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Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 15, 2012, Pages 5025-5030

Design, synthesis, modeling, biological evaluation and photoaffinity labeling studies of novel series of photoreactive benzamide probes for histone deacetylase 2

(7) Vaidya, Aditya Sudheer a Karumudi, Bhargava a Mendonca, Emma b Madriaga, Antonett a Abdelkarim, Hazem a Van Breemen, Richard B a Petukhov, Pavel A a

a UNIVERSITY OF ILLINOIS AT CHICAGO (United States)

b University of Illinois at Chicago (United States)

Author keywords

Benzamides; Diazides; HDAC 1 and 2; Photoaffinity labeling; Time dependent inhibition

Indexed keywords

BENZAMIDE DERIVATIVE; HISTONE DEACETYLASE 1; HISTONE DEACETYLASE 2;

ARTICLE; DRUG ACTIVITY; DRUG DESIGN; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION; HUMAN; MOLECULAR PROBE; NONHUMAN; PHOTOAFFINITY LABELING; STRUCTURE ACTIVITY RELATION;

AFFINITY LABELS; BENZAMIDES; BIOTIN; CATALYTIC DOMAIN; CELL LINE, TUMOR; DRUG DESIGN; HISTONE DEACETYLASE 1; HISTONE DEACETYLASE 2; HISTONE DEACETYLASE INHIBITORS; HUMANS; MODELS, MOLECULAR; PROTEIN BINDING; PROTEIN ISOFORMS;

EID: 84863983721 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2012.06.017 Document Type: Article

Times cited : (14)

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