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Volumn 80, Issue 2, 2012, Pages 340-347

Antimalarial Activity of Newly Synthesized Chalcone Derivatives In Vitro

Author keywords

Antimalarial activity; Chalcone synthesis; in vitro; Plasmodium falciparum

Indexed keywords

1 (4 BENZIMIDAZOL 1 YLPHENYL) 3 (2,4 DIMETHOXYPHENYL)PROPEN 1 ONE; ANTIMALARIAL AGENT; CHALCONE DERIVATIVE; CYSTEINE PROTEINASE; FUNCTIONAL GROUP; LICOCHALCONE A; UNCLASSIFIED DRUG;

EID: 84864013231     PISSN: 17470277     EISSN: 17470285     Source Type: Journal    
DOI: 10.1111/j.1747-0285.2012.01383.x     Document Type: Review
Times cited : (125)

References (23)
  • 1
    • 0035139250 scopus 로고    scopus 로고
    • Current status of malaria and potential for control
    • Phillips R.S. (2001) Current status of malaria and potential for control. Clin Microbiol Rev;14:208-226.
    • (2001) Clin Microbiol Rev , vol.14 , pp. 208-226
    • Phillips, R.S.1
  • 2
    • 2442507656 scopus 로고    scopus 로고
    • Antibacterial chalcones - bioisosteric replacement of the 4′-hydroxy group
    • Nielsen S.F., Bosen T., Larsen M., Schonning K., Kromann H. (2004) Antibacterial chalcones - bioisosteric replacement of the 4′-hydroxy group. Bioorg Med Chem;12:3047-3054.
    • (2004) Bioorg Med Chem , vol.12 , pp. 3047-3054
    • Nielsen, S.F.1    Bosen, T.2    Larsen, M.3    Schonning, K.4    Kromann, H.5
  • 3
    • 17144427687 scopus 로고    scopus 로고
    • Cationic chalcone antibiotics: design, synthesis, and mechanism of action
    • Nielsen S.F., Larsen M., Bosen T., Schonning K., Kromann H. (2005) Cationic chalcone antibiotics: design, synthesis, and mechanism of action. J Med Chem;48:2667-2677.
    • (2005) J Med Chem , vol.48 , pp. 2667-2677
    • Nielsen, S.F.1    Larsen, M.2    Bosen, T.3    Schonning, K.4    Kromann, H.5
  • 4
    • 66149110763 scopus 로고    scopus 로고
    • Antifilarial activity of 1, 3-diarylpropen-1-one: effect on glutathione-S-transferase, a phase II detoxification enzyme
    • Awasthi S.K., Mishra N., Dixit S.K., Singh A., Yadav M., Yadav S.S., Rathaur S. (2009) Antifilarial activity of 1, 3-diarylpropen-1-one: effect on glutathione-S-transferase, a phase II detoxification enzyme. Am J Trop Med Hyg;80:764-768.
    • (2009) Am J Trop Med Hyg , vol.80 , pp. 764-768
    • Awasthi, S.K.1    Mishra, N.2    Dixit, S.K.3    Singh, A.4    Yadav, M.5    Yadav, S.S.6    Rathaur, S.7
  • 7
    • 0038548308 scopus 로고    scopus 로고
    • Structure-activity relationships of antileishmanial and antimalarial chalcones
    • Liu M., Wilairat P., Croft S.L., Tan A.L., Go M.L. (2003) Structure-activity relationships of antileishmanial and antimalarial chalcones. Bioorg Med Chem;11:2729-2738.
    • (2003) Bioorg Med Chem , vol.11 , pp. 2729-2738
    • Liu, M.1    Wilairat, P.2    Croft, S.L.3    Tan, A.L.4    Go, M.L.5
  • 9
    • 2142640813 scopus 로고    scopus 로고
    • Differential effects of synthesized 2′-oxygenated chalcone derivatives: modulation of human cell cycle phase distribution
    • Rao Y.K., Fang F.S., Tzeng Y.M. (2004) Differential effects of synthesized 2′-oxygenated chalcone derivatives: modulation of human cell cycle phase distribution. Bioorg Med Chem;122:2679-2686.
    • (2004) Bioorg Med Chem , vol.122 , pp. 2679-2686
    • Rao, Y.K.1    Fang, F.S.2    Tzeng, Y.M.3
  • 10
    • 0028357495 scopus 로고
    • Licochalcone A, a new antimalarial agent, inhibits in vitro growth of the human malaria parasite Plasmodium falciparum and protects mice from P. yoelii infection
    • Chen M., Theander T.G., Christensen B.S., Hviid I., Zhai L., Kharazmi A. (1994) Licochalcone A, a new antimalarial agent, inhibits in vitro growth of the human malaria parasite Plasmodium falciparum and protects mice from P. yoelii infection. Antimicrob Agents Chemother;38:1470-1475.
    • (1994) Antimicrob Agents Chemother , vol.38 , pp. 1470-1475
    • Chen, M.1    Theander, T.G.2    Christensen, B.S.3    Hviid, I.4    Zhai, L.5    Kharazmi, A.6
  • 11
    • 45849124658 scopus 로고    scopus 로고
    • Synthesis of novel substituted 1,3-diaryl propenone derivatives and their antimalarial activity in vitro
    • Mishra N., Arora P., Kumar B., Mishra L.C., Bhattacharya A., Awasthi S.K., Bhasin V.K. (2008) Synthesis of novel substituted 1, 3-diaryl propenone derivatives and their antimalarial activity in vitro. Eur J Med Chem;43:1530-1535.
    • (2008) Eur J Med Chem , vol.43 , pp. 1530-1535
    • Mishra, N.1    Arora, P.2    Kumar, B.3    Mishra, L.C.4    Bhattacharya, A.5    Awasthi, S.K.6    Bhasin, V.K.7
  • 12
    • 59049101538 scopus 로고    scopus 로고
    • Phytochemical licochalcone A enhances antimalarial activity of artemisinin in vitro
    • Mishra L.C., Bhattacharya A., Bhasin V.K. (2009) Phytochemical licochalcone A enhances antimalarial activity of artemisinin in vitro. Acta Trop;109:194-198.
    • (2009) Acta Trop , vol.109 , pp. 194-198
    • Mishra, L.C.1    Bhattacharya, A.2    Bhasin, V.K.3
  • 15
    • 10444280081 scopus 로고    scopus 로고
    • Chalcones as potent tyrosinase inhibitors: the importance of a 2, 4-substituted resorcinol moiety
    • Khatib S., Nerya O., Musa R., Shmuel M., Tamir S., Vaya J. (2005) Chalcones as potent tyrosinase inhibitors: the importance of a 2, 4-substituted resorcinol moiety. Bioorg Med Chem;13:433-441.
    • (2005) Bioorg Med Chem , vol.13 , pp. 433-441
    • Khatib, S.1    Nerya, O.2    Musa, R.3    Shmuel, M.4    Tamir, S.5    Vaya, J.6
  • 16
    • 0017311840 scopus 로고
    • Human malaria parasites in continuous culture
    • Trager W., Jensen J.B. (1976) Human malaria parasites in continuous culture. Science;193:673-675.
    • (1976) Science , vol.193 , pp. 673-675
    • Trager, W.1    Jensen, J.B.2
  • 17
    • 67650456777 scopus 로고    scopus 로고
    • Antimalarial pharmacodynamics of chalcone derivatives in combination with artemisinin against Plasmodium falciparum in vitro
    • Bhattacharya A., Mishra L.C., Sharma M., Awasthi S.K., Bhasin V.K. (2009) Antimalarial pharmacodynamics of chalcone derivatives in combination with artemisinin against Plasmodium falciparum in vitro. Eur J Med Chem;44:3388-3393.
    • (2009) Eur J Med Chem , vol.44 , pp. 3388-3393
    • Bhattacharya, A.1    Mishra, L.C.2    Sharma, M.3    Awasthi, S.K.4    Bhasin, V.K.5
  • 18
    • 0018704491 scopus 로고
    • Synchronization of Plasmodium falciparum erythrocytic stages in culture
    • Lambros C., Vanderberg J.P. (1979) Synchronization of Plasmodium falciparum erythrocytic stages in culture. J Parasitol;65:418-420.
    • (1979) J Parasitol , vol.65 , pp. 418-420
    • Lambros, C.1    Vanderberg, J.P.2
  • 19
    • 0019164230 scopus 로고
    • Pyrimethamine sensitivity in Plasmodium falciparum: determination in vitro by a modified 48-hour test
    • Nguyen-Dinh P., Payne D. (1980) Pyrimethamine sensitivity in Plasmodium falciparum: determination in vitro by a modified 48-hour test. Bull World Health Organ;58:909-912.
    • (1980) Bull World Health Organ , vol.58 , pp. 909-912
    • Nguyen-Dinh, P.1    Payne, D.2
  • 20
    • 0029013807 scopus 로고
    • The Plasmodium digestive vacuole: metabolic headquarters and choice drug target
    • Olliaro P.L., Goldberg D.E. (1995) The Plasmodium digestive vacuole: metabolic headquarters and choice drug target. Parasitol Today;11:294-297.
    • (1995) Parasitol Today , vol.11 , pp. 294-297
    • Olliaro, P.L.1    Goldberg, D.E.2
  • 21
    • 0001402353 scopus 로고    scopus 로고
    • Cysteine proteinase inhibitors block early steps in hemoglobin degradation by cultured malaria parasites
    • Gamboa de Dominguez N.D., Rosenthal P.J. (1996) Cysteine proteinase inhibitors block early steps in hemoglobin degradation by cultured malaria parasites. Blood;87:4448-4454.
    • (1996) Blood , vol.87 , pp. 4448-4454
    • Gamboa de Dominguez, N.D.1    Rosenthal, P.J.2
  • 22
    • 0030879653 scopus 로고    scopus 로고
    • Hemoglobin metabolism in the malaria parasite, Plasmodium falciparum
    • Francis S.E., Sullivan D.J., Goldberg D.E. (1997) Hemoglobin metabolism in the malaria parasite, Plasmodium falciparum. Annu Rev Microbiol;51:97-123.
    • (1997) Annu Rev Microbiol , vol.51 , pp. 97-123
    • Francis, S.E.1    Sullivan, D.J.2    Goldberg, D.E.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.