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Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 7, 2012, Pages 2635-2639

2-Amidino analogs of glycine-amiloride conjugates: Inhibitors of urokinase-type plasminogen activator

(5) Massey, Archna P a Harley, William R b Pasupuleti, Nagarekha b Gorin, Fredric A b Nantz, Michael H a

a UNIVERSITY OF LOUISVILLE (United States)

b UNIVERSITY OF CALIFORNIA (United States)

Author keywords

Lactate dehydrogenase; Plasminogen activator inhibitor protein 1; Tissue plasminogen activator; Urokinase type plasminogen activator; Urokinase type plasminogen activator receptor

Indexed keywords

AMIDINE; AMILORIDE; AMILORIDE DERIVATIVE; GLYCINE; UROKINASE;

ARTICLE; CANCER CELL; CONJUGATE; CYTOTOXICITY; ENZYME INHIBITION; GLIOBLASTOMA; HUMAN; HUMAN CELL; HYDROPHOBICITY; IC 50; SUBSTITUTION REACTION;

AMIDINES; AMILORIDE; ANTINEOPLASTIC AGENTS; CELL LINE, TUMOR; CELL SURVIVAL; DRUG SCREENING ASSAYS, ANTITUMOR; GLYCINE; HUMANS; HYDROPHOBIC AND HYDROPHILIC INTERACTIONS; SERINE PROTEINASE INHIBITORS; STRUCTURE-ACTIVITY RELATIONSHIP; TISSUE PLASMINOGEN ACTIVATOR; UROKINASE-TYPE PLASMINOGEN ACTIVATOR;

EID: 84858700139 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2011.12.123 Document Type: Article

Times cited : (7)

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