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Bioorganic and Medicinal Chemistry Letters

Volumn 20, Issue 17, 2010, Pages 5245-5250

Triaryl (Z)-olefins suitable for radiolabeling with carbon-11 or fluorine-18 radionuclides for positron emission tomography imaging of cyclooxygenase-2 expression in pathological disease

(5) Abdellatif, Khaled R A a Velázquez, Carlos A a Huang, Zhangjian a Chowdhury, Morshed A a Knaus, Edward E a

a UNIVERSITY OF ALBERTA (Canada)

Author keywords

Cyclooxygenase 2; Positron emission tomography imaging; Tricyclic (Z) olefins

Indexed keywords

1 (4 HYDROXYPHENYL) 1 PHENYL 2 (4 METHYLSULFONYLPHENYL)BUT 1 ENE; 1 (4 HYDROXYPHENYL) 1 PHENYL 2 (4 METHYLSULFONYLPHENYL)HEX 1 ENE; 1 (4 METHOXYPHENYL) 1 PHENYL 2 (4 METHYLSULFONYLPHENYL)BUT 1 ENE; 1 (4 METHOXYPHENYL) 1 PHENYL 2 (4 METHYLSULFONYLPHENYL)HEX 1 ENE; 1 [4 (2 FLUOROETHOXY)PHENYL] 1 PHENYL 2 (4 METHYLSULFONYLPHENYL)HEX 1 ENE; 1,1 DIPHENYL 2 (4 METHYLSULFONYLPHENYL)ALK 1 ENE DERIVATIVE; 4 FLUORO 1,1 DIPHENYL 2 (4 METHYLSULPHONYLPHENYL)BUT 1 ENE; ALKENE DERIVATIVE; CARBON 11; CELECOXIB; CYCLOOXYGENASE 1 INHIBITOR; CYCLOOXYGENASE 2; CYCLOOXYGENASE 2 INHIBITOR; FLUORINE 18; RADIOISOTOPE; ROFECOXIB; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL BOND; ISOTOPE LABELING; POSITRON EMISSION TOMOGRAPHY; PROTEIN EXPRESSION; STRUCTURE ACTIVITY RELATION; UPREGULATION;

ALKENES; CARBON RADIOISOTOPES; CYCLOOXYGENASE 2; DISEASE; FLUORINE RADIOISOTOPES; HUMANS; POSITRON-EMISSION TOMOGRAPHY;

EID: 77955714043 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2010.06.155 Document Type: Article

Times cited : (5)

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