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Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 54, Issue 9, 2011, Pages 633-636

A first synthesis of 18F-radiolabeled lapatinib: A potential tracer for positron emission tomographic imaging of ErbB1/ErbB2 tyrosine kinase activity

(6) Basuli, Falguni a Wu, Haitao a Li, Changhui a Shi, Zhen Dan a Sulima, Agnieszka a Griffiths, Gary L a

a NATIONAL HEART LUNG AND BLOOD INSTITUTE (United States)

Author keywords

Fluorine 18; Radiolabeling

Indexed keywords

AMINO ACIDS; FLUORINE; POTASH;

BOC GROUP; DEPROTECTION; FLUORINE-18; KINASE ACTIVITY; LAPATINIB; POSITRON EMISSION; RADIOLABELLING; SYNTHESISED; TOMOGRAPHIC IMAGING; TYROSINE KINASE;

DIMETHYLFORMAMIDE;

BROMIDE; EPIDERMAL GROWTH FACTOR RECEPTOR; EPIDERMAL GROWTH FACTOR RECEPTOR 2; LAPATINIB; LAPATINIB F 18; N,N DIMETHYLFORMAMIDE; POTASSIUM CARBONATE; TRACER; TRIFLUOROACETIC ACID; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL REACTION; DEPROTECTION REACTION; DRUG SYNTHESIS; ENZYME ACTIVITY; FLUORINATION; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; ISOTOPE LABELING; POSITRON EMISSION TOMOGRAPHY; RADIOCHEMISTRY; TEMPERATURE;

EID: 80051868110 PISSN: 03624803 EISSN: 10991344 Source Type: Journal
DOI: 10.1002/jlcr.1898 Document Type: Article

Times cited : (21)

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