.³ Pedersen, T.L.⁴ Ma, S.J.⁵ Hammock, B.D.⁶

8
- 22244443733
- K.R. Schmelzer, L. Kubala, J.W. Newman, I.H. Kim, J.P. Eiserich, and B.D. Hammock Proc. Natl. Acad. Sci. U.S.A. 102 2005 9772
- (2005) Proc. Natl. Acad. Sci. U.S.A. , vol.102 , pp. 9772
- Schmelzer, K.R.¹ Kubala, L.² Newman, J.W.³ Kim, I.H.⁴ Eiserich, J.P.⁵ Hammock, B.D.⁶

9
- 0033588034
- K. Node, Y. Huo, X. Ruan, B. Yang, M. Spiecker, K. Ley, D.C. Zeldin, and J.K. Liao Science 285 1999 1276
- (1999) Science , vol.285 , pp. 1276
- Node, K.¹ Huo, Y.² Ruan, X.³ Yang, B.⁴ Spiecker, M.⁵ Ley, K.⁶ Zeldin, D.C.⁷ Liao, J.K.⁸

10
- 0034176077
- W.B. Campbell Trends Pharmacol. Sci. 21 2000 125
- (2000) Trends Pharmacol. Sci. , vol.21 , pp. 125
- Campbell, W.B.¹

11
- 0034923447
- B. Yang, L. Graham, S. Dikalov, R.P. Mason, J.R. Falck, J.K. Liao, and D.C. Zeldin Mol. Pharmacol. 60 2001 310
- (2001) Mol. Pharmacol. , vol.60 , pp. 310
- Yang, B.¹ Graham, L.² Dikalov, S.³ Mason, R.P.⁴ Falck, J.R.⁵ Liao, J.K.⁶ Zeldin, D.C.⁷

12
- 0035844126
- K. Node, X. Ruan, J. Dai, S. Yang, L. Graham, D.C. Zeldin, and J.K. Liao J. Biol. Chem. 276 2001 15983
- (2001) J. Biol. Chem. , vol.276 , pp. 15983
- Node, K.¹ Ruan, X.² Dai, J.³ Yang, S.⁴ Graham, L.⁵ Zeldin, D.C.⁶ Liao, J.K.⁷

13
- 33845474465
- D. Xu, N. Li, Y. He, V. Timofeyev, L. Lu, H.-J. Tsai, I.H. Kim, D. Tuteja, R.K.P. Mateo, A. Singapuri, B.B. Davis, R. Low, B.D. Hammock, and N. Chiamvimonvat Proc. Natl. Acad. Sci. U.S.A. 103 2006 18733
- (2006) Proc. Natl. Acad. Sci. U.S.A. , vol.103 , pp. 18733
- Xu, D.¹ Li, N.² He, Y.³ Timofeyev, V.⁴ Lu, L.⁵ Tsai, H.-J.⁶ Kim, I.H.⁷ Tuteja, D.⁸ Mateo, R.K.P.⁹ Singapuri, A.¹⁰ Davis, B.B.¹¹ Low, R.¹² Hammock, B.D.¹³ Chiamvimonvat, N.¹⁴

14
- 79953177021
- B. Inceoglu, K. Wagner, N.H. Schebb, C. Morisseau, S.L. Jinks, A. Ulu, C. Hegedus, T. Rose, R. Brosnan, and B.D. Hammock Proc. Natl. Acad. Sci. U.S.A. 108 2011 5093
- (2011) Proc. Natl. Acad. Sci. U.S.A. , vol.108 , pp. 5093
- Inceoglu, B.¹ Wagner, K.² Schebb, N.H.³ Morisseau, C.⁴ Jinks, S.L.⁵ Ulu, A.⁶ Hegedus, C.⁷ Rose, T.⁸ Brosnan, R.⁹ Hammock, B.D.¹⁰

15
- 0031004964
- M.F. Moghaddam, D.F. Grant, J.M. Cheek, J.F. Greene, K.C. Williamson, and B.D. Hammock Nat. Med. 3 1997 562
- (1997) Nat. Med. , vol.3 , pp. 562
- Moghaddam, M.F.¹ Grant, D.F.² Cheek, J.M.³ Greene, J.F.⁴ Williamson, K.C.⁵ Hammock, B.D.⁶

16
- 0035150448
- J.W. Newman, D.L. Denton, C. Morisseau, C.S. Koger, C.E. Wheelock, D.E. Hinton, and B.D. Hammock Environ. Health Perspect. 109 2001 61
- (2001) Environ. Health Perspect. , vol.109 , pp. 61
- Newman, J.W.¹ Denton, D.L.² Morisseau, C.³ Koger, C.S.⁴ Wheelock, C.E.⁵ Hinton, D.E.⁶ Hammock, B.D.⁷

17
- 0036570198
- C. Morisseau, M.H. Goodrow, J.W. Newman, C.E. Wheelock, D.L. Dowdy, and B.D. Hammock Biochem. Pharmacol. 63 2002 1599
- (2002) Biochem. Pharmacol. , vol.63 , pp. 1599
- Morisseau, C.¹ Goodrow, M.H.² Newman, J.W.³ Wheelock, C.E.⁴ Dowdy, D.L.⁵ Hammock, B.D.⁶

18
- 1842555060
- I.H. Kim, C. Morisseau, T. Watanabe, and B.D. Hammock J. Med. Chem. 47 2004 2110
- (2004) J. Med. Chem. , vol.47 , pp. 2110
- Kim, I.H.¹ Morisseau, C.² Watanabe, T.³ Hammock, B.D.⁴

19
- 18644374475
- I.H. Kim, F.R. Heirtzler, C. Morisseau, K. Nishi, H.J. Tsai, and B.D. Hammock J. Med. Chem. 48 2005 3621
- (2005) J. Med. Chem. , vol.48 , pp. 3621
- Kim, I.H.¹ Heirtzler, F.R.² Morisseau, C.³ Nishi, K.⁴ Tsai, H.J.⁵ Hammock, B.D.⁶

20
- 33750949953
- I.H. Kim, K. Nishi, H.-J. Tsai, T. Bradford, Y. Koda, T. Watanabe, C. Morisseau, J. Blanchfield, I. Toth, and B.D. Hammock Bioorg. Med. Chem. 15 2007 312
- (2007) Bioorg. Med. Chem. , vol.15 , pp. 312
- Kim, I.H.¹ Nishi, K.² Tsai, H.-J.³ Bradford, T.⁴ Koda, Y.⁵ Watanabe, T.⁶ Morisseau, C.⁷ Blanchfield, J.⁸ Toth, I.⁹ Hammock, B.D.¹⁰

21
- 35348826197
- I.H. Kim, H.-J. Tsai, K. Nishi, T. Kasagami, C. Morisseau, and B.D. Hammock J. Med. Chem. 50 2007 5217
- (2007) J. Med. Chem. , vol.50 , pp. 5217
- Kim, I.H.¹ Tsai, H.-J.² Nishi, K.³ Kasagami, T.⁴ Morisseau, C.⁵ Hammock, B.D.⁶

22
- 61349106718
- T. Kasagami, I.H. Kim, H.-J. Tsai, K. Nishi, B.D. Hammock, and C. Morisseau Bioorg. Med. Chem. Lett. 19 2009 1784
- (2009) Bioorg. Med. Chem. Lett. , vol.19 , pp. 1784
- Kasagami, T.¹ Kim, I.H.² Tsai, H.-J.³ Nishi, K.⁴ Hammock, B.D.⁵ Morisseau, C.⁶

23
- 79952794917
- I.H. Kim, Y.K. Park, B.D. Hammock, and K. Nishi J. Med. Chem. 54 2011 1752
- (2011) J. Med. Chem. , vol.54 , pp. 1752
- Kim, I.H.¹ Park, Y.K.² Hammock, B.D.³ Nishi, K.⁴

24
- 77950864854
- S.-K. Anandan, and R.D. Gless Bioorg. Med. Chem. Lett. 20 2010 2740
- (2010) Bioorg. Med. Chem. Lett. , vol.20 , pp. 2740
- Anandan, S.-K.¹ Gless, R.D.²

25
- 66349134398
- H.C. Shen, F.-X. Ding, S. Wang, S. Xu, H.-S. Chen, X. Tong, V. Tong, K. Mitra, S. Kumar, X. Zhang, Y. Chen, G. Zhou, L.-Y. Pai, M. Alonso-Galicia, X. Chen, B. Zhang, J.R. Tata, J.P. Berger, and S. Colletti Bioorg. Med. Chem. Lett. 19 2009 3398
- (2009) Bioorg. Med. Chem. Lett. , vol.19 , pp. 3398
- Shen, H.C.¹ Ding, F.-X.² Wang, S.³ Xu, S.⁴ Chen, H.-S.⁵ Tong, X.⁶ Tong, V.⁷ Mitra, K.⁸ Kumar, S.⁹ Zhang, X.¹⁰ Chen, Y.¹¹ Zhou, G.¹² Pai, L.-Y.¹³ Alonso-Galicia, M.¹⁴ Chen, X.¹⁵ Zhang, B.¹⁶ Tata, J.R.¹⁷ Berger, J.P.¹⁸ Colletti, S.¹⁹

26
- 84865451537
- 2nd ed. Elsevier Academic Press
- B.S. Richard The Organic Chemistry of Drug Design and Drug Action 2nd ed. 2004 Elsevier Academic Press pp 471-473
- (2004) The Organic Chemistry of Drug Design and Drug Action
- Richard, B.S.¹

27
- 34548070313
- S.H. Hwang, H.-J. Tsai, J.-Y. Liu, C. Morisseau, and B.D. Hammock J. Med. Chem. 50 2007 3825
- (2007) J. Med. Chem. , vol.50 , pp. 3825
- Hwang, S.H.¹ Tsai, H.-J.² Liu, J.-Y.³ Morisseau, C.⁴ Hammock, B.D.⁵

28
- 84857740699
- S. Pillarisetti, and I. Khanna Inflamm. Allergy Drug Targets 11 2012 143
- (2012) Inflamm. Allergy Drug Targets , vol.11 , pp. 143
- Pillarisetti, S.¹ Khanna, I.²

29
- 49249116223
- G.J. Gross, K.M. Gauthier, J. Moore, J.R. Falck, B.D. Hammock, W.B. Campbell, and K. Nithipatikom Am. J. Physiol. Heart Circ. Physiol. 294 2008 H2838
- (2008) Am. J. Physiol. Heart Circ. Physiol. , vol.294 , pp. 2838
- Gross, G.J.¹ Gauthier, K.M.² Moore, J.³ Falck, J.R.⁴ Hammock, B.D.⁵ Campbell, W.B.⁶ Nithipatikom, K.⁷

30
- 84858032383
- H. Shen, and B.D. Hammock J. Med. Chem. 55 2012 1789
- (2012) J. Med. Chem. , vol.55 , pp. 1789
- Shen, H.¹ Hammock, B.D.²

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