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Volumn 7, Issue 2, 2012, Pages 223-228

Design, Synthesis and Biological Evaluation of Noncovalent Inhibitors of Human CD38 NADase

(10) Zhou, Yi a Ting, Kai Yiu b Lam, Connie Mo Ching b Kwong, Anna Ka Yee b Xia, Jie a Jin, Hongwei a Liu, Zhenming a Zhang, Liangren a CheungLee, Hon b Zhang, Lihe a

a PEKING UNIVERSITY HEALTH SCIENCE CENTER (China)

b UNIVERSITY OF HONG KONG (Hong Kong)

Author keywords

Calcium ion messengers; CD38; Noncovalent inhibitors; Structure activity relationships

Indexed keywords

CD38 NICOTINAMIDE ADENINE DINUCLEOTIDE NUCLEOSIDASE INHIBITOR; ENZYME INHIBITOR; UNCLASSIFIED DRUG;

ARTICLE; DRUG ACTIVITY; DRUG BINDING; DRUG DESIGN; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; EVALUATION; HUMAN; HYDROGEN BOND; IC 50; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION;

ANTIGENS, CD38; BINDING SITES; CATALYTIC DOMAIN; DRUG DESIGN; ENZYME ACTIVATION; ENZYME INHIBITORS; FURANS; HUMANS; PHENYLUREA COMPOUNDS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84863039641 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201100487 Document Type: Article

Times cited : (22)

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