The pharmacological profile of ELIC, a prokaryotic GABA-gated receptor

Neuropharmacology

Volumn 63, Issue 4, 2012, Pages 761-767

  Thompson, Andrew J ^a   Alqazzaz, Mona ^a   Ulens, Chris ^b   Lummis, Sarah C R ^a  

^a UNIVERSITY OF CAMBRIDGE   (United Kingdom)

^b LABORATORY OF MOLECULAR AND CELLULAR SIGNALING   (Belgium)

Author keywords

Antagonist; Cys loop; ELIC; Erwinia; GABA; GLIC; Ligand gated; Nicotinic

Indexed keywords

2 AMINOBUTYRIC ACID; 2 OXOGLUTARIC ACID; 4 AMINOBUTYRIC ACID A RECEPTOR STIMULATING AGENT; 4 AMINOBUTYRIC ACID RECEPTOR; 4 HYDROXYBUTYRIC ACID; 5 AMINOVALERIC ACID; CYSTEINE; DIELDRIN; ENDOSULFAN; ERWINIA LIGAND GATED ION CHANNEL; GAMMA BUTYROLACTONE; GLUTAMIC ACID; LIGAND GATED ION CHANNEL; PICROTOXININ; PYROGLUTAMIC ACID; SUCCINIC ACID; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CHANNEL GATING; CONTROLLED STUDY; CRYSTAL STRUCTURE; MOLECULAR INTERACTION; MUTAGENESIS; NONHUMAN; PRIORITY JOURNAL; RECEPTOR BLOCKING; RECEPTOR UPREGULATION; XENOPUS LAEVIS;

AMINO ACID SEQUENCE; ANIMALS; BACTERIAL PROTEINS; CELLS, CULTURED; COMPUTER SIMULATION; DATABASES, PROTEIN; ERWINIA; FEMALE; GABA AGONISTS; GABA ANTAGONISTS; GAMMA-AMINOBUTYRIC ACID; KINETICS; LIGAND-GATED ION CHANNELS; LIGANDS; MOLECULAR SEQUENCE DATA; MUTANT PROTEINS; PATCH-CLAMP TECHNIQUES; PROTEIN BINDING; PROTEIN CONFORMATION; RECOMBINANT PROTEINS; SEQUENCE ALIGNMENT; XENOPUS LAEVIS;

EID: 84863629046     PISSN: 00283908     EISSN: 18737064     Source Type: Journal    
DOI: 10.1016/j.neuropharm.2012.05.027     Document Type: Article

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