-
1
-
-
0033756052
-
In vivo inhibition of PC-3 human androgen-independent prostate cancer by a targeted cytotoxic bombesin analogue, AN-215
-
Plonowski A, Nagy A, Schally AV, et al. In vivo inhibition of PC-3 human androgen-independent prostate cancer by a targeted cytotoxic bombesin analogue, AN-215. Int J Cancer 2000;88:652.
-
(2000)
Int J Cancer
, vol.88
, pp. 652
-
-
Plonowski, A.1
Nagy, A.2
Schally, A.V.3
-
2
-
-
0032587895
-
99mTc labeling and in vivo studies of a bombesin analogue with a novel water-soluble dithiadiphosphine-based bifunctional chelating agent
-
Karra SR, Schibli R, Gali H, et al. 99mTc labeling and in vivo studies of a bombesin analogue with a novel water-soluble dithiadiphosphine-based bifunctional chelating agent. Bioconj Chem 1999;10:254.
-
(1999)
Bioconj Chem
, vol.10
, pp. 254
-
-
Karra, S.R.1
Schibli, R.2
Gali, H.3
-
3
-
-
0035114167
-
Dierckx, is there a role for agonist gastrin-releasing peptide receptor radioligands in tumour imaging
-
Van deWiele C, Dumont F, van Belle S, et al Dierckx, is there a role for agonist gastrin-releasing peptide receptor radioligands in tumour imaging. Nucl Med Commun 2001; 22: 5.
-
(2001)
Nucl Med Commun
, vol.22
, pp. 5
-
-
Van Dewiele, C.1
Dumont, F.2
Van Belle, S.3
-
4
-
-
0021807624
-
Bombesin-like peptides as autocrine growth factors in human small-cell lung cancer
-
Cuttitta F, Carney DN, Mulshine J, et al. Bombesin-like peptides as autocrine growth factors in human small-cell lung cancer. Nature 1985;316:823.
-
(1985)
Nature
, vol.316
, pp. 823
-
-
Cuttitta, F.1
Carney, D.N.2
Mulshine, J.3
-
5
-
-
0025922873
-
Bombesin analogues inhibit growth of small cell lung cancer in vitro and in vivo
-
Mahmoud S, Staley J, Taylor J, et al. Bombesin analogues inhibit growth of small cell lung cancer in vitro and in vivo. Cancer Res 1991;51:1798.
-
(1991)
Cancer Res
, vol.51
, pp. 1798
-
-
Mahmoud, S.1
Staley, J.2
Taylor, J.3
-
6
-
-
0029034647
-
Highaffinity binding sites for gastrin-releasing peptide on human colorectal cancer tissue but not uninvolved mucosa
-
Preston SR, Woodhouse LF, Jones-Blackett GV, et al. Highaffinity binding sites for gastrin-releasing peptide on human colorectal cancer tissue but not uninvolved mucosa. Br J Cancer 1995;71:1097.
-
(1995)
Br J Cancer
, vol.71
, pp. 1097
-
-
Preston, S.R.1
Woodhouse, L.F.2
Jones-Blackett, G.V.3
-
7
-
-
4644360336
-
Synthesis and evaluation of bombesin derivatives on the basis of pan-bombesin peptides labeled with indium-111, lutetium-177, and yttrium- 90 for targeting bombesin receptor-expressing tumors
-
Zhang H, Chen J, Waldherr C, et al. Synthesis and evaluation of bombesin derivatives on the basis of pan-bombesin peptides labeled with indium-111, lutetium-177, and yttrium- 90 for targeting bombesin receptor-expressing tumors. Cancer Res 2004;64:6707.
-
(2004)
Cancer Res
, vol.64
, pp. 6707
-
-
Zhang, H.1
Chen, J.2
Waldherr, C.3
-
8
-
-
0037291708
-
Radiochemical investigations of 177Lu-DOTA-8-Aoc-BBN[7-14]NH2: An in vitro/ in vivo assessment of the targeting ability of this new radiopharmaceutical for PC-3 human prostate cancer cells
-
Smith CJ, Gali H, Sieckman GL, et al. Radiochemical investigations of 177Lu-DOTA-8-Aoc-BBN[7-14]NH2: An in vitro/ in vivo assessment of the targeting ability of this new radiopharmaceutical for PC-3 human prostate cancer cells. Nucl Med Biol 2003;30:101.
-
(2003)
Nucl Med Biol
, vol.30
, pp. 101
-
-
Smith, C.J.1
Gali, H.2
Sieckman, G.L.3
-
9
-
-
0032958842
-
Evaluation of radiolabelled bombesin analogues for receptor-targeted scintigraphy and radiotherapy
-
Breeman WA, Hofland LJ, de Jong M, et al. Evaluation of radiolabelled bombesin analogues for receptor-targeted scintigraphy and radiotherapy. Int J Cancer 1999;81:658.
-
(1999)
Int J Cancer
, vol.81
, pp. 658
-
-
Breeman, W.A.1
Hofland, L.J.2
De Jong, M.3
-
10
-
-
0033754433
-
Technetium-99m RP527, a GRP analogue for visualisation of GRP receptor-expressing malignancies: A feasibility study
-
Van de Wiele C, Dumont F, Vanden Broecke R, et al. Technetium-99m RP527, a GRP analogue for visualisation of GRP receptor-expressing malignancies: A feasibility study. Eur J Nucl Med 2000;27:1694.
-
(2000)
Eur J Nucl Med
, vol.27
, pp. 1694
-
-
Van De Wiele, C.1
Dumont, F.2
Vanden Broecke, R.3
-
11
-
-
0347991822
-
Gastrin releasing peptide (GRP) receptor targeted radiopharmaceuticals: A concise update
-
Smith CJ, Volkert WA, Hoffman TJ. Gastrin releasing peptide (GRP) receptor targeted radiopharmaceuticals: A concise update. Nucl Med Biol 2003;30:861.
-
(2003)
Nucl Med Biol
, vol.30
, pp. 861
-
-
Smith, C.J.1
Volkert, W.A.2
Hoffman, T.J.3
-
12
-
-
0037945450
-
Novel series of 111In-labeled bombesin analogs as potential radiopharmaceuticals for specific targeting of gastrinreleasing peptide receptors expressed on human prostate cancer cells
-
Hoffman TJ, Gali H,SmithCJ, et al.Novel series of 111In-labeled bombesin analogs as potential radiopharmaceuticals for specific targeting of gastrinreleasing peptide receptors expressed on human prostate cancer cells. J Nucl Med 2003;44:823.
-
(2003)
J Nucl Med
, vol.44
, pp. 823
-
-
Hoffman, T.J.1
Gali, H.2
Smith, C.J.3
-
13
-
-
4544291850
-
MicroPET and autoradiographic imaging of GRP receptor expression with 64Cu- DOTA-[Lys3] bombesin in human prostate adenocarcinoma xenografts
-
Chen X, Park R, Hou Y, et al. microPET and autoradiographic imaging of GRP receptor expression with 64Cu- DOTA-[Lys3] bombesin in human prostate adenocarcinoma xenografts. J Nucl Med 2004;45:1390.
-
(2004)
J Nucl Med
, vol.45
, pp. 1390
-
-
Chen, X.1
Park, R.2
Hou, Y.3
-
14
-
-
12144279487
-
Potent bombesinlike peptides for GRP-receptor targeting of tumors with 99mTc: A preclinical study
-
Nock BA, Nikolopoulou A, Galanis A, et al. Potent bombesinlike peptides for GRP-receptor targeting of tumors with 99mTc: A preclinical study. J Med Chem 2005;48:100.
-
(2005)
J Med Chem
, vol.48
, pp. 100
-
-
Nock, B.A.1
Nikolopoulou, A.2
Galanis, A.3
-
15
-
-
0032032589
-
Design syn thesis, and initial evaluation of high-affinity technetium bombesin analogues
-
Baidoo KE, Lin KS, Zhan Y, et al. Design, synthesis, and initial evaluation of high-affinity technetium bombesin analogues. Bioconjug Chem 1998;9:218.
-
(1998)
Bioconjug Chem
, vol.9
, pp. 218
-
-
Baidoo, K.E.1
Lin, K.S.2
Zhan, Y.3
-
17
-
-
0035999172
-
In vitro and in vivo evaluation of a 99mTc (I)-labeled bombesin analogue for imaging of gastrin releasing peptide receptor-positive tumors
-
La Bella R, Garcia-Garayoa E, Langer M, et al. In vitro and in vivo evaluation of a 99mTc (I)-labeled bombesin analogue for imaging of gastrin releasing peptide receptor-positive tumors. Nucl Med Biol 2002;29:553.
-
(2002)
Nucl Med Biol
, vol.29
, pp. 553
-
-
La Bella, R.1
Garcia-Garayoa, E.2
Langer, M.3
-
18
-
-
0043267475
-
Radiochemical investigations of gastrin-releasing peptide receptor-specific [99mTc (X)(CO)3-Dpr-Ser-Ser-Ser-Gln-Trp-Ala-Val-Gly-His- Leu-Met-(NH2)] in PC-3, tumor-bearing, rodent models: Syntheses, radiolabeling, and in vitro/in vivo studies where Dpr2,3-diaminopropionic acid and XH2Oor P (CH2OH)3
-
Smith CJ, Sieckman GL, Owen NK, et al. Radiochemical investigations of gastrin-releasing peptide receptor-specific [99mTc (X)(CO)3-Dpr-Ser-Ser-Ser-Gln- Trp-Ala-Val-Gly-His- Leu-Met-(NH2)] in PC-3, tumor-bearing, rodent models: Syntheses, radiolabeling, and in vitro/in vivo studies where Dpr2,3-diaminopropionic acid and XH2Oor P (CH2OH)3. Cancer Res 2003;63:4082.
-
(2003)
Cancer Res
, vol.63
, pp. 4082
-
-
Smith, C.J.1
Sieckman, G.L.2
Owen, N.K.3
-
19
-
-
34548119383
-
Formulation and in vitro metabolism studies with 177Lu-AMBA; A radiotherapeutic compound that targets gastrin releasing peptide receptors
-
Chen J, Nguyen H, Metcalfe E, et al. Formulation and in vitro metabolism studies with 177Lu-AMBA; a radiotherapeutic compound that targets gastrin releasing peptide receptors. Eur J Nucl Med Mol Imaging 2004;31 Suppl 2:S281.
-
(2004)
Eur J Nucl Med Mol Imaging
, vol.2
, Issue.31 SUPPL.
-
-
Chen, J.1
Nguyen, H.2
Metcalfe, E.3
-
20
-
-
0038579396
-
[99mTc] Demobesin 1, a novel potent bombesin analogue for GRP receptortargeted tumour imaging
-
Nock B, Nikolopoulou A, Chiotellis E, et al. [99mTc] Demobesin 1, a novel potent bombesin analogue for GRP receptortargeted tumour imaging. Eur J Nucl Med Mol Imaging 2003;30:247.
-
(2003)
Eur J Nucl Med Mol Imaging
, vol.30
, pp. 247
-
-
Nock, B.1
Nikolopoulou, A.2
Chiotellis, E.3
-
21
-
-
0035205681
-
Biodistribution and dosimetry of 99mTc-RP527, a gastrin-releasing peptide (GRP) agonist for the visualization of GRP receptorexpressing malignancies
-
Van de Wiele C, Dumont F, Dierckx RA, et al. Biodistribution and dosimetry of 99mTc-RP527, a gastrin-releasing peptide (GRP) agonist for the visualization of GRP receptorexpressing malignancies. J Nucl Med 2001;42:1722.
-
(2001)
J Nucl Med
, vol.42
, pp. 1722
-
-
Van De Wiele, C.1
Dumont, F.2
Dierckx, R.A.3
-
22
-
-
19644372238
-
GRP receptor-targeted PET of a rat pancreas carcinoma xenograft in nude mice with a 68Ga-labeled bombesin(6-14) analog
-
Schuhmacher J, Zhang H, Doll J, et al. GRP receptor-targeted PET of a rat pancreas carcinoma xenograft in nude mice with a 68Ga-labeled bombesin(6-14) analog. J Nucl Med 2005;46:691.
-
(2005)
J Nucl Med
, vol.46
, pp. 691
-
-
Schuhmacher, J.1
Zhang, H.2
Doll, J.3
-
23
-
-
0038455833
-
MicroPET imaging of a gastrin-releasing peptide receptor-positive tumor in a mouse model of human prostate cancer using a 64Culabeled bombesin analogue
-
Rogers BE, Bigott HN, McCarthy DW, et al. MicroPET imaging of a gastrin-releasing peptide receptor-positive tumor in a mouse model of human prostate cancer using a 64Culabeled bombesin analogue. Bioconjug Chem 2003;14:756.
-
(2003)
Bioconjug Chem
, vol.14
, pp. 756
-
-
Rogers, B.E.1
Bigott, H.N.2
McCarthy, D.W.3
-
25
-
-
0032706253
-
Pre-clinical evaluation of [111In-DTPA-Pro1, Tyr4]bombesin, a new radioligand for bombesin-receptor scintigraphy
-
Breeman WA, De Jong M, Bernard BF, et al. Pre-clinical evaluation of [111In-DTPA-Pro1, Tyr4]bombesin, a new radioligand for bombesin-receptor scintigraphy. Int J Cancer 1999;83:657.
-
(1999)
Int J Cancer
, vol.83
, pp. 657
-
-
Breeman, W.A.1
De Jong, M.2
Bernard, B.F.3
-
26
-
-
0036898728
-
Preclinical comparison of 111In -labeled DTPA or DOTA-bombesin analogs for receptor-targeted scintigraphy and radionuclide therapy
-
Breeman WA, de Jong M, Erion JL, et al. Preclinical comparison of 111In -labeled DTPA or DOTA-bombesin analogs for receptor-targeted scintigraphy and radionuclide therapy. J Nucl Med 2002;43:1650.
-
(2002)
J Nucl Med
, vol.43
, pp. 1650
-
-
Breeman, W.A.1
De Jong, M.2
Erion, J.L.3
-
27
-
-
77949268332
-
Preparation and evaluation of a new 99mTc labeled bombesin derivative for tumor imaging
-
Sadeghzadeh N, Gandomkar M, Najafi R, et al. Preparation and evaluation of a new 99mTc labeled bombesin derivative for tumor imaging. J Radioanal Nucl Chem 2010;283:181.
-
(2010)
J Radioanal Nucl Chem
, vol.283
, pp. 181
-
-
Sadeghzadeh, N.1
Gandomkar, M.2
Najafi, R.3
-
28
-
-
73949139190
-
Synthesis and evaluation of a new radiolabeled bombesin analogue for diagnosis of GRP receptor expressing tumors
-
Sadeghzadeh N, Gandomkar M, Shafiee M, et al. Synthesis and evaluation of a new radiolabeled bombesin analogue for diagnosis of GRP receptor expressing tumors. Iran J Nucl Med 2009;17:18.
-
(2009)
Iran J Nucl Med
, vol.17
, pp. 18
-
-
Sadeghzadeh, N.1
Gandomkar, M.2
Shafiee, M.3
-
29
-
-
34547839755
-
Preclinical evaluation of [99mTc/EDDA/tricine/HYNIC0, 1-Nal3, Thr8]- octreotide as a new analogue in the detection of somatostatinreceptor- positive tumors
-
Gandomkar M, Najafi R, Shafiei M, et al. Preclinical evaluation of [99mTc/EDDA/tricine/HYNIC0, 1-Nal3, Thr8]- octreotide as a new analogue in the detection of somatostatinreceptor- positive tumors. Nucl Med Biol 2007;34:651.
-
(2007)
Nucl Med Biol
, vol.34
, pp. 651
-
-
Gandomkar, M.1
Najafi, R.2
Shafiei, M.3
-
30
-
-
59649130283
-
Clinical evaluation of antimicrobial peptide [99mTc/Tricine/HYNIC0] ubiquicidin 29-41 as a human-specific infection imaging agent
-
Gandomkar M, Najafi R, Shafiei M, et al. Clinical evaluation of antimicrobial peptide [99mTc/Tricine/HYNIC0] ubiquicidin 29-41 as a human-specific infection imaging agent. Nucl Med Biol 2009;36:199.
-
(2009)
Nucl Med Biol
, vol.36
, pp. 199
-
-
Gandomkar, M.1
Najafi, R.2
Shafiei, M.3
-
31
-
-
0000317874
-
Ochrymowcycz, synthesis and characterization of 105Rh labeled bombesin analogues: Enhancement of GRP receptor binding affinity utilizing aliphatic carbon chain linkers
-
Hoffman TJ, Li N, Volkert WA, et al. Ochrymowcycz, synthesis and characterization of 105Rh labeled bombesin analogues: Enhancement of GRP receptor binding affinity utilizing aliphatic carbon chain linkers. J Label Compd Radiopharm 1997;40:490.
-
(1997)
J Label Compd Radiopharm
, vol.40
, pp. 490
-
-
Hoffman, T.J.1
Li, N.2
Volkert, W.A.3
-
32
-
-
0000210044
-
Accumulation and retention of Tc-99m RP527 by GRP receptor expressing tumors in scid mice [abstract]
-
Hoffman TJ, Simpson SD, Smith CJ. Accumulation and retention of Tc-99m RP527 by GRP receptor expressing tumors in scid mice [abstract]. J Nucl Med 1999;40(suppl):104P.
-
(1999)
J Nucl Med
, vol.40
, Issue.SUPPL.
, pp. 104
-
-
Hoffman, T.J.1
Simpson, S.D.2
Smith, C.J.3
-
33
-
-
4243678171
-
Optimizing pharmacokinetics of 99mTc-GRP receptor targeting peptides using multi-amino acid linking groups [abstract]
-
Hoffman TJ, Smith CJ, and Simpson SD. Optimizing pharmacokinetics of 99mTc-GRP receptor targeting peptides using multi-amino acid linking groups [abstract]. J Nucl Med 2000;41(suppl):228P.
-
(2000)
J Nucl Med
, vol.41
, Issue.SUPPL.
-
-
Hoffman, T.J.1
Smith, C.J.2
Simpson, S.D.3
-
34
-
-
34548119893
-
DOTA-PESIN, a DOTA-conjugated bombesin derivative designed for the imaging and targeted radionuclide treatment of bombesin receptor-positive tumors
-
Zhang H, Schuhmacher J, Waser B, et al. DOTA-PESIN, a DOTA-conjugated bombesin derivative designed for the imaging and targeted radionuclide treatment of bombesin receptor-positive tumors. Eur J Nucl Med Mol Imaging 2007;34:1198.
-
(2007)
Eur J Nucl Med Mol Imaging
, vol.34
, pp. 1198
-
-
Zhang, H.1
Schuhmacher, J.2
Waser, B.3
-
35
-
-
34547835136
-
Novel 111In-labelled bombesin analogues for molecular imaging of prostate tumors
-
de Visser M, Bernard HF, Erion JL, et al. Novel 111In-labelled bombesin analogues for molecular imaging of prostate tumors. Eur J Nucl Med Mol Imaging 2007;34:1228.
-
(2007)
Eur J Nucl Med Mol Imaging
, vol.34
, pp. 1228
-
-
De Visser, M.1
Bernard, H.F.2
Erion, J.L.3
-
36
-
-
52249089417
-
Evaluation of the pharmacokinetic effects of various linking groups using the 111In-DOTA-X-BBN(7-14)NH2 structural paradigm in a prostate cancer model
-
Garrison JC, Tammy LR, Sieckman GL, et al. Evaluation of the pharmacokinetic effects of various linking groups using the 111In-DOTA-X-BBN(7- 14)NH2 structural paradigm in a prostate cancer model. Bioconjug Chem 2008;19:1803.
-
(2008)
Bioconjug Chem
, vol.19
, pp. 1803
-
-
Garrison, J.C.1
Tammy, L.R.2
Sieckman, G.L.3
-
37
-
-
39749174303
-
Peptide motifs for insertion of radiolabeled biomolcules into cells and routing to the neucleus for cancer imaging or radiotherapeutic applications
-
Costantini DL, Hu M, Reilly R. Peptide motifs for insertion of radiolabeled biomolcules into cells and routing to the neucleus for cancer imaging or radiotherapeutic applications. Cancer Biother Radiopharm 2008;23:3.
-
(2008)
Cancer Biother Radiopharm
, vol.23
, pp. 3
-
-
Costantini, D.L.1
Hu, M.2
Reilly, R.3
-
38
-
-
0033033382
-
Radiometallabeled macrocyclic chelator derivatised somatostatin analogue with superb tumor targeting properties and potential for receptor mediated internal radiotherapy
-
Heppeler A, Froidevaux S, Macke HR, et al. Radiometallabeled macrocyclic chelator derivatised somatostatin analogue with superb tumor targeting properties and potential for receptor mediated internal radiotherapy. Chem Eur J 1999;5:1974.
-
(1999)
Chem Eur J
, vol.5
, pp. 1974
-
-
Heppeler, A.1
Froidevaux, S.2
MacKe, H.R.3
-
39
-
-
33747105269
-
177Lu- AMBA: Synthesis and characterization of a selective 177Lulabeled GRP-R agonist for systemic radiotherapy of prostate cancer
-
Lantry LE, Cappelletti E, Maddalena ME, et al. 177Lu- AMBA: Synthesis and characterization of a selective 177Lulabeled GRP-R agonist for systemic radiotherapy of prostate cancer. J Nucl Med 2006;47:1144.
-
(2006)
J Nucl Med
, vol.47
, pp. 1144
-
-
Lantry, L.E.1
Cappelletti, E.2
Maddalena, M.E.3
-
40
-
-
33744812175
-
Evaluation of combined Lu-177-DOTA-8-AOC-BBN (7-14) NH2 GRP receptortargeted radiotherapy and chemotherapy in PC-3 human prostate tumor cell xenografted SCID mice
-
Johnson CV, Shelton T, Smith CJ, et al. Evaluation of combined Lu-177-DOTA-8-AOC-BBN (7-14) NH2 GRP receptortargeted radiotherapy and chemotherapy in PC-3 human prostate tumor cell xenografted SCID mice. Cancer Biother Radiopharm 2006;21:155.
-
(2006)
Cancer Biother Radiopharm
, vol.21
, pp. 155
-
-
Johnson, C.V.1
Shelton, T.2
Smith, C.J.3
-
41
-
-
34250349188
-
Are radiogalliumlabelled DOTA-conjugated somatostatin analogues superior to those labelled with other radiometals?
-
Antunes P, Ginj M, Zhang H, et al. Are radiogalliumlabelled DOTA-conjugated somatostatin analogues superior to those labelled with other radiometals? Eur J Nucl Med Mol Imaging 2007;34:982.
-
(2007)
Eur J Nucl Med Mol Imaging
, vol.34
, pp. 982
-
-
Antunes, P.1
Ginj, M.2
Zhang, H.3
|