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Volumn 39, Issue 4, 2012, Pages 461-471

Bombesin analogues for gastrin-releasing peptide receptor imaging

Author keywords

64Cu; Antagonist; Bombesin (BBN); Gastrin releasing peptide receptor (GRPR); Positron emission tomography (PET)

Indexed keywords

BOMBESIN DERIVATIVE; COPPER 1,4,7 TRIAZACYCLONONANE 1,4 DIACETIC ACID 6 AMINO HEXANOIC ACID BOMBESIN[6-13][6 DEXTRO PHENYLALANINE]ETHYLAMIDE CU 64; COPPER 1,4,7 TRIAZACYCLONONANE 1,4 DIACETIC ACID 9 AMINONONANOIC ACID BOMBESIN[6-13][6 DEXTRO PHENYLALANINE]ETHYLAMIDE CU 64; GASTRIN RELEASING PEPTIDE RECEPTOR; UNCLASSIFIED DRUG;

EID: 84862819921     PISSN: 09698051     EISSN: 18729614     Source Type: Journal    
DOI: 10.1016/j.nucmedbio.2011.10.009     Document Type: Article
Times cited : (32)

References (35)
  • 1
    • 0033770607 scopus 로고    scopus 로고
    • Therapeutic use of radiolabelled peptides
    • Krenning E.P., De Jong M. Therapeutic use of radiolabelled peptides. Ann Oncol 2000, 11:267-271.
    • (2000) Ann Oncol , vol.11 , pp. 267-271
    • Krenning, E.P.1    De Jong, M.2
  • 3
    • 0035993355 scopus 로고    scopus 로고
    • Small peptide radiopharmaceuticals in the imaging of acute thrombus
    • Blum J.E., Handmaker H. Small peptide radiopharmaceuticals in the imaging of acute thrombus. Curr Pharm Des 2002, 8:1815-1826.
    • (2002) Curr Pharm Des , vol.8 , pp. 1815-1826
    • Blum, J.E.1    Handmaker, H.2
  • 4
    • 0034945777 scopus 로고    scopus 로고
    • Imaging tumors with peptide-based radioligands
    • Behr T.M., Gotthardt M., Barth A., Behe M. Imaging tumors with peptide-based radioligands. Q J Nucl Med 2001, 45:189-200.
    • (2001) Q J Nucl Med , vol.45 , pp. 189-200
    • Behr, T.M.1    Gotthardt, M.2    Barth, A.3    Behe, M.4
  • 6
    • 0034911579 scopus 로고    scopus 로고
    • Recent progress in fluorine-18 labelled peptide radiopharmaceuticals
    • Okarvi S.M. Recent progress in fluorine-18 labelled peptide radiopharmaceuticals. Eur J Nucl Med 2001, 28:929-938.
    • (2001) Eur J Nucl Med , vol.28 , pp. 929-938
    • Okarvi, S.M.1
  • 7
    • 27144533633 scopus 로고    scopus 로고
    • Radiolabeled peptide conjugates for targeting of the bombesin receptor superfamily subtypes
    • Smith C.J., Volkert W.A., Hoffman T.J. Radiolabeled peptide conjugates for targeting of the bombesin receptor superfamily subtypes. Nucl Med Biol 2005, 32:733-740.
    • (2005) Nucl Med Biol , vol.32 , pp. 733-740
    • Smith, C.J.1    Volkert, W.A.2    Hoffman, T.J.3
  • 8
    • 0033104343 scopus 로고    scopus 로고
    • Gastrin-releasing peptide receptors in the human prostate: relation to neoplastic transformation
    • Markwalder R., Reubi J.C. Gastrin-releasing peptide receptors in the human prostate: relation to neoplastic transformation. Cancer Res 1999, 59:1152-1159.
    • (1999) Cancer Res , vol.59 , pp. 1152-1159
    • Markwalder, R.1    Reubi, J.C.2
  • 9
    • 0008883289 scopus 로고    scopus 로고
    • 99mTc-labeled small peptides as diagnostic radiopharmaceuticals
    • 99mTc-labeled small peptides as diagnostic radiopharmaceuticals. Chem Rev 1999, 99:2235-2268.
    • (1999) Chem Rev , vol.99 , pp. 2235-2268
    • Liu, S.1    Edwards, D.S.2
  • 12
    • 0003964361 scopus 로고    scopus 로고
    • American Cancer Society, American Cancer Society, Atlanta
    • Cancer facts and figures 2010 2010, American Cancer Society, American Cancer Society, Atlanta.
    • (2010) Cancer facts and figures 2010
  • 13
    • 0033953894 scopus 로고    scopus 로고
    • Presence of receptors for bombesin/gastrin-releasing peptide and mRNA for three receptor subtypes in human prostate cancers
    • Sun B., Halmos G., Schally A.V., Wang X., Martinez M. Presence of receptors for bombesin/gastrin-releasing peptide and mRNA for three receptor subtypes in human prostate cancers. Prostate 2000, 42:295-303.
    • (2000) Prostate , vol.42 , pp. 295-303
    • Sun, B.1    Halmos, G.2    Schally, A.V.3    Wang, X.4    Martinez, M.5
  • 15
    • 33846120590 scopus 로고    scopus 로고
    • Copper chelation chemistry and its role in copper radiopharmaceuticals
    • Wadas T.J., Wong E.H., Weisman G.R., Anderson C.J. Copper chelation chemistry and its role in copper radiopharmaceuticals. Curr Pharm Des 2007, 13:3-16.
    • (2007) Curr Pharm Des , vol.13 , pp. 3-16
    • Wadas, T.J.1    Wong, E.H.2    Weisman, G.R.3    Anderson, C.J.4
  • 16
    • 67651151216 scopus 로고    scopus 로고
    • True radiotracers: Cu-64 targeting vectors based upon bombesin peptide
    • Hoffman T.J., Smith C.J. True radiotracers: Cu-64 targeting vectors based upon bombesin peptide. Nucl Med Biol 2009, 36:579-585.
    • (2009) Nucl Med Biol , vol.36 , pp. 579-585
    • Hoffman, T.J.1    Smith, C.J.2
  • 18
    • 0001579481 scopus 로고    scopus 로고
    • Radiometal-labeled agents (non-technetium) for diagnostic imaging
    • Anderson C.J., Welch M.J. Radiometal-labeled agents (non-technetium) for diagnostic imaging. Chem Rev 1999, 99:2219-2234.
    • (1999) Chem Rev , vol.99 , pp. 2219-2234
    • Anderson, C.J.1    Welch, M.J.2
  • 19
    • 0030292909 scopus 로고    scopus 로고
    • Copper radionuclides and radiopharmaceuticals in nuclear medicine
    • Blower P.J., Lewis J.S., Zweit J. Copper radionuclides and radiopharmaceuticals in nuclear medicine. Nucl Med Biol 1996, 23:957-980.
    • (1996) Nucl Med Biol , vol.23 , pp. 957-980
    • Blower, P.J.1    Lewis, J.S.2    Zweit, J.3
  • 20
    • 33645974333 scopus 로고    scopus 로고
    • Receptor radionuclide therapy of tumors: a road from basic research to clinical applications
    • Bodei L., Paganelli G., Mariani G. Receptor radionuclide therapy of tumors: a road from basic research to clinical applications. J Nucl Med 2006, 47:375-377.
    • (2006) J Nucl Med , vol.47 , pp. 375-377
    • Bodei, L.1    Paganelli, G.2    Mariani, G.3
  • 21
    • 0030756892 scopus 로고    scopus 로고
    • Endocytosis and recycling of G protein-coupled receptors
    • Koenig J.A., Edwardson J.M. Endocytosis and recycling of G protein-coupled receptors. Trends Pharmacol Sci 1997, 18:276-287.
    • (1997) Trends Pharmacol Sci , vol.18 , pp. 276-287
    • Koenig, J.A.1    Edwardson, J.M.2
  • 22
    • 33646005541 scopus 로고    scopus 로고
    • Internalization of sst2, sst3, and sst5 receptors: effects of somatostatin agonists and antagonists
    • Cescato R., Schulz S., Waser B., Eltschinger V., Rivier J.E., Wester H.J., et al. Internalization of sst2, sst3, and sst5 receptors: effects of somatostatin agonists and antagonists. J Nucl Med 2006, 47:502-511.
    • (2006) J Nucl Med , vol.47 , pp. 502-511
    • Cescato, R.1    Schulz, S.2    Waser, B.3    Eltschinger, V.4    Rivier, J.E.5    Wester, H.J.6
  • 23
    • 33750823665 scopus 로고    scopus 로고
    • Radiolabeled somatostatin receptor antagonists are preferable to agonists for in vivo peptide receptor targeting of tumors
    • Ginj M., Zhang H., Waser B., Cescato R., Wild D., Wang X., et al. Radiolabeled somatostatin receptor antagonists are preferable to agonists for in vivo peptide receptor targeting of tumors. Proc Natl Acad Sci USA 2006, 103:16436-16441.
    • (2006) Proc Natl Acad Sci USA , vol.103 , pp. 16436-16441
    • Ginj, M.1    Zhang, H.2    Waser, B.3    Cescato, R.4    Wild, D.5    Wang, X.6
  • 25
    • 0030975625 scopus 로고    scopus 로고
    • Pharmacokinetic considerations in the development of peptide-based imaging agents
    • Lister-James J., Moyer B.R., Dean R.T. Pharmacokinetic considerations in the development of peptide-based imaging agents. Q J Nucl Med 1997, 41:111-118.
    • (1997) Q J Nucl Med , vol.41 , pp. 111-118
    • Lister-James, J.1    Moyer, B.R.2    Dean, R.T.3
  • 26
    • 0032408581 scopus 로고    scopus 로고
    • Strategies to reduce renal radioactivity levels of antibody fragments
    • Arano Y. Strategies to reduce renal radioactivity levels of antibody fragments. Q J Nucl Med 1998, 42:262-270.
    • (1998) Q J Nucl Med , vol.42 , pp. 262-270
    • Arano, Y.1
  • 30
    • 69349102846 scopus 로고    scopus 로고
    • Evaluation of a 1,4,7,10-tetraazacyclododecane-1,4,7,10-tetraacetic acid-conjugated bombesin-based radioantagonist for the labeling with single-photon emission computed tomography, positron emission tomography, and therapeutic radionuclides
    • Mansi R., Wang X., Forrer F., Kneifel S., Tamma M.L., Waser B., et al. Evaluation of a 1,4,7,10-tetraazacyclododecane-1,4,7,10-tetraacetic acid-conjugated bombesin-based radioantagonist for the labeling with single-photon emission computed tomography, positron emission tomography, and therapeutic radionuclides. Clin Cancer Res 2009, 15:5240-5249.
    • (2009) Clin Cancer Res , vol.15 , pp. 5240-5249
    • Mansi, R.1    Wang, X.2    Forrer, F.3    Kneifel, S.4    Tamma, M.L.5    Waser, B.6
  • 31
    • 79551537113 scopus 로고    scopus 로고
    • Development of a potent DOTA-conjugated bombesin antagonist for targeting GRPr-positive tumours
    • Mansi R., Wang X., Forrer F., Waser B., Cescato R., Graham K., et al. Development of a potent DOTA-conjugated bombesin antagonist for targeting GRPr-positive tumours. Eur J Nucl Med Mol Imaging 2011, 38:97-107.
    • (2011) Eur J Nucl Med Mol Imaging , vol.38 , pp. 97-107
    • Mansi, R.1    Wang, X.2    Forrer, F.3    Waser, B.4    Cescato, R.5    Graham, K.6
  • 32
    • 0037945450 scopus 로고    scopus 로고
    • 111In-labeled bombesin analogs as potential radiopharmaceuticals for specific targeting of gastrin-releasing peptide receptors expressed on human prostate cancer cells
    • 111In-labeled bombesin analogs as potential radiopharmaceuticals for specific targeting of gastrin-releasing peptide receptors expressed on human prostate cancer cells. J Nucl Med 2003, 44:823-831.
    • (2003) J Nucl Med , vol.44 , pp. 823-831
    • Hoffman, T.J.1    Gali, H.2    Smith, C.J.3    Sieckman, G.L.4    Hayes, D.L.5    Owen, N.K.6
  • 33
    • 33745511768 scopus 로고    scopus 로고
    • Slow antagonist dissociation and long-lasting in vivo receptor protection
    • Vauquelin G., Van Liefde I. Slow antagonist dissociation and long-lasting in vivo receptor protection. Trends Pharmacol Sci 2006, 27:356-359.
    • (2006) Trends Pharmacol Sci , vol.27 , pp. 356-359
    • Vauquelin, G.1    Van Liefde, I.2
  • 34
    • 33846472504 scopus 로고    scopus 로고
    • Peptide receptors in neuroendocrine tumors of the lung as potential tools for radionuclide diagnosis and therapy
    • Pelosi G., Volante M., Papotti M., Sonzogni A., Masullo M., Viale G. Peptide receptors in neuroendocrine tumors of the lung as potential tools for radionuclide diagnosis and therapy. Q J Nucl Med Mol Imaging 2006, 50:272-287.
    • (2006) Q J Nucl Med Mol Imaging , vol.50 , pp. 272-287
    • Pelosi, G.1    Volante, M.2    Papotti, M.3    Sonzogni, A.4    Masullo, M.5    Viale, G.6
  • 35
    • 38049132623 scopus 로고    scopus 로고
    • Bombesin-related peptides and their receptors: recent advances in their role in physiology and disease states
    • Gonzalez N., Moody T.W., Igarashi H., Ito T., Jensen R.T. Bombesin-related peptides and their receptors: recent advances in their role in physiology and disease states. Curr Opin Endocrinol Diabetes Obes 2008, 15:58-64.
    • (2008) Curr Opin Endocrinol Diabetes Obes , vol.15 , pp. 58-64
    • Gonzalez, N.1    Moody, T.W.2    Igarashi, H.3    Ito, T.4    Jensen, R.T.5


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