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Volumn 46, Issue 9, 2011, Pages 4760-4767

Synthesis and preliminary in vitro biological evaluation of new carbon-11-labeled celecoxib derivatives as candidate PET tracers for imaging of COX-2 expression in cancer

(4) Gao, Mingzhang a Wang, Min a Miller, Kathy D b Zheng, Qi Huang a

a INDIANA UNIVERSITY SCHOOL OF MEDICINE (United States)

b INDIANA UNIVERSITY (United States)

Author keywords

Cancer imaging; Carbon 11 labeled celecoxib derivatives; Cyclooxygenase 2 (COX 2); Positron emission tomography (PET); Radiotracers

Indexed keywords

4 [5 (2 METHOXYPHENYL) 3 (TRIFLUOROMETHYL) 1H PYRAZOL 1 YL]BENZENESULFONAMIDE; 4 [5 (2 METHOXYPHENYL) 3 (TRIFLUOROMETHYL) 1H PYRAZOL 1 YL]BENZOATE; 4 [5 (3 METHOXYPHENYL) 3 (TRIFLUOROMETHYL) 1H PYRAZOL 1 YL]BENZENESULFONAMIDE; 4 [5 (4 METHOXYPHENYL) 3 (TRIFLUOROMETHYL) 1H PYRAZOL 1 YL]BENZENESULFONAMIDE; CARBON 11; CELECOXIB; CYCLOOXYGENASE 2; METHYL 4 [5 (3 METHOXYPHENYL) 3 (TRIFLUOROMETHYL) 1H PYRAZOL 1 YL]BENZOATE; METHYL 4 [5 (4 METHOXYPHENYL) 3 (TRIFLUOROMETHYL) 1H PYRAZOL 1 YL]BENZOATE; METHYL 4 [5 (P TOLYL) 3 (TRIFLUOROMETHYL) 1H PYRAZOL 1 YL]BENZOATE; TRACER; UNCLASSIFIED DRUG;

ARTICLE; CANCER CELL CULTURE; CANCER DIAGNOSIS; DRUG PURITY; DRUG SYNTHESIS; HUMAN; HUMAN CELL; IN VITRO STUDY; METHYLATION; POSITRON EMISSION TOMOGRAPHY; PROTEIN EXPRESSION; RADIOCHEMISTRY; SOLID PHASE EXTRACTION;

CARBON RADIOISOTOPES; CELL LINE, TUMOR; CELL PROLIFERATION; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; CYCLOOXYGENASE 2; HUMANS; MAGNETIC RESONANCE SPECTROSCOPY; NEOPLASMS; POSITRON-EMISSION TOMOGRAPHY; PYRAZOLES; SULFONAMIDES;

EID: 80052920865 PISSN: 02235234 EISSN: 17683254 Source Type: Journal
DOI: 10.1016/j.ejmech.2011.05.024 Document Type: Article

Times cited : (19)

References (38)

1
- 78649329129
- R. Fioravanti, A. Bolasco, F. Manna, F. Rossi, F. Orallo, F. Ortuso, S. Alcaro, and R. Cirilli Eur. J. Med. Chem. 45 2010 6135 6138
- (2010) Eur. J. Med. Chem. , vol.45 , pp. 6135-6138
- Fioravanti, R.¹ Bolasco, A.² Manna, F.³ Rossi, F.⁴ Orallo, F.⁵ Ortuso, F.⁶ Alcaro, S.⁷ Cirilli, R.⁸

2
- 77956735860
- Y. Harrak, G. Casula, J. Basset, G. Rosell, S. Plescia, D. Raffa, M.G. Cusimano, R. Pouplana, and M.D. Pujol J. Med. Chem. 53 2010 6560 6571
- (2010) J. Med. Chem. , vol.53 , pp. 6560-6571
- Harrak, Y.¹ Casula, G.² Basset, J.³ Rosell, G.⁴ Plescia, S.⁵ Raffa, D.⁶ Cusimano, M.G.⁷ Pouplana, R.⁸ Pujol, M.D.⁹

3
- 11144228243
- F. Julémont, X. de Leval, C. Michaux, J.F. Renard, J.Y. Winum, J.L. Montero, J. Damas, J.M. Dogné, and B. Pirotte J. Med. Chem. 47 2004 6749 6759
- (2004) J. Med. Chem. , vol.47 , pp. 6749-6759
- Julémont, F.¹ De Leval, X.² Michaux, C.³ Renard, J.F.⁴ Winum, J.Y.⁵ Montero, J.L.⁶ Damas, J.⁷ Dogné, J.M.⁸ Pirotte, B.⁹

4
- 77956412010
- N.V. Cunha, S.B. de Abreu, C. Panis, S. Grassiolli, F.A. Guarnier, R. Cecchini, T.L. Mazzuco, P. Pinge-Filho, and M.C. Martins-Pinge Life Sci. 87 2010 375 381
- (2010) Life Sci. , vol.87 , pp. 375-381
- Cunha, N.V.¹ De Abreu, S.B.² Panis, C.³ Grassiolli, S.⁴ Guarnier, F.A.⁵ Cecchini, R.⁶ Mazzuco, T.L.⁷ Pinge-Filho, P.⁸ Martins-Pinge, M.C.⁹

5
- 77955801063
- C. Bocca, F. Bozzo, A. Bassignana, and A. Miglietta Anticancer Res. 30 2010 2659 2666
- (2010) Anticancer Res. , vol.30 , pp. 2659-2666
- Bocca, C.¹ Bozzo, F.² Bassignana, A.³ Miglietta, A.⁴

6
- 78049457767
- A. Jukić, D.M. Kaliterna, and M. Radi&cacute Reumatizam 57 2010 26 28
- (2010) Reumatizam , vol.57 , pp. 26-28
- Jukić, A.¹ Kaliterna, D.M.² Radi³ Cacute, M.⁴

7
- 78049297452
- J.Y. Liu, N. Li, J. Yang, N. Li, H. Qiu, D. Ai, N. Chiamvimonvat, Y. Zhu, and B.D. Hammock Proc. Natl. Acad. Sci. U.S.A. 107 2010 17017 17022
- (2010) Proc. Natl. Acad. Sci. U.S.A. , vol.107 , pp. 17017-17022
- Liu, J.Y.¹ Li, N.² Yang, J.³ Li, N.⁴ Qiu, H.⁵ Ai, D.⁶ Chiamvimonvat, N.⁷ Zhu, Y.⁸ Hammock, B.D.⁹

8
- 78049438246
- C. Cerella, C. Sobolewski, M. Dicato, and M. Diederich Biochem. Pharmacol. 80 2010 1801 1815
- (2010) Biochem. Pharmacol. , vol.80 , pp. 1801-1815
- Cerella, C.¹ Sobolewski, C.² Dicato, M.³ Diederich, M.⁴

9
- 77953329962
- P. Jones, and R. Lamdin Clin. Drug Investig. 30 2010 419 437
- (2010) Clin. Drug Investig. , vol.30 , pp. 419-437
- Jones, P.¹ Lamdin, R.²

10
- 77955714043
- K.R. Abdellatif, C.A. Velázquez, Z. Huang, M.A. Chowdhury, and E.E. Knaus Bioorg. Med. Chem. Lett. 20 2010 5245 5250
- (2010) Bioorg. Med. Chem. Lett. , vol.20 , pp. 5245-5250
- Abdellatif, K.R.¹ Velázquez, C.A.² Huang, Z.³ Chowdhury, M.A.⁴ Knaus, E.E.⁵

11
- 77950630920
- F. Krötz, and L. Struthmann Cardiovasc. Hematol. Disord. Drug Targets 10 2010 53 65
- (2010) Cardiovasc. Hematol. Disord. Drug Targets , vol.10 , pp. 53-65
- Krötz, F.¹ Struthmann, L.²

12
- 77953506537
- A.K. Chakraborti, S.K. Garg, R. Kumar, H.F. Motiwala, and P.S. Jadhavar Curr. Med. Chem. 17 2010 1563 1593
- (2010) Curr. Med. Chem. , vol.17 , pp. 1563-1593
- Chakraborti, A.K.¹ Garg, S.K.² Kumar, R.³ Motiwala, H.F.⁴ Jadhavar, P.S.⁵

13
- 69949150537
- T.C. Ramalho, M.V. Rocha, E.F. da Cunha, and M.P. Freitas Expert Opin. Ther. Pat. 19 2009 1193 1228
- (2009) Expert Opin. Ther. Pat. , vol.19 , pp. 1193-1228
- Ramalho, T.C.¹ Rocha, M.V.² Da Cunha, E.F.³ Freitas, M.P.⁴

14
- 37849035499
- G. Szabó, J. Fischer, A. Kis-Varga, and K. Gyires J. Med. Chem. 51 2008 142 147
- (2008) J. Med. Chem. , vol.51 , pp. 142-147
- Szabó, G.¹ Fischer, J.² Kis-Varga, A.³ Gyires, K.⁴

15
- 33749828011
- E.F. de Vries Curr. Pharm. Des 12 2006 3847 3856
- (2006) Curr. Pharm. des , vol.12 , pp. 3847-3856
- De Vries, E.F.¹

16
- 37349054262
- E.F. de Vries, J. Doorduin, R.A. Dierckx, and A. van Waarde Nucl. Med. Biol. 35 2008 35 42
- (2008) Nucl. Med. Biol. , vol.35 , pp. 35-42
- De Vries, E.F.¹ Doorduin, J.² Dierckx, R.A.³ Van Waarde, A.⁴

17
- 70350234582
- Y. Kuge, N. Obokata, H. Kimura, Y. Katada, T. Temma, Y. Sugimoto, K. Aita, K. Seki, N. Tamaki, and H. Saji Nucl. Med. Biol. 36 2009 869 876
- (2009) Nucl. Med. Biol. , vol.36 , pp. 869-876
- Kuge, Y.¹ Obokata, N.² Kimura, H.³ Katada, Y.⁴ Temma, T.⁵ Sugimoto, Y.⁶ Aita, K.⁷ Seki, K.⁸ Tamaki, N.⁹ Saji, H.¹⁰

18
- 31844440302
- Y. Kuge, Y. Katada, S. Shimonaka, T. Temma, H. Kimura, Y. Kiyono, C. Yokota, K. Minematsu, K. Seki, N. Tamaki, K. Ohkura, and H. Saji Nucl. Med. Biol. 33 2006 21 27
- (2006) Nucl. Med. Biol. , vol.33 , pp. 21-27
- Kuge, Y.¹ Katada, Y.² Shimonaka, S.³ Temma, T.⁴ Kimura, H.⁵ Kiyono, Y.⁶ Yokota, C.⁷ Minematsu, K.⁸ Seki, K.⁹ Tamaki, N.¹⁰ Ohkura, K.¹¹ Saji, H.¹²

19
- 27844543335
- J. Prabhakaran, V.J. Majo, N.S. Simpson, R.L. van Heertum, J.J. Monn, and J.S.D. Kumar J. Labelled Compd. Radiopharm. 48 2005 887 895
- (2005) J. Labelled Compd. Radiopharm. , vol.48 , pp. 887-895
- Prabhakaran, J.¹ Majo, V.J.² Simpson, N.S.³ Van Heertum, R.L.⁴ Monn, J.J.⁵ Kumar, J.S.D.⁶

20
- 33847783301
- J. Prabhakaran, M.D. Underwood, R.V. Parsey, V. Arango, V.J. Majo, N.R. Simpson, R. van Heertum, J.J. Mann, and J.S.D. Kumar Bioorg. Med. Chem. 15 2007 1802 1807
- (2007) Bioorg. Med. Chem. , vol.15 , pp. 1802-1807
- Prabhakaran, J.¹ Underwood, M.D.² Parsey, R.V.³ Arango, V.⁴ Majo, V.J.⁵ Simpson, N.R.⁶ Van Heertum, R.⁷ Mann, J.J.⁸ Kumar, J.S.D.⁹

21
- 49149103216
- F. Wuest, T. Kniess, R. Bergmann, and J. Pietzsch Bioorg. Med. Chem. 16 2008 7662 7670
- (2008) Bioorg. Med. Chem. , vol.16 , pp. 7662-7670
- Wuest, F.¹ Kniess, T.² Bergmann, R.³ Pietzsch, J.⁴

22
- 69549135103
- M. Gao, M. Wang, K.D. Miller, G.D. Hutchins, and Q.H. Zheng Appl. Radiat. Isot. 67 2009 2019 2024
- (2009) Appl. Radiat. Isot. , vol.67 , pp. 2019-2024
- Gao, M.¹ Wang, M.² Miller, K.D.³ Hutchins, G.D.⁴ Zheng, Q.H.⁵

23
- 13444266910
- T.D. Penning, J.J. Talley, S.R. Bertenshaw, J.S. Carter, P.W. Collins, S. Docter, M.J. Graneto, L.F. Lee, J.W. Malecha, J.M. Miyashiro, R.S. Rogers, D.J. Rogier, S.S. Yu, G.D. Anderson, E.G. Burton, J.N. Cogburn, S.A. Gregory, C.M. Koboldt, W.E. Perkins, K. Seibert, A.W. Veenhuizen, Y.Y. Zhang, and P.C. Isakson J. Med. Chem. 40 1997 1347 1365
- (1997) J. Med. Chem. , vol.40 , pp. 1347-1365
- Penning, T.D.¹ Talley, J.J.² Bertenshaw, S.R.³ Carter, J.S.⁴ Collins, P.W.⁵ Docter, S.⁶ Graneto, M.J.⁷ Lee, L.F.⁸ Malecha, J.W.⁹ Miyashiro, J.M.¹⁰ Rogers, R.S.¹¹ Rogier, D.J.¹² Yu, S.S.¹³ Anderson, G.D.¹⁴ Burton, E.G.¹⁵ Cogburn, J.N.¹⁶ Gregory, S.A.¹⁷ Koboldt, C.M.¹⁸ Perkins, W.E.¹⁹ Seibert, K.²⁰ more..

24
- 34548501268
- M.M. Ahlström, M. Ridderström, I. Zamora, and K. Luthman J. Med. Chem. 50 2007 4444 4452
- (2007) J. Med. Chem. , vol.50 , pp. 4444-4452
- Ahlström, M.M.¹ Ridderström, M.² Zamora, I.³ Luthman, K.⁴

25
- 10744221608
- Q.H. Zheng, X. Fei, T.R. DeGrado, J.Q. Wang, K.L. Stone, T.D. Martinez, D.J. Gay, W.L. Baity, B.H. Mock, B.E. Glick-Wilson, M.L. Sullivan, K.D. Miller, G.W. Sledge, and G.D. Hutchins Nucl. Med. Biol. 30 2003 753 760
- (2003) Nucl. Med. Biol. , vol.30 , pp. 753-760
- Zheng, Q.H.¹ Fei, X.² Degrado, T.R.³ Wang, J.Q.⁴ Stone, K.L.⁵ Martinez, T.D.⁶ Gay, D.J.⁷ Baity, W.L.⁸ Mock, B.H.⁹ Glick-Wilson, B.E.¹⁰ Sullivan, M.L.¹¹ Miller, K.D.¹² Sledge, G.W.¹³ Hutchins, G.D.¹⁴

26
- 0037291678
- S. Furumoto, K. Takashima, K. Kubota, T. Ido, R. Iwata, and H. Fukuda Nucl. Med. Biol. 30 2003 119 125
- (2003) Nucl. Med. Biol. , vol.30 , pp. 119-125
- Furumoto, S.¹ Takashima, K.² Kubota, K.³ Ido, T.⁴ Iwata, R.⁵ Fukuda, H.⁶

27
- 0033014492
- B.H. Mock, G.K. Mulholland, and M.T. Vavrek Nucl. Med. Biol. 26 1999 467 471
- (1999) Nucl. Med. Biol. , vol.26 , pp. 467-471
- Mock, B.H.¹ Mulholland, G.K.² Vavrek, M.T.³

28
- 0026440649
- D.M. Jewett Int. J. Rad. Appl. Instrum. A 43 1992 1383 1385
- (1992) Int. J. Rad. Appl. Instrum. A , vol.43 , pp. 1383-1385
- Jewett, D.M.¹

29
- 53549088596
- M. Gao, M. Wang, G.D. Hutchins, and Q.H. Zheng Appl. Radiat. Isot 66 2008 1891 1897
- (2008) Appl. Radiat. Isot , vol.66 , pp. 1891-1897
- Gao, M.¹ Wang, M.² Hutchins, G.D.³ Zheng, Q.H.⁴

30
- 58749093948
- K.K. Yoder, G.D. Hutchins, B.H. Mock, X. Fei, W.L. Winkle, B.D. Gitter, P.R. Territo, and Q.H. Zheng Nucl. Med. Biol. 36 2009 11 16
- (2009) Nucl. Med. Biol. , vol.36 , pp. 11-16
- Yoder, K.K.¹ Hutchins, G.D.² Mock, B.H.³ Fei, X.⁴ Winkle, W.L.⁵ Gitter, B.D.⁶ Territo, P.R.⁷ Zheng, Q.H.⁸

31
- 0030294781
- Q.H. Zheng, and G.K. Mulholland Nucl. Med. Biol. 23 1996 981 986
- (1996) Nucl. Med. Biol. , vol.23 , pp. 981-986
- Zheng, Q.H.¹ Mulholland, G.K.²

32
- 33746630372
- B.H. Mock, Q.-H. Zheng, and T.R. DeGrado J. Labelled Compd. Radiopharm. 48 2005 S225
- (2005) J. Labelled Compd. Radiopharm. , vol.48 , pp. 225
- Mock, B.H.¹ Zheng, Q.-H.² Degrado, T.R.³

33
- 33746659597
- B.H. Mock, B.E. Glick-Wilson, Q.H. Zheng, and T.R. DeGrado J. Labelled Compd. Radiopharm. 48 2005 S224
- (2005) J. Labelled Compd. Radiopharm. , vol.48 , pp. 224
- Mock, B.H.¹ Glick-Wilson, B.E.² Zheng, Q.H.³ Degrado, T.R.⁴

34
- 33947702669
- Q.H. Zheng, M. Gao, B.H. Mock, S. Wang, T. Hara, R. Nazih, M.A. Miller, T.J. Receveur, J.C. Lopshire, W.J. Groh, D.P. Zipes, G.D. Hutchins, and T.R. DeGrado Bioorg. Med. Chem. Lett. 17 2007 2220 2224
- (2007) Bioorg. Med. Chem. Lett. , vol.17 , pp. 2220-2224
- Zheng, Q.H.¹ Gao, M.² Mock, B.H.³ Wang, S.⁴ Hara, T.⁵ Nazih, R.⁶ Miller, M.A.⁷ Receveur, T.J.⁸ Lopshire, J.C.⁹ Groh, W.J.¹⁰ Zipes, D.P.¹¹ Hutchins, G.D.¹² Degrado, T.R.¹³

35
- 28444492607
- Q.H. Zheng, and B.H. Mock Biomed. Chromatogr. 19 2005 671 67676
- (2005) Biomed. Chromatogr. , vol.19 , pp. 671-67676
- Zheng, Q.H.¹ Mock, B.H.²

36
- 64549150228
- D. Boschi, L. Lazzarato, B. Rolando, A. Fillieri, C. Cena, A. Di Stilo, R. Fruttereo, and A. Gasco Chem. Biodivers. 6 2009 369 379
- (2009) Chem. Biodivers. , vol.6 , pp. 369-379
- Boschi, D.¹ Lazzarato, L.² Rolando, B.³ Fillieri, A.⁴ Cena, C.⁵ Di Stilo, A.⁶ Fruttereo, R.⁷ Gasco, A.⁸

37
- 7644228315
- R.S. Fife, B. Stott, and R.E. Carr Cancer Biol. Ther. 3 2004 228 232
- (2004) Cancer Biol. Ther. , vol.3 , pp. 228-232
- Fife, R.S.¹ Stott, B.² Carr, R.E.³

38
- 53149108620
- M. Gao, M. Wang, K.D. Miller, G.W. Sledge, and Q.H. Zheng Eur. J. Med. Chem. 43 2008 2211 2219
- (2008) Eur. J. Med. Chem. , vol.43 , pp. 2211-2219
- Gao, M.¹ Wang, M.² Miller, K.D.³ Sledge, G.W.⁴ Zheng, Q.H.⁵

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