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Volumn 44, Issue 5, 2003, Pages 823-831

Novel series of 111In-labeled bombesin analogs as potential radiopharmaceuticals for specific targeting of gastrin-releasing peptide receptors expressed on human prostate cancer cells

Author keywords

111In; Bombesin; Gastrin releasing peptide; Prostate cancer

Indexed keywords

1,4,7,10 TETRAAZACYCLODODECANE 1,4,7,10 TETRAACETIC ACID; BOMBESIN DERIVATIVE; GASTRIN RELEASING PEPTIDE; INDIUM 111; RADIOPHARMACEUTICAL AGENT; BOMBESIN RECEPTOR; DIAGNOSTIC AGENT; INDIUM;

EID: 0037945450     PISSN: 01615505     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article
Times cited : (158)

References (40)
  • 1
    • 0033233437 scopus 로고    scopus 로고
    • 99mTc-labelled peptide-based radiopharmaceuticals an overview
    • 99mTc-labelled peptide-based radiopharmaceuticals an overview. Nucl Med Commun. 1999;20:1093-1112
    • (1999) Nucl Med Commun , vol.20 , pp. 1093-1112
    • Okarvi, S.M.1
  • 2
    • 0034976943 scopus 로고    scopus 로고
    • Radiometallated receptor-avid peptide conjugates for specific in vivo targeting of cancer cells
    • Hoffman TJ, Quinn TP, Volkert WA. Radiometallated receptor-avid peptide conjugates for specific in vivo targeting of cancer cells. Nucl Med Biol. 2001; 28:527-539.
    • (2001) Nucl Med Biol , vol.28 , pp. 527-539
    • Hoffman, T.J.1    Quinn, T.P.2    Volkert, W.A.3
  • 3
    • 0015224130 scopus 로고
    • Isolation and structure of bombesin and alytesin, two analogous active peptides from the skin of the European amphibians Bombina and Alytes
    • Anastasia A, Erspamer V, Bucci H. Isolation and structure of bombesin and alytesin, two analogous active peptides from the skin of the European amphibians Bombina and Alytes. Experientia. 1971;27:166-168.
    • (1971) Experientia , vol.27 , pp. 166-168
    • Anastasia, A.1    Erspamer, V.2    Bucci, H.3
  • 5
    • 0028347654 scopus 로고
    • Inhibitory effect of bombesin receptor antagonist RC-3095 on the growth of human pancreatic cancer cells in vivo and in vitro
    • Qin Y, Ertl T, Cai R-Z, Halmos G, Schally AV Inhibitory effect of bombesin receptor antagonist RC-3095 on the growth of human pancreatic cancer cells in vivo and in vitro. Cancer Res. 1994;54:1035-1041
    • (1994) Cancer Res , vol.54 , pp. 1035-1041
    • Qin, Y.1    Ertl, T.2    Cai, R.-Z.3    Halmos, G.4    Schally, A.V.5
  • 6
    • 0000257596 scopus 로고
    • 13, 14 Bombesin analogues inhibit growth of small cell lung cancer in vitro and in vivo
    • 13, 14] Bombesin analogues inhibit growth of small cell lung cancer in vitro and in vivo. Life Sci. 1985;37:105-113.
    • (1985) Life Sci , vol.37 , pp. 105-113
    • Mahmoud, S.1    Staley, J.2    Taylor, J.3
  • 7
    • 0026472872 scopus 로고
    • Systematic development of bombesin/gastrin-releasing peptide antagonists
    • Coy DH, Jensen RT, Jiang NY. Systematic development of bombesin/gastrin-releasing peptide antagonists. J Natl Cancer Inst Monogr. 1992;13:133-139
    • (1992) J Natl Cancer Inst Monogr , vol.13 , pp. 133-139
    • Coy, D.H.1    Jensen, R.T.2    Jiang, N.Y.3
  • 8
    • 0030012609 scopus 로고    scopus 로고
    • Review, peptides and growth factors in non-small cell lung cancer
    • Moody TW. Review, peptides and growth factors in non-small cell lung cancer. Peptides. 1996;17:545-555.
    • (1996) Peptides , vol.17 , pp. 545-555
    • Moody, T.W.1
  • 10
    • 0022560610 scopus 로고
    • 4-bombesin with specific receptors on normal human pancreatic membranes
    • 4-bombesin with specific receptors on normal human pancreatic membranes. Regul Pept. 1986; 13:125-132.
    • (1986) Regul Pept , vol.13 , pp. 125-132
    • Scemama, J.L.1    Zahidi, A.2    Fourmy, D.3
  • 11
    • 0033754433 scopus 로고    scopus 로고
    • Technetium-99m RP525, a GRP analogue for visualization of GRP receptor-expressing malignancies: A feasibility study
    • Van de Wiele C, Dumont F, Broecke RV, et al Technetium-99m RP525, a GRP analogue for visualization of GRP receptor-expressing malignancies: a feasibility study Eur J Nucl Med 2000;27:1694-1699.
    • (2000) Eur J Nucl Med , vol.27 , pp. 1694-1699
    • Van De Wiele, C.1    Dumont, F.2    Broecke, R.V.3
  • 13
    • 0000860002 scopus 로고    scopus 로고
    • Iodinated bombesin analogs: Effect of a N-terminal vs. side chain iodine attachment of BBN/GRP receptor binding
    • Hoffman TJ, Sieckman GL, Volkert WA. Iodinated bombesin analogs: effect of a N-terminal vs. side chain iodine attachment of BBN/GRP receptor binding [abstract]. J Nucl Med. 1996;37(suppl):185P.
    • (1996) J Nucl Med , vol.37 , Issue.SUPPL.
    • Hoffman, T.J.1    Sieckman, G.L.2    Volkert, W.A.3
  • 15
    • 0032587895 scopus 로고    scopus 로고
    • 99mTc labelling and in vivo studies of a bombesin analog with a novel water-soluble bifunctional chelating agent
    • 99mTc labelling and in vivo studies of a bombesin analog with a novel water-soluble bifunctional chelating agent. Bioconjug Chem. 1999;10:254-260.
    • (1999) Bioconjug Chem , vol.10 , pp. 254-260
    • Karra, S.R.1    Schlbli, R.2    Gali, H.3
  • 16
    • 0000210044 scopus 로고    scopus 로고
    • Accumulation and retention of Tc-99m RP527 by GRP receptor expressing tumors in scid mice
    • Hoffman TJ, Simpson SD, Smith CJ, et al. Accumulation and retention of Tc-99m RP527 by GRP receptor expressing tumors in scid mice [abstract]. J Nucl Med. 1999;40(suppl) 104P.
    • (1999) J Nucl Med , vol.40 , Issue.SUPPL.
    • Hoffman, T.J.1    Simpson, S.D.2    Smith, C.J.3
  • 17
    • 4243678171 scopus 로고    scopus 로고
    • 99mTc-GRP receptor targeting peptides using multi-amino acid linking groups
    • 99mTc-GRP receptor targeting peptides using multi-amino acid linking groups [abstract]. J Nucl Med. 2000;41(suppl).228P.
    • (2000) J Nucl Med , vol.41 , Issue.SUPPL.
    • Hoffman, T.J.1    Smith, C.J.2    Simpson, S.D.3
  • 19
    • 0031458825 scopus 로고    scopus 로고
    • Synthesis of bombesin analogues for radiolabeling with rhenium-188
    • Safavy A, Khazaeli MB, Qin H, Buchsbaum DJ. Synthesis of bombesin analogues for radiolabeling with rhenium-188. Cancer Suppl 1997;80:2354-2359.
    • (1997) Cancer Suppl , vol.80 , pp. 2354-2359
    • Safavy, A.1    Khazaeli, M.B.2    Qin, H.3    Buchsbaum, D.J.4
  • 21
    • 0032958842 scopus 로고    scopus 로고
    • Evaluation of radiolabelled bombesin analogues for receptor-targeted scintigraphy and radiotherapy
    • Breeman WAP, Hofland LJ, DeJong M, et al. Evaluation of radiolabelled bombesin analogues for receptor-targeted scintigraphy and radiotherapy. Int J Cancer. 1999;81:658-665.
    • (1999) Int J Cancer , vol.81 , pp. 658-665
    • Breeman, W.A.P.1    Hofland, L.J.2    DeJong, M.3
  • 22
  • 24
    • 1942472187 scopus 로고    scopus 로고
    • 64Cu-labeled bombesin analogue for diagnosis of gastrin-releasing peptide receptor positive tumors by microPET imaging
    • 64Cu-labeled bombesin analogue for diagnosis of gastrin-releasing peptide receptor positive tumors by microPET imaging. J Labelled Compds Radiopharm. 2001;44(suppl): S81-S83.
    • (2001) J Labelled Compds Radiopharm , vol.44 , Issue.SUPPL.
    • Rogers, B.E.1    McCarthy, D.W.2    Sharp, T.L.3
  • 25
    • 0002737749 scopus 로고
    • Selective drug delivery by means of receplor-mediated endocytosis
    • Bijsterbosch MK. Selective drug delivery by means of receplor-mediated endocytosis. Q J Nucl Med 1995;39:4-9.
    • (1995) Q J Nucl Med , vol.39 , pp. 4-9
    • Bijsterbosch, M.K.1
  • 26
    • 0029316517 scopus 로고
    • Structural and functional analysis of G protein-coupled receptors and potential diagnostic ligands
    • Fraser CM Structural and functional analysis of G protein-coupled receptors and potential diagnostic ligands J Nucl Med 1995;36(suppl):17S-21S
    • (1995) J Nucl Med , vol.36 , Issue.SUPPL.
    • Fraser, C.M.1
  • 27
    • 0000558958 scopus 로고    scopus 로고
    • Drug analysis based on signaling responses to G-protein-coupled receptors
    • Left P, ed. New York, NY: Marcel Dekker, Inc
    • Harden TK, Boyer JL, Dougherty RW. Drug analysis based on signaling responses to G-protein-coupled receptors. In. Left P, ed. Receptor-Based Drug Design. New York, NY: Marcel Dekker, Inc; 1998:79-105.
    • (1998) Receptor-Based Drug Design , pp. 79-105
    • Harden, T.K.1    Boyer, J.L.2    Dougherty, R.W.3
  • 28
    • 0030136744 scopus 로고    scopus 로고
    • Improved prospects for cancer therapy with radiolabeled antibody fragments and peptides
    • Behr TM, Goldenberg DM. Improved prospects for cancer therapy with radiolabeled antibody fragments and peptides. J Nucl Med. 1996;37:834-836
    • (1996) J Nucl Med , vol.37 , pp. 834-836
    • Behr, T.M.1    Goldenberg, D.M.2
  • 29
    • 0035155042 scopus 로고    scopus 로고
    • Bifunctional chelators for therapeutic lanthanide radiopharmaceuticals
    • Liu S, Edwards DS. Bifunctional chelators for therapeutic lanthanide radiopharmaceuticals. Bioconjug Chem. 2001;12:7-34
    • (2001) Bioconjug Chem , vol.12 , pp. 7-34
    • Liu, S.1    Edwards, D.S.2
  • 32
    • 0042929352 scopus 로고    scopus 로고
    • 3]octreotide, a promising somatostatin analogue for radionuclide therapy
    • 3]octreotide, a promising somatostatin analogue for radionuclide therapy. Eur J Nucl Med 1997;24:368-371.
    • (1997) Eur J Nucl Med , vol.24 , pp. 368-371
    • Jong, M.1    Bakker, W.H.2    Krenning, E.P.3
  • 33
    • 0033033382 scopus 로고    scopus 로고
    • Radiometal-labelled macrocyclic chelator derivatized somatostatin analogue with superb tumor targeting properties and potential for receptor mediated internal radiotherapy
    • Heppeler A, Froidevaux S, Macke HR, et al. Radiometal-labelled macrocyclic chelator derivatized somatostatin analogue with superb tumor targeting properties and potential for receptor mediated internal radiotherapy. Chem Eur J. 1999;5: 1974-1981
    • (1999) Chem Eur J , vol.5 , pp. 1974-1981
    • Heppeler, A.1    Froidevaux, S.2    Macke, H.R.3
  • 34
    • 0030975625 scopus 로고    scopus 로고
    • Pharmacokinetic considerations in the development of peptide-based imaging agents
    • Lister-James J, Moyer BR, Dean RT. Pharmacokinetic considerations in the development of peptide-based imaging agents. Q J Nucl Med 1997;41:111-118.
    • (1997) Q J Nucl Med , vol.41 , pp. 111-118
    • Lister-James, J.1    Moyer, B.R.2    Dean, R.T.3
  • 35
    • 0001699495 scopus 로고    scopus 로고
    • Structural characterization and binding sites of G-protein-coupled receptors
    • Beck-Sickinger AG. Structural characterization and binding sites of G-protein-coupled receptors. Drug Discov Today, 1996;1:502-513.
    • (1996) Drug Discov Today , vol.1 , pp. 502-513
    • Beck-Sickinger, A.G.1
  • 36
    • 0027368237 scopus 로고
    • Intracellular metabolism of indium-111-DTPA-labeled receptor targeted proteins
    • Duncan JR, Welch MJ. Intracellular metabolism of indium-111-DTPA-labeled receptor targeted proteins. J Nucl Med. 1993;34:1728-1738.
    • (1993) J Nucl Med , vol.34 , pp. 1728-1738
    • Duncan, J.R.1    Welch, M.J.2
  • 37
    • 0028364617 scopus 로고
    • Internalization and degradation of monoclonal antibody chCE7 by human neuroblastoma cells
    • Novak-Hofer I, Amstutz HP, Morgenthaler JJ, Schubiger PA. Internalization and degradation of monoclonal antibody chCE7 by human neuroblastoma cells. Int J Cancer. 1994;57:427-432.
    • (1994) Int J Cancer , vol.57 , pp. 427-432
    • Novak-Hofer, I.1    Amstutz, H.P.2    Morgenthaler, J.J.3    Schubiger, P.A.4
  • 38
    • 0032408581 scopus 로고    scopus 로고
    • Strategies to reduce renal radioactivity levels of antibody fragments
    • Arano Y. Strategies to reduce renal radioactivity levels of antibody fragments Q J Nucl Med 1998;42:262-267.
    • (1998) Q J Nucl Med , vol.42 , pp. 262-267
    • Arano, Y.1
  • 39
    • 0034667352 scopus 로고    scopus 로고
    • Melanoma-targeting properties of (99m)technetium-labeled cyclic alpha-melanocyte-stimulating hormone peptide analogues
    • Chen J, Chen Z, Hoffman TJ, Jurisson SS, Quinn TP. Melanoma-targeting properties of (99m)technetium-labeled cyclic alpha-melanocyte-stimulating hormone peptide analogues. Cancer Res. 2000;60:5649-5658.
    • (2000) Cancer Res , vol.60 , pp. 5649-5658
    • Chen, J.1    Chen, Z.2    Hoffman, T.J.3    Jurisson, S.S.4    Quinn, T.P.5
  • 40
    • 0012725753 scopus 로고    scopus 로고
    • Therapeutic radiopharmaceuticals
    • Volkert WA, Hoffman TJ. Therapeutic radiopharmaceuticals. Chem Rev. 1999; 99:2269-2292
    • (1999) Chem Rev , vol.99 , pp. 2269-2292
    • Volkert, W.A.1    Hoffman, T.J.2


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