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Volumn 56, Issue 1, 2012, Pages 11-18

Evaluation of the in vitro antiretroviral potential of some Biginelli-type pyrimidines

Author keywords

Antivirals; Biginelli type pyrimidines; HIV 1

Indexed keywords

ANTI HUMAN IMMUNODEFICIENCY VIRUS AGENT; PYRIMIDINE DERIVATIVE; GREEN FLUORESCENT PROTEIN; LUCIFERASE;

EID: 84862245323     PISSN: 0001723X     EISSN: None     Source Type: Journal    
DOI: 10.4149/av_2012_01_11     Document Type: Article
Times cited : (33)

References (46)
  • 1
    • 0029984987 scopus 로고    scopus 로고
    • Cell type-specific fusion cofactors determine human immunodeficiency virus type 1 tropism for T-cell lines versus primary macrophages
    • Alkhatib G, Broder CC, Berger EA (1996): Cell type-specific fusion cofactors determine human immunodeficiency virus type 1 tropism for T-cell lines versus primary macrophages. J. Virol. 70, 5487-5494.
    • (1996) J. Virol. , vol.70 , pp. 5487-5494
    • Alkhatib, G.1    Broder, C.C.2    Berger, E.A.3
  • 2
    • 33847753903 scopus 로고    scopus 로고
    • Convenient one pot synthesis of some novel derivatives of thiazolo[2 3-b] dihydropyrimidinone possessing 4-methylthiophenyl moiety and evaluation of their antibacterial and antifungal activities
    • Ashok M, Holla BS, Kumari NS (2007): Convenient one pot synthesis of some novel derivatives of thiazolo[2,3-b] dihydropyrimidinone possessing 4-methylthiophenyl moiety and evaluation of their antibacterial and antifungal activities. Eur. J. Med. Chem. 42, 380-385. http://dx.doi.org/10.1016/j.ejmech.2006.09.003
    • (2007) Eur. J. Med. Chem. , vol.42 , pp. 380-385
    • Ashok, M.1    Holla, B.S.2    Kumari, N.S.3
  • 3
    • 1542404601 scopus 로고    scopus 로고
    • Synthesis and anti-inflammatory activity of some [4,6-(4-substituted aryl)-2-thioxo-1,2,3 4-tetrahydro-pyrimidin-5-yl]-acetic acid derivatives
    • Bahekar SS, Shinde DB (2004): Synthesis and anti-inflammatory activity of some [4,6-(4-substituted aryl)-2-thioxo-1,2,3,4-tetrahydro-pyrimidin-5-yl]-acetic acid derivatives. Bioorg. Med. Chem. Lett. 14, 1733-1736. http://dx.doi.org/10.1016/j.bmcl.2004.01.039
    • (2004) Bioorg. Med. Chem. Lett. , vol.14 , pp. 1733-1736
    • Bahekar, S.S.1    Shinde, D.B.2
  • 7
    • 0032978963 scopus 로고    scopus 로고
    • Human immunodeficiency virus type 1 Tat induces apoptosis and increases sensitivity to apoptotic signals by up-regulating FLICE/caspase-8
    • Bartz SR, Emerman M (1999): Human immunodeficiency virus type 1 Tat induces apoptosis and increases sensitivity to apoptotic signals by up-regulating FLICE/caspase-8. J. Virol. 73, 1956-1963.
    • (1999) J. Virol. , vol.73 , pp. 1956-1963
    • Bartz, S.R.1    Emerman, M.2
  • 8
    • 40649089628 scopus 로고    scopus 로고
    • Solvent-free synthesis of dihydropyrimidinones catalyzed by alumina sulfuric acid at room temperature
    • Besoluk S, Kucukislamoglu M, Nebioglu M, Zengin M, Arslan M (2008): Solvent-free synthesis of dihydropyrimidinones catalyzed by alumina sulfuric acid at room temperature. J. Iran Chem. Soc. 5, 62-66.
    • (2008) J. Iran Chem. Soc. , vol.5 , pp. 62-66
    • Besoluk, S.1    Kucukislamoglu, M.2    Nebioglu, M.3    Zengin, M.4    Arslan, M.5
  • 9
    • 0000176059 scopus 로고
    • Aldehyde-urea derivatives of aceto-and oxaloacetic acids
    • Biginelli P (1893): Aldehyde-urea derivatives of aceto-and oxaloacetic acids. Gaz. Chim. Ital. 23, 360-413.
    • (1893) Gaz. Chim. Ital. , vol.23 , pp. 360-413
    • Biginelli, P.1
  • 10
    • 33947601363 scopus 로고    scopus 로고
    • Labeling HIV-1 virions with two fluorescent proteins allows identification of virions that have productively entered the target cell
    • Campbell EM, Perez O, Melar M, Hope TJ (2007): Labeling HIV-1 virions with two fluorescent proteins allows identification of virions that have productively entered the target cell. Virology 360, 286-293. http://dx.doi.org/10.1016/j.virol.2006.10.025
    • (2007) Virology , vol.360 , pp. 286-293
    • Campbell, E.M.1    Perez, O.2    Melar, M.3    Hope, T.J.4
  • 11
    • 0030053308 scopus 로고    scopus 로고
    • Molecular determinants of acute single-cell lysis by human immunodefi-ciency virus type 1
    • Cao J, Park IW, Cooper A, Sodroski J (1996): Molecular determinants of acute single-cell lysis by human immunodefi-ciency virus type 1. J. Virol. 70, 1340-1354.
    • (1996) J. Virol. , vol.70 , pp. 1340-1354
    • Cao, J.1    Park, I.W.2    Cooper, A.3    Sodroski, J.4
  • 12
    • 4544240500 scopus 로고    scopus 로고
    • HIV-1 virion fusion assay: uncoating not required and no eff ect of Nef on fusion
    • Cavrois M, Neidleman J, Yonemoto W, Fenard D, Greene WC (2004): HIV-1 virion fusion assay: uncoating not required and no eff ect of Nef on fusion. Virology 328, 36-44. http://dx.doi.org/10.1016/j.virol.2004.07.015
    • (2004) Virology , vol.328 , pp. 36-44
    • Cavrois, M.1    Neidleman, J.2    Yonemoto, W.3    Fenard, D.4    Greene, W.C.5
  • 13
    • 0033050673 scopus 로고    scopus 로고
    • Mutational analysis of Vprinduced G2 arrest, nuclear localization, and cell death in fission yeast
    • Chen M, Elder RT, Yu M, O'Gorman MG, Selig L, Benarous R, Yamamoto A, Zhao Y (1999): Mutational analysis of Vprinduced G2 arrest, nuclear localization, and cell death in fission yeast. J. Virol. 73, 3236-3245.
    • (1999) J. Virol. , vol.73 , pp. 3236-3245
    • Chen, M.1    Elder, R.T.2    Yu, M.3    O'Gorman, M.G.4    Selig, L.5    Benarous, R.6    Yamamoto, A.7    Zhao, Y.8
  • 15
    • 0027500534 scopus 로고
    • A model for reverse transcription by a dimeric enzyme
    • Cook PR (1993): A model for reverse transcription by a dimeric enzyme. J. Gen. Virol. 74, 691-697. http://dx.doi.org/10.1099/0022-1317-74-4-691
    • (1993) J. Gen. Virol. , vol.74 , pp. 691-697
    • Cook, P.R.1
  • 16
    • 0026086345 scopus 로고
    • Demonstration of two distinct cytopathic effects with syncytium formation-defective human immunodeficiency virus type 1 mutants
    • Dedera D, Ratner L (1991): Demonstration of two distinct cytopathic effects with syncytium formation-defective human immunodeficiency virus type 1 mutants. J. Virol. 65, 6129-6136.
    • (1991) J. Virol. , vol.65 , pp. 6129-6136
    • Dedera, D.1    Ratner, L.2
  • 18
    • 0021315381 scopus 로고
    • NIH conference. Acquired immunodeficiency syndrome: epidemiologic, clinical, immunologic, and therapeutic considerations
    • Fauci AS, Macher AM, Longo DL, Lane HC, Rook AH, Masur H, Gelmann EP (1984): NIH conference. Acquired immunodeficiency syndrome: epidemiologic, clinical, immunologic, and therapeutic considerations. Ann. Intern. Med. 100, 92-106.
    • (1984) Ann. Intern. Med. , vol.100 , pp. 92-106
    • Fauci, A.S.1    Macher, A.M.2    Longo, D.L.3    Lane, H.C.4    Rook, A.H.5    Masur, H.6    Gelmann, E.P.7
  • 20
    • 0006618044 scopus 로고
    • Experimental chemotherapy of infection with agents of the psittacosis-lymphogranuloma-trachoma group
    • Hurst EW (1962): Experimental chemotherapy of infection with agents of the psittacosis-lymphogranuloma-trachoma group. Ann. NY Acad. Sci. 98, 275-286. http://dx.doi.org/10.1111/j.1749-6632.1962.tb30551.x
    • (1962) Ann. NY Acad. Sci. , vol.98 , pp. 275-286
    • Hurst, E.W.1
  • 21
    • 0001457151 scopus 로고
    • Two new synthetic substances active against viruses of the psittacosis-lymphogranulomatrachoma group
    • Hurst EW, Hull R (1961): Two new synthetic substances active against viruses of the psittacosis-lymphogranulomatrachoma group. J. Med. Pharm. Chem. 3, 215-229. http://dx.doi.org/10.1021/jm50015a002
    • (1961) J. Med. Pharm. Chem. , vol.3 , pp. 215-229
    • Hurst, E.W.1    Hull, R.2
  • 22
    • 10644280992 scopus 로고    scopus 로고
    • Action of anti-HIV drugs and resistance: reverse transcriptase inhibitors and protease inhibitors
    • Imamichi T (2004): Action of anti-HIV drugs and resistance: reverse transcriptase inhibitors and protease inhibitors. Curr. Pharm. Des. 10, 4039-4053. http://dx.doi.org/10.2174/1381612043382440
    • (2004) Curr. Pharm. Des. , vol.10 , pp. 4039-4053
    • Imamichi, T.1
  • 23
    • 34249826040 scopus 로고    scopus 로고
    • An efficient and solvent-free one-pot synthesis of dihydropyrimidinones under microwave irradiation
    • Jiang C, You QD (2007): An efficient and solvent-free one-pot synthesis of dihydropyrimidinones under microwave irradiation. Chinese Chem. Lett. 18, 647-650. http://dx.doi.org/10.1016/j.cclet.2007.04.002
    • (2007) Chinese Chem. Lett. , vol.18 , pp. 647-650
    • Jiang, C.1    You, Q.D.2
  • 24
    • 0034519777 scopus 로고    scopus 로고
    • Biologically active dihydropyrimidones of the Biginelli-type-a literature survey
    • Kappe CO (2000): Biologically active dihydropyrimidones of the Biginelli-type-a literature survey. Eur. J. Med. Chem. 35, 1043-1052. http://dx.doi.org/10.1016/S0223-5234(00)01189-2
    • (2000) Eur. J. Med. Chem. , vol.35 , pp. 1043-1052
    • Kappe, C.O.1
  • 26
    • 33845233147 scopus 로고    scopus 로고
    • An environmentally benign protocol for the synthesis of 3 4-dihydropyrimidine-2(1H)-ones using solid acid catalysts under solvent-free conditions
    • Kumar D, Mishra BG, Rao VS (2006): An environmentally benign protocol for the synthesis of 3,4-dihydropyrimidine-2(1H)-ones using solid acid catalysts under solvent-free conditions. Indian J. Chem. 45, 2325-2329.
    • (2006) Indian J. Chem. , vol.45 , pp. 2325-2329
    • Kumar, D.1    Mishra, B.G.2    Rao, V.S.3
  • 27
    • 0038619031 scopus 로고    scopus 로고
    • Cytolysis by CCR5-using human immunodeficiency virus type 1 envelope glycoproteins is dependent on membrane fusion and can be inhibited by high levels of CD4+ expression
    • LaBonte JA, Madani N, Sodroski J (2003): Cytolysis by CCR5-using human immunodeficiency virus type 1 envelope glycoproteins is dependent on membrane fusion and can be inhibited by high levels of CD4+ expression. J. Virol. 77, 6645-6659. http://dx.doi.org/10.1128/JVI.77.12.6645-6659.2003
    • (2003) J. Virol. , vol.77 , pp. 6645-6659
    • LaBonte, J.A.1    Madani, N.2    Sodroski, J.3
  • 29
    • 4043100135 scopus 로고    scopus 로고
    • CoC12 6H2O or LaCl3 7H2O catalyzed Biginelli reaction One-pot synthesis of 3 4-dihydropyrimidin-2(1H)-ones
    • Lu J, Bai YJ, Wang ZJ, Ma HR (2002): CoC12 6H2O or LaCl3 7H2O catalyzed Biginelli reaction. One-pot synthesis of 3 4-dihydropyrimidin-2(1H)-ones. Chinese Chem. Lett. 20, 681-687.
    • (2002) Chinese Chem. Lett. , vol.20 , pp. 681-687
    • Lu, J.1    Bai, Y.J.2    Wang, Z.J.3    Ma, H.R.4
  • 30
    • 33846087827 scopus 로고    scopus 로고
    • Inhibition of human immunodeficiency virus envelope glycoprotein-mediated single cell lysis by lowmolecular-weight antagonists of viral entry
    • Madani N, Hubicki AM, Perdigoto AL, Springer M, Sodroski J (2007): Inhibition of human immunodeficiency virus envelope glycoprotein-mediated single cell lysis by lowmolecular-weight antagonists of viral entry. J. Virol. 81, 532-538. http://dx.doi.org/10.1128/JVI.01079-06
    • (2007) J. Virol. , vol.81 , pp. 532-538
    • Madani, N.1    Hubicki, A.M.2    Perdigoto, A.L.3    Springer, M.4    Sodroski, J.5
  • 32
    • 77957288978 scopus 로고    scopus 로고
    • Antiretroviral drug resistance-implications for HIV/AIDS reduction in sub-Saharan Africa and other developing countries
    • Obiako OR, Murktar HM, Ogoina D (2010): Antiretroviral drug resistance-implications for HIV/AIDS reduction in sub-Saharan Africa and other developing countries. Niger J. Med. 19, 302-310.
    • (2010) Niger J. Med. , vol.19 , pp. 302-310
    • Obiako, O.R.1    Murktar, H.M.2    Ogoina, D.3
  • 33
    • 0030768607 scopus 로고    scopus 로고
    • HIV-1 Nef protein-induced apoptotic cytolysis of a broad spectrum of uninfected human blood cells independently of CD95(Fas)
    • Okada H, Takei R, Tashiro M (1997): HIV-1 Nef protein-induced apoptotic cytolysis of a broad spectrum of uninfected human blood cells independently of CD95(Fas). FEBS Lett. 414, 603-606. http://dx.doi.org/10.1016/S0014-5793(97)01080-6
    • (1997) FEBS Lett , vol.414 , pp. 603-606
    • Okada, H.1    Takei, R.2    Tashiro, M.3
  • 36
    • 0026759681 scopus 로고
    • Dihydropyrimidine calcium channel blockers. 4. Basic 3-substituted-4-aryl-1 4-dihydropyrimidine-5-carboxylic acid esters. Potent antihypertensive agents
    • Rovnyak GC, Atwal KS, Hedberg A, Kimball SD, Moreland S, Gougoutas JZ, O'Reilly BC, Schwartz J, Malley MF (1992): Dihydropyrimidine calcium channel blockers. 4. Basic 3-substituted-4-aryl-1,4-dihydropyrimidine-5-carboxylic acid esters. Potent antihypertensive agents. J. Med. Chem. 35, 3254-3263. http://dx.doi.org/10.1021/jm00095a023
    • (1992) J. Med. Chem. , vol.35 , pp. 3254-3263
    • Rovnyak, G.C.1    Atwal, K.S.2    Hedberg, A.3    Kimball, S.D.4    Moreland, S.5    Gougoutas, J.Z.6    O'Reilly, B.C.7    Schwartz, J.8    Malley, M.F.9
  • 37
    • 4043126308 scopus 로고    scopus 로고
    • Multicomponent Biginelli's synthesis of 3 4-dihydropyrimidin-2(1H)-ones promoted by SnCl2. 2H2O
    • Russowsky D, Lopes FA, da SV, Canto KFS, D'Oca MGM, Godoi MN. (2004): Multicomponent Biginelli's synthesis of 3,4-dihydropyrimidin-2(1H)-ones promoted by SnCl2.2H2O. J. Braz. Chem. Soc. 15, 165-169. http://dx.doi.org/10.1590/S0103-50532004000200002
    • (2004) J. Braz. Chem. Soc. , vol.15 , pp. 165
    • Russowsky, D.1    Lopes, F.A.2    da Silva, V.S.S.3    Canto, K.F.S.4    D'Oca, M.G.M.5    Godoi, M.N.6
  • 40
    • 0022518143 scopus 로고
    • Role of the HTLV-III/LAV envelope in syncytium formation and cytopathicity
    • Sodroski J, Goh WC, Rosen C, Campbell K, Haseltine WA (1986): Role of the HTLV-III/LAV envelope in syncytium formation and cytopathicity. Nature 322, 470-474. http://dx.doi.org/10.1038/322470a0
    • (1986) Nature , vol.322 , pp. 470-474
    • Sodroski, J.1    Goh, W.C.2    Rosen, C.3    Campbell, K.4    Haseltine, W.A.5
  • 41
    • 77953867676 scopus 로고    scopus 로고
    • Synthesis of 3 4-dihydropyrimidin-2(1H)-one-5-carboxamides
    • Soleymani M, Memarian HR (2010): Synthesis of 3,4-dihydropyrimidin-2(1H)-one-5-carboxamides. Z. Naturforsch. 65, 485-492.
    • (2010) Z. Naturforsch. , vol.65 , pp. 485-492
    • Soleymani, M.1    Memarian, H.R.2
  • 43
    • 77649232123 scopus 로고    scopus 로고
    • Therapeutic strategies underpinning the development of novel techniques for the treatment of HIV infection
    • Tan JJ, Cong XJ, Hu LM, Wang CX, Jia L, Liang XJ (2010): Therapeutic strategies underpinning the development of novel techniques for the treatment of HIV infection. Drug Discov. Today 15, 186-197. http://dx.doi.org/10.1016/j.drudis.2010.01.004
    • (2010) Drug Discov. Today , vol.15 , pp. 186-197
    • Tan, J.J.1    Cong, X.J.2    Hu, L.M.3    Wang, C.X.4    Jia, L.5    Liang, X.J.6
  • 46
    • 52049098921 scopus 로고    scopus 로고
    • Solvent-and catalyst-free synthesis of dihydropyrimidinthiones in one-pot under focused microwave irradiation conditions
    • Zhan HW, Wang JX, Wang XT (2008): Solvent-and catalyst-free synthesis of dihydropyrimidinthiones in one-pot under focused microwave irradiation conditions. Chinese Chem. Lett. 19, 1183-1185. http://dx.doi.org/10.1016/j.cclet.2008.06.039
    • (2008) Chinese Chem. Lett. , vol.19 , pp. 1183-1185
    • Zhan, H.W.1    Wang, J.X.2    Wang, X.T.3


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