Benzodiazepinone derivatives as CRTH2 antagonists

ACS Medicinal Chemistry Letters

Volumn 2, Issue 7, 2011, Pages 515-518

  Liu, Jiwen ^a   Cheng, Alan C ^a   Tang, H Lucy ^a   Medina, Julio C ^a  

^a AMGEN INC   (United States)

Author keywords

antagonist; asthma; benzodiazepinones; CRTH2; PGD 2; pharmacophore

Indexed keywords

BENZODIAZEPINE DERIVATIVE;

ARTICLE; CHRONIC OBSTRUCTIVE LUNG DISEASE; HYDROGEN BOND; PHARMACOPHORE; PRIORITY JOURNAL; TH2 CELL;

EID: 79960400846     PISSN: None     EISSN: 19485875     Source Type: Journal    
DOI: 10.1021/ml200019y     Document Type: Article

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