Biodistribution, toxicology, and radiation dosimetry of 5-HT 1A-receptor agonist positron emission tomography ligand [ 11C]CUMI-101

International Journal of Toxicology

Volumn 30, Issue 6, 2011, Pages 611-618

  Kumar, Dileep J S ^a,b   Bai, Bing ^a   Ng, Hanna H ^c   Mirsalis, Jon C ^c   Erlandsson, Kjell ^a   Milak, Matthew S ^a,b   Majo, Vattoly J ^a   Prabhakaran, Jaya ^a   Mann, J J ^a,b   Parsey, R V ^a,b  

^a Department of Medicine   (United States)

^b NEW YORK STATE PSYCHIATRIC INSTITUTE   (United States)

^c SRI INTERNATIONAL   (United States)

Author keywords

Dosimetry; PET; Radioligand; Toxicity

Indexed keywords

[O METHYL C 11] 2 [4 [4 (2 METHOXYPHENYL)PIPERAZIN 1 YL]BUTYL] 4 METHYL 1,2,4 TRIAZINE 3,5(2H,4H)DIONE; SEROTONIN 1 RECEPTOR; SEROTONIN 1A AGONIST; TRACER; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ARTICLE; BLADDER; CONTROLLED STUDY; DOSIMETRY; DRUG TOLERABILITY; FEMALE; MALE; MAXIMUM TOLERATED DOSE; NONHUMAN; POSITRON EMISSION TOMOGRAPHY; RADIATION DOSE; RAT; TESTIS;

ANIMALS; CARBON RADIOISOTOPES; FEMALE; LIGANDS; MALE; PAPIO; PIPERAZINES; POSITRON-EMISSION TOMOGRAPHY; RADIOMETRY; RATS; RATS, SPRAGUE-DAWLEY; SEROTONIN 5-HT1 RECEPTOR AGONISTS; TISSUE DISTRIBUTION; TRIAZINES;

PAPIO; RATTUS;

EID: 84856904485     PISSN: 10915818     EISSN: 1092874X     Source Type: Journal    
DOI: 10.1177/1091581811419024     Document Type: Article

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