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Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 18, 2011, Pages 5353-5357

Identification of SQ609 as a lead compound from a library of dipiperidines

(10) Bogatcheva, Elena a Hanrahan, Colleen b Nikonenko, Boris a De Los Santos, Gladys e Reddy, Venkata a Chen, Ping c Barbosa, Francis d Einck, Leo a Nacy, Carol a Protopopova, Marina a

a SEQUELLA INC (United States)

b JOHNS HOPKINS UNIVERSITY SCHOOL OF MEDICINE (United States)

c NATIONAL INSTITUTE OF ALLERGY AND INFECTIOUS DISEASES (United States)

d Sibley Hospital (United States)

e CENTRO DE INVESTIGACIÓN EN QUÍMICA APLICADA (Mexico)

Author keywords

(Piperidin 4 ylmethyl)piperidine; Combinatorial library; Dipiperidine scaffold; Tuberculosis

Indexed keywords

(PIPERIDIN 4 YLMETHYL)PIPERIDINE; DIPIPERIDINE DERIVATIVE; PIPERIDINE DERIVATIVE; SQ 609; SQ 614; SQ 615; TUBERCULOSTATIC AGENT; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL EXPERIMENT; ANTIBACTERIAL ACTIVITY; ARTICLE; BACTERIAL GROWTH; CONTROLLED STUDY; DRUG SYNTHESIS; IN VITRO STUDY; IN VIVO STUDY; MACROPHAGE; MINIMUM INHIBITORY CONCENTRATION; MOUSE; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN; STRUCTURE ACTIVITY RELATION; WEIGHT REDUCTION;

ADAMANTANE; ANIMALS; ANTITUBERCULAR AGENTS; DISEASE MODELS, ANIMAL; DOSE-RESPONSE RELATIONSHIP, DRUG; MACROPHAGES; MICE; MICE, INBRED C3H; MICROBIAL SENSITIVITY TESTS; MYCOBACTERIUM TUBERCULOSIS; PIPERIDINES; SMALL MOLECULE LIBRARIES; STRUCTURE-ACTIVITY RELATIONSHIP; WEIGHT LOSS;

BACTERIA (MICROORGANISMS); MUS; MYCOBACTERIUM TUBERCULOSIS;

EID: 80051919730 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2011.07.015 Document Type: Article

Times cited : (66)

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