메뉴 건너뛰기




Volumn 66, Issue 9, 2011, Pages 710-715

Improved effectiveness of biochanin A as a P-gp inhibitor in solid dispersion

Author keywords

[No Author keywords available]

Indexed keywords

BIOCHANIN A; DEACETYLDILTIAZEM; DILTIAZEM; DRUG METABOLITE; GLYCOPROTEIN P INHIBITOR; HYDROXYPROPYLMETHYLCELLULOSE; RHODAMINE 123; SOLUTOL HS 15;

EID: 84055217418     PISSN: 00317144     EISSN: None     Source Type: Journal    
DOI: 10.1691/ph.2011.1028     Document Type: Article
Times cited : (6)

References (36)
  • 1
    • 34248535178 scopus 로고    scopus 로고
    • Studies on dissolution enhancement and mathematical modeling of drug release of a poorly water-soluble drug using water-soluble carriers
    • DOI 10.1016/j.ejpb.2006.07.007, PII S0939641106001901
    • Ahuja N, Katare OP, Singh B (2007) Studies on dissolution enhancement and mathematical modeling of drug release of a poorlywater-soluble drug using water-soluble carriers. Eur J Pharm Biopharm 65: 26-38. (Pubitemid 44827692)
    • (2007) European Journal of Pharmaceutics and Biopharmaceutics , vol.65 , Issue.1 , pp. 26-38
    • Ahuja, N.1    Katare, O.P.2    Singh, B.3
  • 3
    • 0032876066 scopus 로고    scopus 로고
    • Pharmacokinetic interactions between microemulsion formulated cyclosporine A and diltiazem in renal transplant recipients
    • DOI 10.1007/s002280050644
    • Asberg A, Christensen H, Hartmann A, Carlson E, Molden E, Berg KJ (1999) Pharmacokinetic interactions between microemulsion formulated cyclosporine A and diltiazem in renal transplant recipients. Eur J Clin Pharmacol 55: 383-387. (Pubitemid 29344082)
    • (1999) European Journal of Clinical Pharmacology , vol.55 , Issue.5 , pp. 383-387
    • Asberg, A.1    Christensen, H.2    Hartmann, A.3    Carlson, E.4    Molden, E.5    Berg, K.J.6
  • 5
    • 0037687293 scopus 로고    scopus 로고
    • Impact of Solutol HS 15 on the pharmacokinetic behaviour of colchicine upon intravenous administration to male wistar rats
    • DOI 10.1002/bdd.353
    • Bittner B, González RC, Walter I, Kapps M, Huwyler J (2003) Impact of Solutol HS 15 on the pharmacokinetic behaviour of colchicine upon intravenous administration to male Wistar rats. Biopharm Drug Dispos 24: 173-181. (Pubitemid 36656391)
    • (2003) Biopharmaceutics and Drug Disposition , vol.24 , Issue.4 , pp. 173-181
    • Bittner, B.1    Gonzalez, R.C.B.2    Walter, I.3    Kapps, M.4    Huwyler, J.5
  • 6
    • 33646772577 scopus 로고    scopus 로고
    • Clinical studies of red clover (Trifolium pratense) dietary supplements in menopause: A literature review
    • Booth NL, Piersen CE, Banuvar S, Geller SE, Shulman LP, Farnsworth NR (2006) Clinical studies of red clover (Trifolium pratense) dietary supplements in menopause: a literature review. Menopause 13: 251-264.
    • (2006) Menopause , vol.13 , pp. 251-264
    • Booth, N.L.1    Piersen, C.E.2    Banuvar, S.3    Geller, S.E.4    Shulman, L.P.5    Farnsworth, N.R.6
  • 7
    • 0031060647 scopus 로고    scopus 로고
    • Inhibition of drug transport by genistein in multidrug-resistant cells expressing P-glycoprotein
    • DOI 10.1016/S0006-2952(96)00657-0, PII S0006295296006570
    • Castro AF, Altenberg GA (1997) Inhibition of drug transport by genistein in multidrug-resistant cells expressing P-glycoprotein. Biochem Pharmacol 53: 89-93. (Pubitemid 26419790)
    • (1997) Biochemical Pharmacology , vol.53 , Issue.1 , pp. 89-93
    • Castro, A.F.1    Altenberg, G.A.2
  • 8
    • 1842789744 scopus 로고    scopus 로고
    • Enhanced bioavailability of paclitaxel after the oral coadministration with flavone in rats
    • Choi JS, Choi HK, Shin SC (2004) Enhanced bioavailability of paclitaxel after the oral coadministration with flavone in rats. Int J Pharm 275: 165-170.
    • (2004) Int J Pharm , vol.275 , pp. 165-170
    • Choi, J.S.1    Choi, H.K.2    Shin, S.C.3
  • 9
    • 0026101562 scopus 로고
    • Solutol HS 15, nontoxic polyoxyethylene esters of 12-hydroxystearic acid, reverses multidrug resistance
    • Coon JS, Knudson W, Clodfelter K, Lu B,Weinstein RS (1991) Solutol HS 15, nontoxic polyoxyethylene esters of 12-hydroxystearic acid, reverses multidrug resistance. Cancer Res 51: 897-902.
    • (1991) Cancer Res , vol.51 , pp. 897-902
    • Coon, J.S.1    Knudson, W.2    Clodfelter, K.3    Lu, B.4    Weinstein, R.S.5
  • 10
    • 33846355740 scopus 로고    scopus 로고
    • Trifolium pratense isoflavones in the treatment of menopausal hot flushes: A systematic review and meta-analysis
    • DOI 10.1016/j.phymed.2006.12.009, PII S0944711306002261
    • Coon JT, Pittler MH, Ernst E (2007) Trifolium pratense isoflavones in the treatment of menopausal hot flushes: a systematic review and metaanalysis. Phytomedicine 14: 153-159. (Pubitemid 46136954)
    • (2007) Phytomedicine , vol.14 , Issue.2-3 , pp. 153-159
    • Thompson, C.J.1    Pittler, M.H.2    Ernst, E.3
  • 11
    • 0029954843 scopus 로고    scopus 로고
    • P-Glycoprotein-a mediator of multidrug resistance in tumour cells
    • Germann UA (1996) P-Glycoprotein-a mediator of multidrug resistance in tumour cells. Eur J Cancer 32A: 927-944.
    • (1996) Eur J Cancer , vol.32 A , pp. 927-944
    • Germann, U.A.1
  • 12
    • 0022411041 scopus 로고
    • High-performance liquid chromatographic determination of diltiazem and four of its metabolites in plasma. Application to pharmacokinetics
    • Goebel KJ, Kolle EU (1985) High-performance liquid chromatographic determination of diltiazem and four of its metabolites in plasma. Application to pharmacokinetics. J Chromatogr 345: 355-363.
    • (1985) J Chromatogr , vol.345 , pp. 355-363
    • Goebel, K.J.1    Kolle, E.U.2
  • 13
    • 79960161186 scopus 로고    scopus 로고
    • Enhanced dissolution and bioavailability of biochanin A, poorly soluble bioflavonoid, via the preparation of solid dispersion: In vitro and in vivo evaluation
    • in press
    • Han HK, Lee BJ, Lee HK (2011) Enhanced dissolution and bioavailability of biochanin A, poorly soluble bioflavonoid, via the preparation of solid dispersion: in vitro and in vivo evaluation., Int J Pharm, in press.
    • (2011) Int J Pharm
    • Han, H.K.1    Lee, B.J.2    Lee, H.K.3
  • 14
    • 33645830172 scopus 로고
    • A surface glycoprotein modulating drug permeability in Chinese hamster ovary cell mutants
    • Juliano RL, Ling V (1976) A surface glycoprotein modulating drug permeability in Chinese hamster ovary cell mutants. Biochim Biophys Acta 455: 152-162.
    • (1976) Biochim Biophys Acta , vol.455 , pp. 152-162
    • Juliano, R.L.1    Ling, V.2
  • 15
    • 0020578356 scopus 로고
    • Cell surface P-glycoprotein associated with multidrug resistance in mammalian cell lines
    • Kartner N, Riordan JR, Ling V (1983) Cell surface P-glycoprotein associated with multidrug resistance in mammalian cell lines. Science 221: 1285-1288. (Pubitemid 13005502)
    • (1983) Science , vol.221 , Issue.4617 , pp. 1285-1288
    • Kartner, N.1    Riordan, J.R.2    Ling, V.3
  • 16
    • 0042574839 scopus 로고
    • Inhibition of platelet aggregation by diltiazem. Comparison with verapamil and nifedipine and inhibitory potencies of diltiazem metabolites
    • Kiyomoto A, Sasaki Y, Odawara A, Morita T (1983) Inhibition of platelet aggregation by diltiazem. Comparison with verapamil and nifedipine and inhibitory potencies of diltiazem metabolites. Circ Res 52: I115-119.
    • (1983) Circ Res , vol.52
    • Kiyomoto, A.1    Sasaki, Y.2    Odawara, A.3    Morita, T.4
  • 18
    • 0036132773 scopus 로고    scopus 로고
    • Effect of dietary administration of genistein, nonylphenol or ethinyl estradiol on hepatic testosterone metabolism, cytochrome P-450 enzymes, and estrogen receptor alpha expression
    • DOI 10.1016/S0278-6915(01)00095-3, PII S0278691501000953
    • Laurenzana EM, Weis CC, Bryant CW, Newbold R, Delclos KB (2002) Effect of dietary administration of genistein, nonylphenol or ethinyl estradiol on hepatic testosterone metabolism, cytochrome P-450 enzymes, and estrogen receptor alpha expression. Food Chem Toxicol 40: 53-63. (Pubitemid 33132141)
    • (2002) Food and Chemical Toxicology , vol.40 , Issue.1 , pp. 53-63
    • Laurenzana, E.M.1    Weis, C.C.2    Bryant, C.W.3    Newbold, R.4    Delclos, K.B.5
  • 20
    • 0033637140 scopus 로고    scopus 로고
    • The effects of plant flavonoids on mammalian cells: Implications for inflammation, heart disease, and cancer
    • Middleton E, Jr. Kandaswami C, Theoharides TC (2000) The effects of plant flavonoids on mammalian cells: implications for inflammation, heart disease, and cancer. Pharmacol Rev 52: 673-751.
    • (2000) Pharmacol Rev , vol.52 , pp. 673-751
    • Middleton Jr., E.1    Kandaswami, C.2    Theoharides, T.C.3
  • 21
    • 0033671146 scopus 로고    scopus 로고
    • CYP2D6 is involved in Odemethylation of diltiazem. An in vitro study with transfected human liver cells
    • Molden E, Asberg A, Christensen H (2000) CYP2D6 is involved in Odemethylation of diltiazem. An in vitro study with transfected human liver cells. Eur J Clin Pharmacol 56: 575-579.
    • (2000) Eur J Clin Pharmacol , vol.56 , pp. 575-579
    • Molden, E.1    Asberg, A.2    Christensen, H.3
  • 22
    • 33746197977 scopus 로고    scopus 로고
    • Pharmacokinetics and bioavailability of the isoflavone biochanin A in rats
    • DOI 10.1208/aapsj080351, 51
    • Moon YJ, Sagawa K, Frederick K, Zhang S, Morris ME (2006) Pharmacokinetics and bioavailability of the isoflavone biochanin A in rats. AAPS J 8: E433-442. (Pubitemid 44096604)
    • (2006) AAPS Journal , vol.8 , Issue.3
    • Moon, Y.J.1    Sagawa, K.2    Frederick, K.3    Zhang, S.4    Morris, M.E.5
  • 23
    • 33748931006 scopus 로고    scopus 로고
    • Altered oral bioavailability and pharmacokinetics of P-glycoprotein substrates by coadministration of biochanin A
    • DOI 10.1002/jps.20664
    • Peng SX, Ritchie DM, Cousineau M, Danser E, Dewire R, Floden J (2006) Altered the oral bioavailability and pharmacokinetics of Pglycoprotein substrates by coadministration of biochanin A. J Pharm Sci 95: 1984-1993. (Pubitemid 44433029)
    • (2006) Journal of Pharmaceutical Sciences , vol.95 , Issue.9 , pp. 1984-1993
    • Peng, S.X.1    Ritchie, D.M.2    Cousineau, M.3    Danser, E.4    Dewire, R.5    Floden, J.6
  • 24
  • 25
    • 77955845684 scopus 로고    scopus 로고
    • Effect of maceligan on the systemic exposure of paclitaxel: In vitro and in vivo evaluation
    • Qiang F, Lee BJ, Ha I, Kang KW, Woo ER, Han HK (2010) Effect of maceligan on the systemic exposure of paclitaxel: in vitro and in vivo evaluation. Eur J Pharm Sci 41: 226-231.
    • (2010) Eur J Pharm Sci , vol.41 , pp. 226-231
    • Qiang, F.1    Lee, B.J.2    Ha, I.3    Kang, K.W.4    Woo, E.R.5    Han, H.K.6
  • 27
    • 36549042006 scopus 로고    scopus 로고
    • Solid dispersions as strategy to improve oral bioavailability of poor water soluble drugs
    • DOI 10.1016/j.drudis.2007.09.005, PII S1359644607003753
    • Vasconcelos T, Sarmento B, Costa P (2007) Solid dispersions as strategy to improve the oral bioavailability of poor water soluble drugs. Drug Discov Today 12: 1068-1075. (Pubitemid 350186132)
    • (2007) Drug Discovery Today , vol.12 , Issue.23-24 , pp. 1068-1075
    • Vasconcelos, T.1    Sarmento, B.2    Costa, P.3
  • 28
    • 0035290059 scopus 로고    scopus 로고
    • Active secretion and enterocytic drug metabolism barriers to drug absorption
    • Wacher VJ, Salphati L, Benet LZ (2001) Active secretion and enterocytic drug metabolism barriers to drug absorption. Adv Drug Deliv Rev 46: 89-102.
    • (2001) Adv Drug Deliv Rev , vol.46 , pp. 89-102
    • Wacher, V.J.1    Salphati, L.2    Benet, L.Z.3
  • 29
    • 0029028792 scopus 로고
    • Overlapping substrate specificities and tissue distribution of cytochrome P450 3A and P-glycoprotein: Implications for drug delivery and activity in cancer chemotherapy
    • Wacher VJ, Wu CY, Benet LZ (1995) Overlapping substrate specificities and tissue distribution of cytochrome P450 3A and P-glycoprotein: implications for drug delivery and activity in cancer chemotherapy. Mol Carcinog 13: 129-134.
    • (1995) Mol Carcinog , vol.13 , pp. 129-134
    • Wacher, V.J.1    Wu, C.Y.2    Benet, L.Z.3
  • 30
    • 33749255173 scopus 로고    scopus 로고
    • Down-regulation of P-glycoprotein expression in MDR breast cancer cell MCF-7/ADR by honokiol
    • DOI 10.1016/j.canlet.2005.11.031, PII S0304383505010359
    • Xu D, Lu Q, Hu X (2006) Down-regulation of P-glycoprotein expression in MDR breast cancer cell MCF-7/ADR by honokiol. Cancer Lett 243: 274-280. (Pubitemid 44485849)
    • (2006) Cancer Letters , vol.243 , Issue.2 , pp. 274-280
    • Xu, D.1    Lu, Q.2    Hu, X.3
  • 31
    • 0021918578 scopus 로고
    • Cardiovascular effects of the metabolites of diltiazem in dogs
    • Yabana H, Nagao T, Sato M (1985) Cardiovascular effects of the metabolites of diltiazem in dogs. J Cardiovasc Pharmacol 7: 152-157. (Pubitemid 15162258)
    • (1985) Journal of Cardiovascular Pharmacology , vol.7 , Issue.1 , pp. 152-157
    • Yabana, H.1    Nagao, T.2    Sato, M.3
  • 32
    • 0024421664 scopus 로고
    • Reversal mechanism of multidrug resistance by verapamil: Direct binding of verapamil to P-glycoprotein on specific sites and transport of verapamil outward across the plasma membrane of K562/ADM cells
    • Yusa K, Tsuruo T (1989) Reversal mechanism of multidrug resistance by verapamil: direct binding of verapamil to P-glycoprotein on specific sites and transport of verapamil outward across the plasma membrane of K562/ADM cells. Cancer Res 49: 5002-5006. (Pubitemid 19239333)
    • (1989) Cancer Research , vol.49 , Issue.18 , pp. 5002-5006
    • Yusa, K.1    Tsuruo, T.2
  • 33
    • 0037371275 scopus 로고    scopus 로고
    • Effects of the flavonoids biochanin A, morin, phloretin, and silymarin on P-glycoprotein-mediated transport
    • DOI 10.1124/jpet.102.044412
    • Zhang S, Morris ME (2003a) Effects of the flavonoids biochanin A, morin, phloretin, and silymarin on P-glycoprotein-mediated transport. J Pharmacol Exp Ther 304: 1258-1267. (Pubitemid 36254439)
    • (2003) Journal of Pharmacology and Experimental Therapeutics , vol.304 , Issue.3 , pp. 1258-1267
    • Zhang, S.1    Morris, M.E.2
  • 34
    • 0043127383 scopus 로고    scopus 로고
    • Effect of the flavonoids biochanin A and silymarin on the P-glycoprotein-mediated transport of digoxin and vinblastine in human intestinal Caco-2 cells
    • DOI 10.1023/A:1025044913766
    • Zhang S, Morris ME (2003b) Effect of the flavonoids biochanin A and silymarin on the P-glycoprotein-mediated transport of digoxin and vinblastine in human intestinal Caco-2 cells. Pharm Res 20: 1184-1191. (Pubitemid 36951843)
    • (2003) Pharmaceutical Research , vol.20 , Issue.8 , pp. 1184-1191
    • Zhang, S.1    Morris, M.E.2
  • 35
    • 72749084863 scopus 로고    scopus 로고
    • Interactions between the flavonoid biochanin A and P-glycoprotein substrates in rats: In vitro and in vivo
    • Zhang S, Sagawa K, Arnold RD, Tseng E,Wang X, Morris ME (2010) Interactions between the flavonoid biochanin A and P-glycoprotein substrates in rats: in vitro and in vivo. J Pharm Sci 99: 430-441.
    • (2010) J Pharm Sci , vol.99 , pp. 430-441
    • Zhang, S.1    Sagawa, K.2    Arnold, R.D.3    Tseng, E.4    Wang, X.5    Morris, M.E.6
  • 36
    • 2142711101 scopus 로고    scopus 로고
    • Flavonoids are inhibitors of breast cancer resistance protein (ABCG2)-mediated transport
    • DOI 10.1124/mol.65.5.1208
    • Zhang S, Yang X, Morris ME (2004) Flavonoids are inhibitors of breast cancer resistance protein (ABCG2)-mediated transport. Mol Pharmacol 65: 1208-1216. (Pubitemid 38543491)
    • (2004) Molecular Pharmacology , vol.65 , Issue.5 , pp. 1208-1216
    • Zhang, S.1    Yang, X.2    Morris, M.E.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.