-
1
-
-
0035212788
-
A receptors uncouples allosteric binding: Studies on possible mechanisms
-
DOI 10.1046/j.1471-4159.2001.00664.x
-
Ali NJ, Olsen RW. Chronic benzodiazepine treatment of cells expressing recombinant GABA(A) receptors uncouples allosteric binding: studies on possible mechanisms. J Neurochem 2001;79:1100-8. (Pubitemid 33117091)
-
(2001)
Journal of Neurochemistry
, vol.79
, Issue.5
, pp. 1100-1108
-
-
Ali, N.J.1
Olsen, R.W.2
-
2
-
-
0021872980
-
Pharmacological profile of the imidazopyridine zolpidem at benzodiazepine receptors and electrocorticogram in rats
-
DOI 10.1007/BF00572441
-
Arbilla S, Depoortere H, George P, Langer SZ. Pharmacological profile of the imidazopyridine zolpidem at benzodiazepine receptors and electrocorticogram in rats. Naunyn Schmiedebergs Arch Pharmacol 1985;330:248-51. (Pubitemid 15003586)
-
(1985)
Naunyn-Schmiedeberg's Archives of Pharmacology
, vol.330
, Issue.3
, pp. 248-251
-
-
Arbilla, S.1
Depoortere, H.2
George, P.3
Langer, S.Z.4
-
3
-
-
47149083428
-
Imidazenil: A low efficacy agonist at alpha1- But high efficacy at alpha5-GABAA receptors fail to show anticonvulsant cross tolerance to diazepam or zolpidem
-
Auta J, Impagnatiello F, Kadriu B, Guidotti A, Costa E. Imidazenil: a low efficacy agonist at alpha1- but high efficacy at alpha5-GABAA receptors fail to show anticonvulsant cross tolerance to diazepam or zolpidem. Neuropharmacology 2008;55:148-53.
-
(2008)
Neuropharmacology
, vol.55
, pp. 148-153
-
-
Auta, J.1
Impagnatiello, F.2
Kadriu, B.3
Guidotti, A.4
Costa, E.5
-
4
-
-
0036242083
-
Basic pharmacologic mechanisms involved in benzodiazepine tolerance and withdrawal
-
DOI 10.2174/1381612023396681
-
Bateson AN. Basic pharmacological mechanisms involved in benzodiazepine tolerance and withdrawal. Curr Pharm Des 2002;8:5-21. (Pubitemid 34449900)
-
(2002)
Current Pharmaceutical Design
, vol.8
, Issue.1
, pp. 5-21
-
-
Bateson, A.N.1
-
5
-
-
36749096756
-
A receptors
-
DOI 10.2174/138161207782341330
-
Birnir B, Korpi ER. The impact of sub-cellular location and intracellular neuronal proteins on properties of GABA(A) receptors. Curr Pharm Des 2007;13:3169-77. (Pubitemid 350201693)
-
(2007)
Current Pharmaceutical Design
, vol.13
, Issue.31
, pp. 3169-3177
-
-
Birnir, B.1
Korpi, E.R.2
-
6
-
-
0026778836
-
Expression patterns of gamma-aminobutyric acid type A receptor subunit mRNAs in primary cultures of granule neurons and astrocytes from neonatal rat cerebella
-
Bovolin P, Santi MR, Puia G, Costa E, Grayson D. Expression patterns of gamma-aminobutyric acid type A receptor subunit mRNAs in primary cultures of granule neurons and astrocytes from neonatal rat cerebella. Proc Natl Acad Sci 1992;89:9344-8.
-
(1992)
Proc Natl Acad Sci
, vol.89
, pp. 9344-9348
-
-
Bovolin, P.1
Santi, M.R.2
Puia, G.3
Costa, E.4
Grayson, D.5
-
7
-
-
0031595167
-
γ-Aminobutyric acid(A) receptor function is desensitised in rat cultured cerebellar granule cells following chronic flunitrazepam treatment
-
Brown MJ, Wood MD, Coldwell MC, Bristow DR. γ-Aminobutyric acidA receptor function is desensitized in rat cultured cerebellar granule cells following chronic flunitrazepam treatment. J Neurochem 1998;71:1232-40. (Pubitemid 28390278)
-
(1998)
Journal of Neurochemistry
, vol.71
, Issue.3
, pp. 1232-1240
-
-
Brown, M.J.1
Wood, M.D.2
Coldwell, M.C.3
Bristow, D.R.4
-
8
-
-
0030611649
-
2 subunit of γ-aminobutyric acid type A receptors results in altered benzodiazepine binding site specificity
-
DOI 10.1073/pnas.94.16.8824
-
Buhr A, Sigel E. A point mutation in the gamma2 subunit of gamma-aminobutyric acid type A receptors results in altered benzodiazepine binding site specificity. Proc Natl Acad Sci U S A 1997;94:8824-9. (Pubitemid 27335124)
-
(1997)
Proceedings of the National Academy of Sciences of the United States of America
, vol.94
, Issue.16
, pp. 8824-8829
-
-
Buhr, A.1
Sigel, E.2
-
9
-
-
34548283953
-
A receptor and docking studies with zolpidem: Implications for selectivity
-
A receptor and docking studies with zolpidem: implications for selectivity. J Mol Graph Model 2007;26:537-45.
-
(2007)
J Mol Graph Model
, vol.26
, pp. 537-545
-
-
Ci, S.Q.1
Ren, T.R.2
Ma, C.X.3
Su, Z.G.4
-
11
-
-
77957567758
-
Benzodiazepines on trial: A research strategy for their rehabilitation
-
Costa E, Guidotti A. Benzodiazepines on trial: a research strategy for their rehabilitation. Trends Pharmacol Sci 1996;71:1232-40.
-
(1996)
Trends Pharmacol Sci
, vol.71
, pp. 1232-1240
-
-
Costa, E.1
Guidotti, A.2
-
13
-
-
0024332759
-
Calculating receptor number from binding experiments using same compound as radioligand and competitor
-
DOI 10.1016/0165-6147(89)90266-6
-
DeBlasi A, O'Reilly K, Motulsky HJ. Calculating receptor number from binding experiments using same compound as radioligand and competitor. Trends Pharmacol Sci 1989;10:227-9. (Pubitemid 19146394)
-
(1989)
Trends in Pharmacological Sciences
, vol.10
, Issue.6
, pp. 227-229
-
-
DeBlasi, A.1
O'Reilly, K.2
Motulsky, H.J.3
-
14
-
-
0022613409
-
Zolpidem, a novel nonbenzodiazepine hypnotic. I. Neuropharmacological and behavioral effects
-
Depoortere H, Zivkovic B, Lloyd KG, Sanger DJ, Perrault G, Langer SZ, et al. Zolpidem, a novel nonbenzodiazepine hypnotic. I. Neuropharmacological and behavioral effects. J Pharmacol Exp Ther 1986;237:649-58. (Pubitemid 16092830)
-
(1986)
Journal of Pharmacology and Experimental Therapeutics
, vol.237
, Issue.2
, pp. 649-658
-
-
Depoortere, H.1
Zivkovic, B.2
Lloyd, K.G.3
-
15
-
-
0036170814
-
A receptor gene expression induced by withdrawal of, but not by long-term exposure to, zaleplon or zolpidem
-
DOI 10.1016/S0028-3908(01)00167-8, PII S0028390801001678
-
Follesa P, Mancuso L, Biggio F, Cagetti E, Franco M, Trapani G, et al. Changes in GABA(A) receptor gene expression induced by withdrawal of, but not by long-term exposure to, zaleplon or zolpidem. Neuropharmacology 2002;42:191-8. (Pubitemid 34137022)
-
(2002)
Neuropharmacology
, vol.42
, Issue.2
, pp. 191-198
-
-
Follesa, P.1
Mancuso, L.2
Biggio, F.3
Cagetti, E.4
Franco, M.5
Trapani, G.6
Biggio, G.7
-
16
-
-
0029670659
-
Gamma-aminobutyric acidA receptor regulation: Heterologous uncoupling ofmodulatory site interactions induced by chronic steroid, barbiturate, benzodiazepine, or GABA treatment in culture
-
Friedman LK, Gibbs TT, Farb DH. gamma-aminobutyric acidA receptor regulation: heterologous uncoupling ofmodulatory site interactions induced by chronic steroid, barbiturate, benzodiazepine, or GABA treatment in culture. Brain Res 1996;707:100-9.
-
(1996)
Brain Res
, vol.707
, pp. 100-109
-
-
Friedman, L.K.1
Gibbs, T.T.2
Farb, D.H.3
-
17
-
-
0021240080
-
Chronic benzodiazepine treatment decreases postsynaptic GABA sensitivity
-
Gallager DW, Lakoski JM, Gonsalves SF, Rauch SL. Chronic benzodiazepine treatment decreases postsynaptic GABA sensitivity. Nature 1984;308:74-7. (Pubitemid 14130936)
-
(1984)
Nature
, vol.308
, Issue.5954
, pp. 74-77
-
-
Gallager, D.W.1
Lakoski, J.M.2
Gonsalves, R.S.F.S.L.3
-
18
-
-
0030911572
-
Chronic zolpidem treatment alters GABA(A) receptor mRNA levels in the rat cortex
-
Holt RA, Bateson AN, Martin IL. Chronic zolpidem treatment alters GABA(A) receptor mRNA levels in the rat cortex. Eur J Pharmacol 1997;329:129-32.
-
(1997)
Eur J Pharmacol
, vol.329
, pp. 129-132
-
-
Holt, R.A.1
Bateson, A.N.2
Martin, I.L.3
-
19
-
-
0028350779
-
Chronic benzodiazepine agonist treatment produces functional uncoupling of the γ-aminobutyric acid-benzodiazepine receptor ionophore complex in cortical neurons
-
Hu XJ, TickuMK. Chronic benzodiazepine agonist treatment reduces functional uncoupling of the recombinant of the γ-aminobutyric acid-benzodiazepine receptor ionophore complex in cortical neurons. Mol Pharmacol 1994;45:618-25. (Pubitemid 24139188)
-
(1994)
Molecular Pharmacology
, vol.45
, Issue.4
, pp. 618-625
-
-
Hu, X.-J.1
Ticku, M.K.2
-
20
-
-
43949093042
-
The role of transcriptional and translational mechanisms in flumazenil-induced up-regulation of recombinant GABA(A) receptors
-
Jazvinšćak Jembrek M, Švob Štrac D, Vlainić J, Peričić D. The role of transcriptional and translational mechanisms in flumazenil-induced up-regulation of recombinant GABA(A) receptors. Neurosci Res 2008;61:234-41.
-
(2008)
Neurosci Res
, vol.61
, pp. 234-241
-
-
Jazvinšćak Jembrek, M.1
Švob Štrac, D.2
Vlainić, J.3
Peričić, D.4
-
24
-
-
0026615268
-
A receptor subunit mRNAs in the rat brain. III. Embryonic and postnatal development
-
A receptor subunit mRNAs in the rat brain. III. Embryonic and postnatal development. J Neurosci 1992;12:4151-72.
-
(1992)
J Neurosci
, vol.12
, pp. 4151-4172
-
-
Laurie, D.J.1
Wisden, W.2
Seeburg, P.H.3
-
25
-
-
79959304002
-
A receptor benzodiazepine binding pocket mediate benzodiazepine efficacy and binding
-
A receptor benzodiazepine binding pocket mediate benzodiazepine efficacy and binding. Mol Pharmacol 2011;80:14-22.
-
(2011)
Mol Pharmacol
, vol.80
, pp. 14-22
-
-
Morlock, E.V.1
Czajkowski, C.2
-
26
-
-
0032779365
-
Enhanced caspase activity during ethanol-induced apoptosis in rat cerebellar granule cells
-
Oberdoerster J, Rabin RA. Enhanced caspase activity during ethanol-induced apoptosis in rat cerebellar granule cells. Eur J Pharmacol 1999;385:273-82.
-
(1999)
Eur J Pharmacol
, vol.385
, pp. 273-282
-
-
Oberdoerster, J.1
Rabin, R.A.2
-
27
-
-
54049137689
-
International Union of Pharmacology. LXX. Subtypes of gamma-aminobutyric acid(A) receptors: Classification on the basis of subunit composition, pharmacology, and function
-
Olsen RW, Sieghart W. International Union of Pharmacology. LXX. Subtypes of gamma-aminobutyric acid(A) receptors: classification on the basis of subunit composition, pharmacology, and function. Pharmacol Rev 2008;60:243-60.
-
(2008)
Pharmacol Rev
, vol.60
, pp. 243-260
-
-
Olsen, R.W.1
Sieghart, W.2
-
28
-
-
7544248891
-
A receptors to benzodiazepine antagonist flumazenil enhances the maximum number of benzodiazepine binding sites
-
DOI 10.1016/j.lfs.2004.07.013, PII S0024320504008148
-
Peričić D, Lazić J, Jazvinšćak JembrekM, Švob Štrac D, Rajčan I. Chronic exposure of cells expressing recombinant GABAA receptors to benzodiazepine antagonist flumazenil enhances themaximum number of benzodiazepine binding sites. Life Sci 2004;76:303-17. (Pubitemid 39452912)
-
(2004)
Life Sciences
, vol.76
, Issue.3
, pp. 303-317
-
-
Pericic, D.1
Lazic, J.2
Jazvinscak, J.M.3
Svob, S.D.4
Rajcan, I.5
-
29
-
-
12344279095
-
Enhancement of benzodiazepine binding sites following chronic treatment with flumazenil
-
DOI 10.1016/j.ejphar.2004.10.057, PII S0014299904013536
-
Peričić D, Jazvinšćak Jembrek M, Švob Štrac D, Lazić J, Špoljarić IR. Enhancement of benzodiazepine binding sites following chronic treatment with flumazenil. Eur J Pharmacol 2005;507:7-13. (Pubitemid 40126834)
-
(2005)
European Journal of Pharmacology
, vol.507
, Issue.1-3
, pp. 7-13
-
-
Pericic, D.1
Jazvinscak, J.M.2
Svob, S.D.3
Lazic, J.4
Spoljaric, I.R.5
-
30
-
-
34047132216
-
A receptors
-
DOI 10.1007/s00210-007-0152-z
-
Peričić D, Švob Štrac D, Jazvinš ćak Jembrek M, Vlainić J. Allosteric uncoupling and upregulation of benzodiazepine and GABA recognition sites following chronic diazepam treatment of HEK 293 cells stably transfected with alpha1beta2gamma2S subunits of GABA(A) receptors. Naunyn Schmiedebergs Arch Pharmacol 2007;375:177-87. (Pubitemid 46525450)
-
(2007)
Naunyn-Schmiedeberg's Archives of Pharmacology
, vol.375
, Issue.3
, pp. 177-187
-
-
Pericic, D.1
Strac, D.S.2
Jembrek, M.J.3
Vlainic, J.4
-
31
-
-
46549084825
-
Sedative and anticonvulsant effects of zolpidem in adult and aged mice
-
Peričić D, Vlainić J, Švob Štrac D. Sedative and anticonvulsant effects of zolpidem in adult and aged mice. J Neural Transm 2008;115:795-802.
-
(2008)
J Neural Transm
, vol.115
, pp. 795-802
-
-
Peričić, D.1
Vlainić, J.2
Švob Štrac, D.3
-
32
-
-
0026768488
-
Lack of tolerance and physical dependence upon repeated treatment with the novel hypnotic zolpidem
-
Perrault G, Morel E, Sanger DJ, Zivkovic B. Lack of tolerance and physical dependence upon repeated treatment with the novel hypnotic zolpidem. J Pharmacol Exp Ther 1992;263:298-303.
-
(1992)
J Pharmacol Exp Ther
, vol.263
, pp. 298-303
-
-
Perrault, G.1
Morel, E.2
Sanger, D.J.3
Zivkovic, B.4
-
35
-
-
0025195928
-
γ-Aminobutyric acid(A) receptor regulation in culture: Altered allosteric interactions following prolonged exposure to benzodiazepnes, barbiturates, and methylxanthines
-
Roca DJ, Schiller GD, Friedman L, Rozenberg I, Gibbs TT, Farb DH. γ-Aminobutyric acidA receptor regulation in culture: altered allosteric interactions following prolonged exposure to benzodiazepines, barbiturates, and methylxanthines. Mol Pharmacol 1990;37:710-9. (Pubitemid 20171507)
-
(1990)
Molecular Pharmacology
, vol.37
, Issue.5
, pp. 710-719
-
-
Roca, D.J.1
Schiller, G.D.2
Friedman, L.3
Rozenberg, I.4
Gibbs, T.T.5
Farb, D.H.6
-
36
-
-
0030579072
-
Comparison of the pharmacological profiles of the hypnotic drugs, zaleplon and zolpidem
-
DOI 10.1016/0014-2999(96)00510-9
-
Sanger DJ, Morel E, Perrault G. Comparison of the pharmacological profiles of the hypnotic drugs, zaleplon and zolpidem. Eur J Pharmacol 1996;313:35-42. (Pubitemid 26342203)
-
(1996)
European Journal of Pharmacology
, vol.313
, Issue.1-2
, pp. 35-42
-
-
Sanger, D.J.1
Morel, E.2
Perrault, G.3
-
37
-
-
0037072577
-
A receptor subtypes
-
DOI 10.1016/S0014-2999(02)02191-X, PII S001429990202191X
-
Sanna E, Busonero F, Talani G, Carta M, Massa F, Peis M, et al. Comparison of the effects of zaleplon, zolpidem, and triazolam at various GABA(A) receptor subtypes. Eur J Pharmacol 2002;451:103-10. (Pubitemid 35253948)
-
(2002)
European Journal of Pharmacology
, vol.451
, Issue.2
, pp. 103-110
-
-
Sanna, E.1
Busonero, F.2
Talani, G.3
Carta, M.4
Massa, F.5
Peis, M.6
Maciocco, E.7
Biggio, G.8
-
38
-
-
0036618178
-
Preferential transformation of human neuronal cells by human adenoviruses and the origin of HEK 293 cells
-
Shaw G, Morse S, Ararat M, Graham FL. Preferential transformation of human neuronal cells by human adenoviruses and the origin of HEK 293 cells. FASEB J 2002;16:869-71.
-
(2002)
FASEB J
, vol.16
, pp. 869-871
-
-
Shaw, G.1
Morse, S.2
Ararat, M.3
Graham, F.L.4
-
39
-
-
0028981088
-
Structure and pharmacology of γ-aminobutyric acidA receptor subtypes
-
Sieghart W. Structure and pharmacology of γ-aminobutyric acidA receptor subtypes. Pharmacol Rev 1995;47:181-234.
-
(1995)
Pharmacol Rev
, vol.47
, pp. 181-234
-
-
Sieghart, W.1
-
40
-
-
57249095716
-
Differential effects of diazepam treatment and withdrawal on recombinant GABAA receptor expression and functional coupling
-
Švob Štrac D, Vlainić J, Jazvinšćak Jembrek M, Peričić D. Differential effects of diazepam treatment and withdrawal on recombinant GABAA receptor expression and functional coupling. Brain Res 2008;1246:29-40.
-
(2008)
Brain Res
, vol.1246
, pp. 29-40
-
-
Švob Štrac, D.1
Vlainić, J.2
Jazvinšćak Jembrek, M.3
Peričić, D.4
-
41
-
-
77949392957
-
A receptor subunit expression by pharmacological agents
-
A receptor subunit expression by pharmacological agents. Pharmacol Rev 2010;62:97-135.
-
(2010)
Pharmacol Rev
, vol.62
, pp. 97-135
-
-
Uusi-Oukari, M.1
Korpi, E.R.2
-
43
-
-
67349227183
-
Effect of acute and repeated zolpidem treatment on pentylenetetrazole- induced seizure threshold and on locomotor activity: Comparison with diazepam
-
Vlainić J, Peričić D. Effect of acute and repeated zolpidem treatment on pentylenetetrazole-induced seizure threshold and on locomotor activity: comparison with diazepam. Neuropharmacology 2009;56:1124-30.
-
(2009)
Neuropharmacology
, vol.56
, pp. 1124-1130
-
-
Vlainić, J.1
Peričić, D.2
-
44
-
-
73149096941
-
Zolpidem is a potent anticonvulsant in adult and aged mice
-
Vlainić J, Peričić D. Zolpidem is a potent anticonvulsant in adult and aged mice. Brain Res 2010;1310:181-8.
-
(2010)
Brain Res
, vol.1310
, pp. 181-188
-
-
Vlainić, J.1
Peričić, D.2
-
45
-
-
77957600516
-
The effects of zolpidem treatment and withdrawal on the in vitro expression of recombinant alpha1beta2gamma2s GABA(A) receptors expressed in HEK 293 cells
-
Vlainić J, Jazvinšćak Jembrek M, Švob Štrac D, Peričić D. The effects of zolpidem treatment and withdrawal on the in vitro expression of recombinant alpha1beta2gamma2s GABA(A) receptors expressed in HEK 293 cells. Naunyn Schmiedebergs Arch Pharmacol 2010;382:201-12.
-
(2010)
Naunyn Schmiedebergs Arch Pharmacol
, vol.382
, pp. 201-212
-
-
Vlainić, J.1
Jazvinšćak Jembrek, M.2
Švob Štrac, D.3
Peričić, D.4
-
46
-
-
12344260655
-
A receptor subtypes: Any clues to the mechanism of benzodiazepine dependence?
-
A receptor subtypes: any clues to the mechanism of benzodiazepine dependence? Curr Opin Pharmacol 2005;5:47-52.
-
(2005)
Curr Opin Pharmacol
, vol.5
, pp. 47-52
-
-
Wafford, K.A.1
-
47
-
-
0028970627
-
NMDA-mediated modulation of gamma-aminobutyric acid type A receptor function in cerebellar granule neurons
-
Zhu WJ, Vicini S, Harris BT, Grayson DR. NMDA-mediated modulation of gamma-aminobutyric acid type A receptor function in cerebellar granule neurons. J Neurosci 1995;15:7692-701. (Pubitemid 3010101)
-
(1995)
Journal of Neuroscience
, vol.15
, Issue.11
, pp. 7692-7701
-
-
Zhu, W.J.1
Vicini, S.2
Harris, B.T.3
Grayson, D.R.4
|