Use and limitations of three TRPV-1 receptor antagonists on smooth muscles of animals and man: A vote for BCTC

European Journal of Pharmacology

Volumn 674, Issue 1, 2012, Pages 44-50

  Benko, Rita ^a   Illényi, Lászlo ^a   Kelemen, Dezsö ^a   Papp, Robert ^a   Papp, András ^a   Bartho, Loránd ^a  

^a UNIVERSITY OF PÉCS   (Hungary)

Author keywords

BCTC; Capsaicin; Capsazepine; Human intestine; Iodo resiniferatoxin; Smooth muscles; TRPV 1 antagonist

Indexed keywords

5' IODORESINIFERATOXIN; CAPSAZEPINE; N (4 TERT BUTYLPHENYL) 4 (3 CHLORO 2 PYRIDINYL) 1 PIPERAZINECARBOXAMIDE; VANILLOID RECEPTOR 1 ANTAGONIST;

ANIMAL TISSUE; ARTICLE; BLADDER; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG SAFETY; FEMALE; GUINEA PIG; HUMAN; HUMAN TISSUE; ILEUM; INHIBITION KINETICS; INOTROPISM; INTESTINE MUSCLE; KIDNEY PELVIS; MALE; MOUSE; MUSCLE EXCITATION; MUSCLE RELAXATION; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR DOWN REGULATION; SENSORY NERVE CELL; SMOOTH MUSCLE CONTRACTILITY; SMOOTH MUSCLE CONTRACTION; TRACHEA;

EID: 82255183918     PISSN: 00142999     EISSN: 18790712     Source Type: Journal    
DOI: 10.1016/j.ejphar.2011.10.021     Document Type: Article

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