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Volumn 61, Issue , 2012, Pages 184-190

Chromatography approaches for early screening of the phospholipidosis-inducing potential of pharmaceuticals

Author keywords

Drug phospholipidosis inducing potential; Phospholipidosis; Surfactant vesicle electrokinetic chromatography; Volume of distribution

Indexed keywords

AMIODARONE; AMITRIPTYLINE; AMPICILLIN; ATENOLOL; ATROPINE; CHLOROQUINE; CLOMIPRAMINE; DIAZEPAM; DISOPYRAMIDE; DOCUSATE SODIUM; FAMOTIDINE; FLUOXETINE; FUROSEMIDE; IMIPRAMINE; KETOPROFEN; LABETALOL; LIDOCAINE; MAPROTILINE; MEPACRINE; MIANSERIN; OCTANOL; PARACETAMOL; PROCAINE; PROPRANOLOL; QUINIDINE; TAMOXIFEN; TETRACYCLINE; UNINDEXED DRUG; WARFARIN; ZIMELDINE;

EID: 84856101453     PISSN: 07317085     EISSN: 1873264X     Source Type: Journal    
DOI: 10.1016/j.jpba.2011.11.033     Document Type: Article
Times cited : (30)

References (44)
  • 1
    • 33749042117 scopus 로고    scopus 로고
    • Drug-induced phospholipidosis
    • Anderson N., Borlak J. Drug-induced phospholipidosis. FEBS Lett. 2006, 580:5533-5540.
    • (2006) FEBS Lett. , vol.580 , pp. 5533-5540
    • Anderson, N.1    Borlak, J.2
  • 2
    • 0035687129 scopus 로고    scopus 로고
    • Drug-induced phospholipidosis: are there functional consequences?
    • Reasor M.J., Kacew S. Drug-induced phospholipidosis: are there functional consequences?. Exp. Biol. Med. 2001, 226:825-830.
    • (2001) Exp. Biol. Med. , vol.226 , pp. 825-830
    • Reasor, M.J.1    Kacew, S.2
  • 3
    • 0025572278 scopus 로고
    • Cationic amphiphilic drugs and phospholipid storage disorder
    • Kodavanti U.P., Mehendale H.M. Cationic amphiphilic drugs and phospholipid storage disorder. Pharmacol. Rev. 1990, 42:327-354.
    • (1990) Pharmacol. Rev. , vol.42 , pp. 327-354
    • Kodavanti, U.P.1    Mehendale, H.M.2
  • 4
    • 0031057309 scopus 로고    scopus 로고
    • Cationic amphiphilic drug-induced phospholipidosis
    • Halliwell W.H. Cationic amphiphilic drug-induced phospholipidosis. Toxicol. Pathol. 1997, 25:53-60.
    • (1997) Toxicol. Pathol. , vol.25 , pp. 53-60
    • Halliwell, W.H.1
  • 5
    • 0024555455 scopus 로고
    • A review of the biology and toxicologic implications of the induction of lysosomal lamellar bodies by drugs
    • Reasor M.J. A review of the biology and toxicologic implications of the induction of lysosomal lamellar bodies by drugs. Toxicol. Appl. Pharmacol. 1989, 97:47-56.
    • (1989) Toxicol. Appl. Pharmacol. , vol.97 , pp. 47-56
    • Reasor, M.J.1
  • 6
    • 0024599878 scopus 로고
    • Amiodarone-induced pulmonary toxicity in rats: biochemical and pharmacological characteristics
    • Reasor M.J., Ogle C.L., Kacew S. Amiodarone-induced pulmonary toxicity in rats: biochemical and pharmacological characteristics. Toxicol. Appl. Pharmacol. 1989, 97:124-133.
    • (1989) Toxicol. Appl. Pharmacol. , vol.97 , pp. 124-133
    • Reasor, M.J.1    Ogle, C.L.2    Kacew, S.3
  • 8
    • 84856097267 scopus 로고    scopus 로고
    • Cerep, Phospholipidosis, ADME-Tox Application note
    • Cerep, Phospholipidosis, ADME-Tox Application note 2009.
    • (2009)
  • 9
    • 68249083749 scopus 로고    scopus 로고
    • Screening for the drug-phospholipidosis interaction: correlation to phospholipidosis
    • Alakoskela J.-M., Vitovič P., Kinnunen P.J. Screening for the drug-phospholipidosis interaction: correlation to phospholipidosis. ChemMedChem 2009, 4:1224-1251.
    • (2009) ChemMedChem , vol.4 , pp. 1224-1251
    • Alakoskela, J.-M.1    Vitovič, P.2    Kinnunen, P.J.3
  • 11
    • 0026073225 scopus 로고
    • Effect of amiodarone on the phospholipid and lamellar body content of lymphoblasts in vitro and peripheral blood lymphocytes in vivo
    • Hostetler K.Y., Vandeberg J., Aldern K.A., Brophy G.T. Effect of amiodarone on the phospholipid and lamellar body content of lymphoblasts in vitro and peripheral blood lymphocytes in vivo. Biochem. Pharmacol. 1991, 41:1007-1013.
    • (1991) Biochem. Pharmacol. , vol.41 , pp. 1007-1013
    • Hostetler, K.Y.1    Vandeberg, J.2    Aldern, K.A.3    Brophy, G.T.4
  • 13
    • 0001969538 scopus 로고
    • An in vitro fluorescence assay for the detection of drug-induced cytoplasmic lamellar bodies
    • Ulrich R.G., Kilgore K.S., Sun E.L., Cramer C.T., Ginsberg L.C. An in vitro fluorescence assay for the detection of drug-induced cytoplasmic lamellar bodies. Toxicol. Methods 1991, 1:89-105.
    • (1991) Toxicol. Methods , vol.1 , pp. 89-105
    • Ulrich, R.G.1    Kilgore, K.S.2    Sun, E.L.3    Cramer, C.T.4    Ginsberg, L.C.5
  • 16
    • 13644258653 scopus 로고    scopus 로고
    • A toxicogenomic approach to drug-induced phospholipidosis: analysis of its induction mechanism and establishment of a novel in vitro screening system
    • Sawada H., Takami K., Asahi S. A toxicogenomic approach to drug-induced phospholipidosis: analysis of its induction mechanism and establishment of a novel in vitro screening system. Toxicol. Sci. 2005, 83:282-292.
    • (2005) Toxicol. Sci. , vol.83 , pp. 282-292
    • Sawada, H.1    Takami, K.2    Asahi, S.3
  • 17
    • 41249084677 scopus 로고    scopus 로고
    • Assessment of drug-lipid complex formation by a high-throughput langmuir-balance and correlation to phospholipidosis
    • Vitovic P., Alakoskela J.M., Kinnunen P.K.J. Assessment of drug-lipid complex formation by a high-throughput langmuir-balance and correlation to phospholipidosis. J. Med. Chem. 2008, 51:1842-1848.
    • (2008) J. Med. Chem. , vol.51 , pp. 1842-1848
    • Vitovic, P.1    Alakoskela, J.M.2    Kinnunen, P.K.J.3
  • 18
    • 33749128073 scopus 로고    scopus 로고
    • Drug-induced phospholipidosis: issues and future directions
    • Reasor M.J., Hastings K.L., Ulrich R.G. Drug-induced phospholipidosis: issues and future directions. Expert Opin. Drug Saf. 2006, 5:567-583.
    • (2006) Expert Opin. Drug Saf. , vol.5 , pp. 567-583
    • Reasor, M.J.1    Hastings, K.L.2    Ulrich, R.G.3
  • 21
    • 33750928793 scopus 로고    scopus 로고
    • Physicochemical and cell-based approach for early screening of phospholipidosis-induced potential
    • Tomizawa K., Sugano K., Yamada H., Horii I. Physicochemical and cell-based approach for early screening of phospholipidosis-induced potential. J. Toxicol. Sci. 2006, 31:315-324.
    • (2006) J. Toxicol. Sci. , vol.31 , pp. 315-324
    • Tomizawa, K.1    Sugano, K.2    Yamada, H.3    Horii, I.4
  • 22
    • 80052810835 scopus 로고    scopus 로고
    • Predicting phospholipidosis: a fluorescence noncell based in vitro assay for the determination of drug-phospholipid complex formation in early drug discovery
    • Zhou L., Geraci G., Hess S., Yang L., Wang J., Argika U. Predicting phospholipidosis: a fluorescence noncell based in vitro assay for the determination of drug-phospholipid complex formation in early drug discovery. Anal. Chem. 2011, 83:6980-6987.
    • (2011) Anal. Chem. , vol.83 , pp. 6980-6987
    • Zhou, L.1    Geraci, G.2    Hess, S.3    Yang, L.4    Wang, J.5    Argika, U.6
  • 23
    • 53149126256 scopus 로고    scopus 로고
    • Prediction of intestinal and blood brain barrier permeability utilizing immobilized artifical membrane chromatography
    • Adejare A., El-Gendy A. Prediction of intestinal and blood brain barrier permeability utilizing immobilized artifical membrane chromatography. Abstracts of Papers of the American Chemical Society, vol. 228 2004, p. U960.
    • (2004) Abstracts of Papers of the American Chemical Society, vol. 228
    • Adejare, A.1    El-Gendy, A.2
  • 24
    • 0028841355 scopus 로고
    • Predicting drug-membrane interactions by HPLC: structural requirements of chromatographic surfaces
    • Liu H.L., Ong S.W., Glunz L., Pidgeon C. Predicting drug-membrane interactions by HPLC: structural requirements of chromatographic surfaces. Anal. Chem. 1995, 67:3550-3557.
    • (1995) Anal. Chem. , vol.67 , pp. 3550-3557
    • Liu, H.L.1    Ong, S.W.2    Glunz, L.3    Pidgeon, C.4
  • 26
    • 0031709543 scopus 로고    scopus 로고
    • Potential of immobilized artificial membranes for predicting drug penetration across the blood-brain barrier
    • Reichel A., Begley D.J. Potential of immobilized artificial membranes for predicting drug penetration across the blood-brain barrier. Pharm. Res. 1998, 15:1270-1274.
    • (1998) Pharm. Res. , vol.15 , pp. 1270-1274
    • Reichel, A.1    Begley, D.J.2
  • 27
    • 0036294084 scopus 로고    scopus 로고
    • Molecular factors influencing retention on immobilized artificial membranes (IAM) compared to partitioning in liposomes and n-octanol
    • Taillardat-Bertschinger A., Martinet C.A.M., Carrupt P.A., Reist M., Caron G., Fruttero R., Testa B. Molecular factors influencing retention on immobilized artificial membranes (IAM) compared to partitioning in liposomes and n-octanol. Pharm. Res. 2002, 19:729-737.
    • (2002) Pharm. Res. , vol.19 , pp. 729-737
    • Taillardat-Bertschinger, A.1    Martinet, C.A.M.2    Carrupt, P.A.3    Reist, M.4    Caron, G.5    Fruttero, R.6    Testa, B.7
  • 28
    • 17644379986 scopus 로고    scopus 로고
    • Interaction of basic drugs with lipid bilayers using liposome electrokinetic chromatography
    • Carrozzino J.M., Khaledi M.G. Interaction of basic drugs with lipid bilayers using liposome electrokinetic chromatography. Pharm. Res. 2004, 21:2327-2335.
    • (2004) Pharm. Res. , vol.21 , pp. 2327-2335
    • Carrozzino, J.M.1    Khaledi, M.G.2
  • 29
    • 20444503357 scopus 로고    scopus 로고
    • PH Effects on drug interactions with lipid bilayers by liposome electrokinetic chromatography
    • Carrozzino J.M., Khaledi M.G. pH Effects on drug interactions with lipid bilayers by liposome electrokinetic chromatography. J. Chromatogr. A 2005, 1079:307-316.
    • (2005) J. Chromatogr. A , vol.1079 , pp. 307-316
    • Carrozzino, J.M.1    Khaledi, M.G.2
  • 30
    • 53149123260 scopus 로고    scopus 로고
    • A method for rapidly predicting drug tissue distribution using surfactant vesicle electrokinetic chromatography
    • Jiang Z., Reilly J., Everatt B. A method for rapidly predicting drug tissue distribution using surfactant vesicle electrokinetic chromatography. Electrophoresis 2008, 29:3674-3684.
    • (2008) Electrophoresis , vol.29 , pp. 3674-3684
    • Jiang, Z.1    Reilly, J.2    Everatt, B.3
  • 31
    • 33644684597 scopus 로고    scopus 로고
    • Investigation of vesicle electrokinetic chromatography as an in vitro assay for the estimation of intestinal permeability of pharmaceutical drug candidates
    • Pascoe R.J., Masucci J.A., Foley J.P. Investigation of vesicle electrokinetic chromatography as an in vitro assay for the estimation of intestinal permeability of pharmaceutical drug candidates. Electrophoresis 2006, 27:793-804.
    • (2006) Electrophoresis , vol.27 , pp. 793-804
    • Pascoe, R.J.1    Masucci, J.A.2    Foley, J.P.3
  • 33
    • 0033818097 scopus 로고    scopus 로고
    • Rapid-gradient HPLC method for measuring drug interactions with immobilized artificial membrane: comparison with other lipophilicity measures
    • Valko K., Du C.M., Bevan C.D., Reynolds D.P., Abraham M.H. Rapid-gradient HPLC method for measuring drug interactions with immobilized artificial membrane: comparison with other lipophilicity measures. J. Pharm. Sci. 2000, 89:1085-1096.
    • (2000) J. Pharm. Sci. , vol.89 , pp. 1085-1096
    • Valko, K.1    Du, C.M.2    Bevan, C.D.3    Reynolds, D.P.4    Abraham, M.H.5
  • 34
    • 0242290408 scopus 로고    scopus 로고
    • Fast gradient HPLC method to determine compounds binding to human serum albumin. Relationships with octanol/water and immobilized artificial membrane lipophilicity
    • Valko K., Nunhuck S., Bevan C., Abraham M.H., Reyncilds D.P. Fast gradient HPLC method to determine compounds binding to human serum albumin. Relationships with octanol/water and immobilized artificial membrane lipophilicity. J. Pharm. Sci. 2003, 92:2236-2248.
    • (2003) J. Pharm. Sci. , vol.92 , pp. 2236-2248
    • Valko, K.1    Nunhuck, S.2    Bevan, C.3    Abraham, M.H.4    Reyncilds, D.P.5
  • 36
    • 33845370513 scopus 로고    scopus 로고
    • Estimation of volume of distribution in humans from high throughput HPLC-based measurements of human serum albumin binding and immobilized artificial membrane partitioning
    • Hollosy F., Valko K., Hersey A., Nunhuck S., Keri G., Bevan C. Estimation of volume of distribution in humans from high throughput HPLC-based measurements of human serum albumin binding and immobilized artificial membrane partitioning. J. Med. Chem. 2006, 49:6958-6971.
    • (2006) J. Med. Chem. , vol.49 , pp. 6958-6971
    • Hollosy, F.1    Valko, K.2    Hersey, A.3    Nunhuck, S.4    Keri, G.5    Bevan, C.6
  • 38
    • 0026085436 scopus 로고
    • Amiodarone pulmonary toxicity: morphologic and biochemical features
    • Reasor M.J., Kacew S. Amiodarone pulmonary toxicity: morphologic and biochemical features. Proc. Soc. Exp. Biol. Med. 1991, 196:1-7.
    • (1991) Proc. Soc. Exp. Biol. Med. , vol.196 , pp. 1-7
    • Reasor, M.J.1    Kacew, S.2
  • 39
    • 0021189040 scopus 로고
    • Lipidosis-like alterations in cultured macrophages exposed to local anaesthetics
    • Jägel M., Lüllmann-Rauch R. Lipidosis-like alterations in cultured macrophages exposed to local anaesthetics. Arch. Toxicol. 1984, 55:229-232.
    • (1984) Arch. Toxicol. , vol.55 , pp. 229-232
    • Jägel, M.1    Lüllmann-Rauch, R.2
  • 40
    • 0016256178 scopus 로고
    • Fenfluramine-induced ultrastructural alterations in tissues of rats and guinea pigs
    • Lüllmann-Rauch R., Reil G.H. Fenfluramine-induced ultrastructural alterations in tissues of rats and guinea pigs. Naunyn Schmiedeberg's Arch. Pharmacol. 1974, 285:175-184.
    • (1974) Naunyn Schmiedeberg's Arch. Pharmacol. , vol.285 , pp. 175-184
    • Lüllmann-Rauch, R.1    Reil, G.H.2
  • 42
    • 34547904254 scopus 로고    scopus 로고
    • In vitro detection of drug-induced phospholipidosis using gene expression and fluorescent phospholipid-based methodologies
    • Nioi P., Perry B.K., Wang E.J., Gu Y.Z., Snyder R.D. In vitro detection of drug-induced phospholipidosis using gene expression and fluorescent phospholipid-based methodologies. Toxicol. Sci. 2007, 99:162-173.
    • (2007) Toxicol. Sci. , vol.99 , pp. 162-173
    • Nioi, P.1    Perry, B.K.2    Wang, E.J.3    Gu, Y.Z.4    Snyder, R.D.5
  • 43
    • 0022002693 scopus 로고
    • Inhibition of purified lysosomal phospholipase A1 by various beta andrenergic blockers
    • Pappu A.S., Yazaki P.J., Hostetler K.Y. Inhibition of purified lysosomal phospholipase A1 by various beta andrenergic blockers. Biochem. Pharmacol. 1985, 34:521-524.
    • (1985) Biochem. Pharmacol. , vol.34 , pp. 521-524
    • Pappu, A.S.1    Yazaki, P.J.2    Hostetler, K.Y.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.