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Volumn 3, Issue 4, 2012, Pages 469-474

Novel selective inhibitors of neutral endopeptidase: Discovery by screening and hit-to-lead optimisation

(10) El Bakali, Jamal a,b Maingot, Lucie a,b Dumont, Julie a,b Host, Helene a,b Hocine, Akila a,b Cousaert, Nicolas a,b Dassonneville, Sandrine a,b Leroux, Florence a,b Deprez, Benoit a,b Deprez Poulain, Rebecca a,b

a UNIV LILLE (France)

b PRIM Pôle de Recherche Interdisciplinaire sur le Médicament (France)

Author keywords

[No Author keywords available]

Indexed keywords

CARBOXYLIC ACID DERIVATIVE; ENKEPHALINASE INHIBITOR; MEMBRANE METALLOENDOPEPTIDASE;

ARTICLE; DRUG IDENTIFICATION; DRUG SCREENING; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION; MOLECULAR WEIGHT; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION;

EID: 84859416116 PISSN: 20402503 EISSN: 20402511 Source Type: Journal
DOI: 10.1039/c2md00287f Document Type: Article

Times cited : (3)

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