F15599, a novel 5-HT1A receptor agonist, as a radioligand for PET neuroimaging

European Journal of Nuclear Medicine and Molecular Imaging

Volumn 37, Issue 3, 2010, Pages 594-605

  Lemoine, Laëtitia ^a,b   Verdurand, Mathieu ^a,b   Vacher, Bernard ^c   Blanc, Elodie ^c   Le Bars, Didier ^b   Newman Tancredi, Adrian ^c   Zimmer, Luc ^a,b  

^a UNIVERSITÉ DE LYON   (France)

^b CERMEP IMAGERIE DU VIVANT   (France)

^c INSTITUT DE RECHERCHE PIERRE FABRE   (France)

Author keywords

Agonist; Cat; PET; Rat; Serotonin 1A receptor

Indexed keywords

3 CHLORO 4 FLUOROPHENYL[(4 FLUORO 4(((5 METHYL PYRIMIDIN 2 YLMETHYL) AMINO) METHY)) PIPERIDIN 1 YL] METHANONE F18; G PROTEIN COUPLED RECEPTOR; RADIOLIGAND; SEROTONIN AGONIST; UNCLASSIFIED DRUG; 3 CHLORO 4 FLUOROPHENYL (4 FLUORO 4 (((5 METHYLPYRIMIDIN 2 YLMETHYL)AMINO)METHYL)PIPERIDIN 1 YL)METHANONE; 3-CHLORO-4-FLUOROPHENYL-(4-FLUORO-4-(((5-METHYLPYRIMIDIN-2-YLMETHYL)AMINO)METHYL)PIPERIDIN-1-YL)METHANONE; DIAGNOSTIC AGENT; FLUORINE; LIGAND; PIPERIDINE DERIVATIVE; PYRIMIDINE DERIVATIVE; SEROTONIN 1A RECEPTOR;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BRAIN CORTEX; CONTROLLED STUDY; EXPERIMENTAL CAT; MALE; NEUROIMAGING; NONHUMAN; POSITRON EMISSION TOMOGRAPHY; RAT; ANIMAL; AUTORADIOGRAPHY; BINDING COMPETITION; BRAIN; CAT; CHEMISTRY; DISSECTION; DRUG POTENTIATION; METABOLISM; PATHOLOGY; SCINTISCANNING;

ANIMALS; AUTORADIOGRAPHY; BINDING, COMPETITIVE; BRAIN; CATS; DISSECTION; FLUORINE RADIOISOTOPES; LIGANDS; MALE; PIPERIDINES; POSITRON-EMISSION TOMOGRAPHY; PYRIMIDINES; RATS; RECEPTOR, SEROTONIN, 5-HT1A; SEROTONIN AGONISTS;

EID: 77949261526     PISSN: 16197070     EISSN: None     Source Type: Journal    
DOI: 10.1007/s00259-009-1274-y     Document Type: Article

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