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Volumn 8, Issue 4, 2012, Pages 307-316

Risperidone release from Solid Lipid Nanoparticles (SLN): Validated HPLC method and modelling kinetic profile

Author keywords

Controlled drug release; Encapsulation efficiency; Encapsulation parameters; High performance liquid chromatography; Kinetic model; Loading capacity; Oral drug delivery; Release profile; Risperidone; Solid lipid nanoparticles

Indexed keywords

DEOXYCHOLATE SODIUM; GLYCEROL STEARATE; IMWITOR; MACROGOL DERIVATIVE; RISPERIDONE; SOLID LIPID NANOPARTICLE; TAGAT S; UNCLASSIFIED DRUG;

EID: 84857786253     PISSN: 15734129     EISSN: 1875676X     Source Type: Journal    
DOI: 10.2174/157341212803341663     Document Type: Article
Times cited : (29)

References (40)
  • 1
    • 84867807788 scopus 로고    scopus 로고
    • The United States Pharmacopeia, United States Pharmacopeial Convention: Rockville, MD
    • The United States Pharmacopeia, United States Pharmacopeia/The National Formulary United States Pharmacopeial Convention: Rockville, MD, 2008.
    • (2008) United States Pharmacopeia/The National Formulary
  • 2
    • 0842263782 scopus 로고    scopus 로고
    • A review of compliance, depot intramuscular antipsychotics and the new longacting injectable atypical antipsychotic risperidone in schizophrenia
    • Bhanji, N.H.; Chouinard, G.; Margolese, H.C. A review of compliance, depot intramuscular antipsychotics and the new longacting injectable atypical antipsychotic risperidone in schizophrenia. Eur. Neuropsychopharmacol 2004, 14 87-92.
    • (2004) Eur. Neuropsychopharmacol , vol.14 , pp. 87-92
    • Bhanji, N.H.1    Chouinard, G.2    Margolese, H.C.3
  • 3
    • 8744234074 scopus 로고    scopus 로고
    • Acceptability and disintegration rates of orally disintegrating risperidone tablets in patients with schizophrenia or schizoaffective disorder
    • Chue, P.; Welch, R.; Binder, C. Acceptability and disintegration rates of orally disintegrating risperidone tablets in patients with schizophrenia or schizoaffective disorder. Can. J. Psychiatry 2004, 49 701-703.
    • (2004) Can. J. Psychiatry , vol.49 , pp. 701-703
    • Chue, P.1    Welch, R.2    Binder, C.3
  • 4
    • 34547524961 scopus 로고    scopus 로고
    • Do formulation switches exacerbate existing medical illness? Results of an open-label transition to orally disintegrating risperidone tablets
    • Chue, P.; Prinzo, R.S.; Binder, C.E. Do formulation switches exacerbate existing medical illness? Results of an open-label transition to orally disintegrating risperidone tablets. Hum. Psychopharmacol 2007, 22 307-314.
    • (2007) Hum. Psychopharmacol , vol.22 , pp. 307-314
    • Chue, P.1    Prinzo, R.S.2    Binder, C.E.3
  • 5
    • 44449106460 scopus 로고    scopus 로고
    • Intranasal nanoemulsion based brain targeting drug delivery system of risperidone
    • Kumar, M.; Misra, A.; Babbar, A.K.; Mishra, A.K.; Mishra, P.; Pathak, K. Intranasal nanoemulsion based brain targeting drug delivery system of risperidone. Int. J. Pharm. 2008, 358(1-2), 285-291.
    • (2008) Int. J. Pharm. , vol.358 , Issue.1-2 , pp. 285-291
    • Kumar, M.1    Misra, A.2    Babbar, A.K.3    Mishra, A.K.4    Mishra, P.5    Pathak, K.6
  • 6
    • 0028948839 scopus 로고
    • A theoretical basis for a biopharmaceutic drug classification: The correlation of in vivo drug product dissolution and in vivo bioavailability
    • Amidon, G.L.; Lennernas, H.; Shah, V.P.; Crison, J.R. A theoretical basis for a biopharmaceutic drug classification: the correlation of in vivo drug product dissolution and in vivo bioavailability. Pharm. Res 1995, 12 413-420.
    • (1995) Pharm. Res , vol.12 , pp. 413-420
    • Amidon, G.L.1    Lennernas, H.2    Shah, V.P.3    Crison, J.R.4
  • 7
    • 0035073301 scopus 로고    scopus 로고
    • Modeling and comparison of dissolution profiles
    • Costa, P.; Sousa Lobo, J.M. Modeling and comparison of dissolution profiles. Eur. J. Pharm. Sci. 2001, 13 123-133.
    • (2001) Eur. J. Pharm. Sci. , vol.13 , pp. 123-133
    • Costa, P.1    Sousa Lobo, J.M.2
  • 8
    • 4544275025 scopus 로고    scopus 로고
    • Challenges and solutions for the delivery of biotech drugs-a review of drug nanocrystal technology and lipid nanoparticles
    • Muller, R.H.; Keck, C.M. Challenges and solutions for the delivery of biotech drugs-a review of drug nanocrystal technology and lipid nanoparticles. J Biotechnol 2004, 113 151-170.
    • (2004) J Biotechnol , vol.113 , pp. 151-170
    • Muller, R.H.1    Keck, C.M.2
  • 9
    • 33751014029 scopus 로고    scopus 로고
    • Formulation of poorly water-soluble drugs for oral administration: Physicochemical and physiological issues and the lipid formulation classification system
    • Pouton, C.W. Formulation of poorly water-soluble drugs for oral administration: physicochemical and physiological issues and the lipid formulation classification system. Eur. J. Pharm. Sci. 2006, 29 278-287.
    • (2006) Eur. J. Pharm. Sci. , vol.29 , pp. 278-287
    • Pouton, C.W.1
  • 10
    • 34548049221 scopus 로고    scopus 로고
    • Oral lipid-based formulations
    • Hauss, D.J. Oral lipid-based formulations. Adv. Drug Deliv. Rev 2007, 59 667-676.
    • (2007) Adv. Drug Deliv. Rev , vol.59 , pp. 667-676
    • Hauss, D.J.1
  • 11
    • 79956102907 scopus 로고    scopus 로고
    • 20 Years of lipid nanoparticles (SLN and NLC): Present state of development and industrial applications
    • Muller, R.H.; Shegokar, R.; Keck, C.M. 20 Years of lipid nanoparticles (SLN and NLC): present state of development and industrial applications. Curr. Drug Discov. Technol 2011, 8(3), 207-27.
    • (2011) Curr. Drug Discov. Technol , vol.8 , Issue.3 , pp. 207-227
    • Muller, R.H.1    Shegokar, R.2    Keck, C.M.3
  • 12
    • 77953283407 scopus 로고    scopus 로고
    • Lipid nanoparticles: Effect on bioavailability and pharmacokinetic changes
    • Souto, E.B.; Muller, R.H. Lipid nanoparticles: effect on bioavailability and pharmacokinetic changes. Handb. Exp. Pharmacol 2011, 197 115-141.
    • (2011) Handb. Exp. Pharmacol , vol.197 , pp. 115-141
    • Souto, E.B.1    Muller, R.H.2
  • 13
    • 79954417472 scopus 로고    scopus 로고
    • Recent advances in lipid nanoparticle formulations with solid matrix for oral drug delivery
    • Das, S.; Chaudhury, A. Recent advances in lipid nanoparticle formulations with solid matrix for oral drug delivery. AAPS PharmSciTech 2010, 12 62-76.
    • (2010) AAPS PharmSciTech , vol.12 , pp. 62-76
    • Das, S.1    Chaudhury, A.2
  • 14
    • 18144423086 scopus 로고    scopus 로고
    • Validation in pharmaceutical analysis. Part II: Central importance of precision to establish acceptance criteria and for verifying and improving the quality of analytical data
    • Ermer, J.; Ploss, H.J. Validation in pharmaceutical analysis. Part II: central importance of precision to establish acceptance criteria and for verifying and improving the quality of analytical data. J. Pharm. Biomed. Anal 2005, 37 859-870.
    • (2005) J. Pharm. Biomed. Anal , vol.37 , pp. 859-870
    • Ermer, J.1    Ploss, H.J.2
  • 15
    • 84889460543 scopus 로고    scopus 로고
    • Method Validation
    • Kazakevich, Y.; LoBrutto, R.; Eds.; John Wiley & Sons: New York
    • LoBrutto, R.; Patel, T. Method Validation, In: HPLC for Pharmaceutical Scientists Kazakevich, Y.; LoBrutto, R.; Eds.; John Wiley & Sons: New York, 2007, pp. 455-502.
    • (2007) HPLC for Pharmaceutical Scientists , pp. 455-502
    • Lo Brutto, R.1    Patel, T.2
  • 16
    • 0035097208 scopus 로고    scopus 로고
    • Validation in pharmaceutical analysis. Part I: An integrated approach
    • Ermer, J. Validation in pharmaceutical analysis. Part I: an integrated approach. J. Pharm. Biomed. Anal 2001, 24 755-767.
    • (2001) J. Pharm. Biomed. Anal , vol.24 , pp. 755-767
    • Ermer, J.1
  • 18
    • 11144256427 scopus 로고    scopus 로고
    • High p4 erformance liquid chromatographic and thin layer densitometric methods for the determination of risperidone in the presence of its degradation products in bulk powder and in tablets
    • El-Sherif, Z.A.; El-Zeany, B.; El-Houssini, O.M. High p4 erformance liquid chromatographic and thin layer densitometric methods for the determination of risperidone in the presence of its degradation products in bulk powder and in tablets. J. Pharm. Biomed. Anal 2005, 36 975-981.
    • (2005) J. Pharm. Biomed. Anal , vol.36 , pp. 975-981
    • El-Sherif, Z.A.1    El-Zeany, B.2    El-Houssini, O.M.3
  • 19
    • 78650160677 scopus 로고    scopus 로고
    • Dose-related effects of clozapine and risperidone on the pattern of brain regional serotonin and dopamine metabolism and on tests related to extrapyramidal functions in rats
    • Batool, F.; Hasnat, A.; Haleem, M.A.; Haleem, D.J. Dose-related effects of clozapine and risperidone on the pattern of brain regional serotonin and dopamine metabolism and on tests related to extrapyramidal functions in rats. Acta Pharm. 2010, 60 129-140.
    • (2010) Acta Pharm. , vol.60 , pp. 129-140
    • Batool, F.1    Hasnat, A.2    Haleem, M.A.3    Haleem, D.J.4
  • 20
    • 34548132384 scopus 로고    scopus 로고
    • Simultaneous determination of five antipsychotic drugs in rat plasma by high performance liquid chromatography with ultraviolet detection
    • Zhang, G.; Terry, A.V. Jr.; Bartlett, M.G. Simultaneous determination of five antipsychotic drugs in rat plasma by high performance liquid chromatography with ultraviolet detection. J. Chromatogr. B Analyt Technol. Biomed. Life Sci. 2007, 856 20-28.
    • (2007) J. Chromatogr. B Analyt Technol. Biomed. Life Sci. , vol.856 , pp. 20-28
    • Zhang, G.1    Terry Jr., A.V.2    Bartlett, M.G.3
  • 23
    • 65749099862 scopus 로고    scopus 로고
    • Formulation and characterization of nanoemulsion-based drug delivery system of risperidone
    • Kumar, M.; Pathak, K.; Misra, A. Formulation and characterization of nanoemulsion-based drug delivery system of risperidone. Drug Dev. Ind. Pharm 2009, 35 387-395.
    • (2009) Drug Dev. Ind. Pharm , vol.35 , pp. 387-395
    • Kumar, M.1    Pathak, K.2    Misra, A.3
  • 24
    • 69249232376 scopus 로고    scopus 로고
    • PLGA nanoparticle formulations of risperidone: Preparation and neuropharmacological evaluation
    • Muthu, M.S.; Rawat, M.K.; Mishra, A.; Singh, S. PLGA nanoparticle formulations of risperidone: preparation and neuropharmacological evaluation. Nanomedicine 2009, 5 323-333.
    • (2009) Nanomedicine , vol.5 , pp. 323-333
    • Muthu, M.S.1    Rawat, M.K.2    Mishra, A.3    Singh, S.4
  • 25
    • 61849094331 scopus 로고    scopus 로고
    • Poly (D, L-lactide) nanosuspensions of risperidone for parenteral delivery: Formulation and in-vitro evaluation
    • Muthu, M.S.; Singh, S. Poly (D, L-lactide) nanosuspensions of risperidone for parenteral delivery: formulation and in-vitro evaluation. Curr. Drug Deliv 2009, 6 62-68.
    • (2009) Curr. Drug Deliv , vol.6 , pp. 62-68
    • Muthu, M.S.1    Singh, S.2
  • 26
    • 0026474637 scopus 로고
    • Determination of risperidone and 9-hydroxyrisperidone in plasma, urine and animal tissues by high-performance liquid chromatography
    • Woestenborghs, R.; Lorreyne, W.; Van Rompaey, F.; Heykants, J. Determination of risperidone and 9-hydroxyrisperidone in plasma, urine and animal tissues by high-performance liquid chromatography. J. Chromatogr 1992, 583 223-230.
    • (1992) J. Chromatogr , vol.583 , pp. 223-230
    • Woestenborghs, R.1    Lorreyne, W.2    van Rompaey, F.3    Heykants, J.4
  • 27
    • 79955794727 scopus 로고    scopus 로고
    • Preparation, characterization and biocompatibility studies on risperidone-loaded solid lipid nanoparticles (SLN): High pressure homogenization versus ultrasound
    • Silva, A.C.; Gonzalez-Mira, E.; Garcia, M.L.; Egea, M.A.; Fonseca, J.; Silva, R.; Santos, D.; Souto, E.B.; Ferreira, D. Preparation, characterization and biocompatibility studies on risperidone-loaded solid lipid nanoparticles (SLN): High pressure homogenization versus ultrasound. Colloids Surf. B Biointerfaces 2011, 86 158-165.
    • (2011) Colloids Surf. B Biointerfaces , vol.86 , pp. 158-165
    • Silva, A.C.1    Gonzalez-Mira, E.2    Garcia, M.L.3    Egea, M.A.4    Fonseca, J.5    Silva, R.6    Santos, D.7    Souto, E.B.8    Ferreira, D.9
  • 28
    • 34247538000 scopus 로고    scopus 로고
    • Cavitation-a novel technique for making stable nano-suspensions
    • Patil, M.N.; Pandit, A.B. Cavitation-a novel technique for making stable nano-suspensions. Ultrason. Sonochem 2007, 14 519-530.
    • (2007) Ultrason. Sonochem , vol.14 , pp. 519-530
    • Patil, M.N.1    Pandit, A.B.2
  • 29
    • 0038032150 scopus 로고    scopus 로고
    • Solid lipid nanoparticles (SLN) for controlled drug delivery-a review of the state of the art
    • Muller, R.H.; Mader, K.; Gohla, S. Solid lipid nanoparticles (SLN) for controlled drug delivery-a review of the state of the art. Eur. J. Pharm. Biopharm., 2000, 50 161-177.
    • (2000) Eur. J. Pharm. Biopharm. , vol.50 , pp. 161-177
    • Muller, R.H.1    Mader, K.2    Gohla, S.3
  • 30
    • 77953356716 scopus 로고    scopus 로고
    • Optimization and physicochemical characterization of a triamcinolone acetonide-loaded NLC for ocular antiangiogenic applications
    • Araujo, J.; Gonzalez-Mira, E.; Egea, M.A.; Garcia, M.L.; Souto, E.B. Optimization and physicochemical characterization of a triamcinolone acetonide-loaded NLC for ocular antiangiogenic applications. Int. J. Pharm. 2010, 393 167-175.
    • (2010) Int. J. Pharm. , vol.393 , pp. 167-175
    • Araujo, J.1    Gonzalez-Mira, E.2    Egea, M.A.3    Garcia, M.L.4    Souto, E.B.5
  • 31
    • 79251585943 scopus 로고    scopus 로고
    • Optimizing flurbiprofen-loaded NLC by central composite factorial design for ocular delivery
    • Gonzalez-Mira, E.; Egea, M.A.; Souto, E.B.; Calpena, A.C.; Garcia, M.L. Optimizing flurbiprofen-loaded NLC by central composite factorial design for ocular delivery. Nanotechnology 2011, 22(4), 045101.
    • (2011) Nanotechnology , vol.22 , Issue.4 , pp. 045101
    • Gonzalez-Mira, E.1    Egea, M.A.2    Souto, E.B.3    Calpena, A.C.4    Garcia, M.L.5
  • 32
    • 35448977211 scopus 로고    scopus 로고
    • Investigations of the effect of the lipid matrix on drug entrapment, in vivo release, and physical stability of olanzapine-loaded solid lipid nanoparticles
    • Vivek, K.; Reddy, H.; Murthy, R.S. Investigations of the effect of the lipid matrix on drug entrapment, in vivo release, and physical stability of olanzapine-loaded solid lipid nanoparticles. AAPS PharmSciTech 2007, 8(4), E83.
    • (2007) AAPS PharmSciTech , vol.8 , Issue.4
    • Vivek, K.1    Reddy, H.2    Murthy, R.S.3
  • 33
    • 0031913402 scopus 로고    scopus 로고
    • Dissolution testing as a prognostic tool for oral drug absorption: Immediate release dosage forms
    • Dressman, J.B.; Amidon, G.L.; Reppas, C.; Shah, V.P. Dissolution testing as a prognostic tool for oral drug absorption: immediate release dosage forms. Pharm. Res 1998, 15 11-22.
    • (1998) Pharm. Res , vol.15 , pp. 11-22
    • Dressman, J.B.1    Amidon, G.L.2    Reppas, C.3    Shah, V.P.4
  • 34
    • 0037435988 scopus 로고    scopus 로고
    • Validation of high-performance liquid chromatography methods for pharmaceutical analysis. Understanding the differences and similarities between validation requirements of the US Food and Drug Administration, the US Pharmacopeia and the International Conference on Harmonization
    • Shabir, G.A. Validation of high-performance liquid chromatography methods for pharmaceutical analysis. Understanding the differences and similarities between validation requirements of the US Food and Drug Administration, the US Pharmacopeia and the International Conference on Harmonization. J. Chromatogr. A 2003, 987 57-66.
    • (2003) J. Chromatogr. A , vol.987 , pp. 57-66
    • Shabir, G.A.1
  • 35
    • 33744973517 scopus 로고    scopus 로고
    • Oral bioavailability of cyclosporine: Solid lipid nanoparticles (SLN) versus drug nanocrystals
    • Muller, R.H.; Runge, S.; Ravelli, V.; Mehnert, W.; Thunemann, A.F.; Souto, E.B. Oral bioavailability of cyclosporine: solid lipid nanoparticles (SLN) versus drug nanocrystals. Int. J. Pharm. 2006, 317 82-89.
    • (2006) Int. J. Pharm. , vol.317 , pp. 82-89
    • Muller, R.H.1    Runge, S.2    Ravelli, V.3    Mehnert, W.4    Thunemann, A.F.5    Souto, E.B.6
  • 36
    • 39849097998 scopus 로고    scopus 로고
    • Cyclosporine-loaded solid lipid nanoparticles (SLN): Drug-lipid physicochemical interactions and characterization of drug incorporation
    • Muller, R.H.; Runge, S.A.; Ravelli, V.; Thunemann, A.F.; Mehnert, W.; Souto, E.B. Cyclosporine-loaded solid lipid nanoparticles (SLN): drug-lipid physicochemical interactions and characterization of drug incorporation. Eur. J. Pharm. Biopharm 2008, 68 535-544.
    • (2008) Eur. J. Pharm. Biopharm , vol.68 , pp. 535-544
    • Muller, R.H.1    Runge, S.A.2    Ravelli, V.3    Thunemann, A.F.4    Mehnert, W.5    Souto, E.B.6
  • 37
    • 57349171371 scopus 로고    scopus 로고
    • Lipid nanoparticles with a solid matrix (SLN, NLC, LDC) for oral drug delivery
    • Muchow, M.; Maincent, P.; Muller, R.H. Lipid nanoparticles with a solid matrix (SLN, NLC, LDC) for oral drug delivery. Drug Dev. Ind. Pharm. 2008, 34 1394-1405.
    • (2008) Drug Dev. Ind. Pharm. , vol.34 , pp. 1394-1405
    • Muchow, M.1    Maincent, P.2    Muller, R.H.3
  • 38
    • 67549110065 scopus 로고    scopus 로고
    • Diazepam-loaded solid lipid nanoparticles: Design and characterization
    • Abdelbary, G.; Fahmy, R.H. Diazepam-loaded solid lipid nanoparticles: design and characterization. AAPS PharmSciTech 2009, 10 211-219.
    • (2009) AAPS PharmSciTech , vol.10 , pp. 211-219
    • Abdelbary, G.1    Fahmy, R.H.2
  • 39
    • 0023195932 scopus 로고
    • A simple equation for description of solute release I. Fickian and non-fickian release from non-swellable devices in the form of slabs, spheres, cylinders or discs
    • Ritger, P.L.; Peppas, N.A. A simple equation for description of solute release I. Fickian and non-fickian release from non-swellable devices in the form of slabs, spheres, cylinders or discs. J. Control. Release 1987, 5 23-36.
    • (1987) J. Control. Release , vol.5 , pp. 23-36
    • Ritger, P.L.1    Peppas, N.A.2
  • 40
    • 0023196815 scopus 로고
    • A simple equation for description of solute release II. Fickian and anomalous release from swellable devices
    • Ritger, P.L.; Peppas, N.A. A simple equation for description of solute release II. Fickian and anomalous release from swellable devices. J. Control. Release 1987, 5 37-42.
    • (1987) J. Control. Release , vol.5 , pp. 37-42
    • Ritger, P.L.1    Peppas, N.A.2


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