메뉴 건너뛰기




Volumn 83, Issue 5, 1999, Pages 657-663

Pre-clinical evaluation of [111In-DTPA-Pro1, Tyr4]bombesin, a new radioligand for bombesin-receptor scintigraphy

Author keywords

[No Author keywords available]

Indexed keywords

BOMBESIN; BOMBESIN RECEPTOR; INDIUM; PENTETATE INDIUM IN 111; PROLACTIN; PROLINE; RADIOLIGAND; TYROSINE;

EID: 0032706253     PISSN: 00207136     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1097-0215(19991126)83:5<657::AID-IJC15>3.0.CO;2-Y     Document Type: Article
Times cited : (91)

References (29)
  • 1
    • 0030787791 scopus 로고    scopus 로고
    • Bombesin stimulates the motility of human prostate-carcinoma cells through tyrosine phosphorylation of focal adhesion kinase and of integrin-associated proteins
    • APRIKIAN, A.G., TREMBLAY, L., HAN, K. and CHEVALIER, S., Bombesin stimulates the motility of human prostate-carcinoma cells through tyrosine phosphorylation of focal adhesion kinase and of integrin-associated proteins. Int. J. Cancer, 72, 498-504 (1997).
    • (1997) Int. J. Cancer , vol.72 , pp. 498-504
    • Aprikian, A.G.1    Tremblay, L.2    Han, K.3    Chevalier, S.4
  • 2
    • 0025925126 scopus 로고
    • 1]octreotide, a potential radiopharmaceutical for imaging of somatostatin-receptor-positive tumors: Synthesis, radiolabeling and in vitro validation
    • 1]octreotide, a potential radiopharmaceutical for imaging of somatostatin-receptor-positive tumors: synthesis, radiolabeling and in vitro validation. Life Sci., 49, 1583-1591 (1991a).
    • (1991) Life Sci. , vol.49 , pp. 1583-1591
    • Bakker, W.H.1
  • 4
    • 0022383308 scopus 로고
    • Gastrin-releasing peptide in human neuro-endocrine tumors
    • BOSTWICK, D.G. and BENSCH, K.G., Gastrin-releasing peptide in human neuro-endocrine tumors. J. Pathol., 147, 237-244 (1985).
    • (1985) J. Pathol. , vol.147 , pp. 237-244
    • Bostwick, D.G.1    Bensch, K.G.2
  • 11
    • 0025096119 scopus 로고
    • Short-chain pseudopeptides with potent bombesin-receptor-antagonist activity in rat and guinea pig pancreatic acinair cells
    • COY, D.H., WANG, L.H., JIANG, N.Y. and JENSEN, R.T., Short-chain pseudopeptides with potent bombesin-receptor-antagonist activity in rat and guinea pig pancreatic acinair cells. Europ. J. Pharmacol., 190, 31-38 (1990).
    • (1990) Europ. J. Pharmacol. , vol.190 , pp. 31-38
    • Coy, D.H.1    Wang, L.H.2    Jiang, N.Y.3    Jensen, R.T.4
  • 13
    • 0026637732 scopus 로고
    • Metabolic stability and tumor inhibition of bombesin/GRP-receptor antagonist
    • DAVIS, T.P., CROWELL, S., TAYLOR, J., CLARK, D.L., COY, D., STALEY, J. and MOODY, T.W., Metabolic stability and tumor inhibition of bombesin/GRP-receptor antagonist. Peptides, 13, 401-407 (1992).
    • (1992) Peptides , vol.13 , pp. 401-407
    • Davis, T.P.1    Crowell, S.2    Taylor, J.3    Clark, D.L.4    Coy, D.5    Staley, J.6    Moody, T.W.7
  • 14
    • 0031987328 scopus 로고    scopus 로고
    • 111In-labeled somatostatin analogues for tumor scintigraphy and radionuclide therapy
    • 111In-labeled somatostatin analogues for tumor scintigraphy and radionuclide therapy. Cancer Res., 58, 437-441 (1998).
    • (1998) Cancer Res. , vol.58 , pp. 437-441
    • De Jong1
  • 16
    • 0031050737 scopus 로고    scopus 로고
    • Indium-111-diethyletriaminepentaacetic acid-octreotide is delivered in vivo to pancreatic, tumor-cell, renal and hepatocyte lysosomes
    • DUNCAN, J.R., STEPHENSON, M.T., WU, H.P. and ANDERSON, C.J., Indium-111-diethyletriaminepentaacetic acid-octreotide is delivered in vivo to pancreatic, tumor-cell, renal and hepatocyte lysosomes. Cancer Res., 57, 659-671 (1997).
    • (1997) Cancer Res. , vol.57 , pp. 659-671
    • Duncan, J.R.1    Stephenson, M.T.2    Wu, H.P.3    Anderson, C.J.4
  • 17
    • 0030067575 scopus 로고    scopus 로고
    • Expression and characterization of gastrin-releasing peptide receptor in normal and cancerous pancreas
    • HAJRI, A., KOENIG, M., BALBONI, G. and DAMGE, C., Expression and characterization of gastrin-releasing peptide receptor in normal and cancerous pancreas. Pancreas, 12, 25-35 (1996).
    • (1996) Pancreas , vol.12 , pp. 25-35
    • Hajri, A.1    Koenig, M.2    Balboni, G.3    Damge, C.4
  • 18
    • 0025233324 scopus 로고
    • Effect of loxiglumide (CR1505) on bombesin-and meal-stimulated plasma-cholecystokinin release in man
    • JANSEN, J.B.M.J., JEBBINK, M.C.W., DOUGLAS, B.R. and LAMERS, C.B.H.W., Effect of loxiglumide (CR1505) on bombesin-and meal-stimulated plasma-cholecystokinin release in man. Europ. J. clin. Pharmacol., 28, 367-370 (1990).
    • (1990) Europ. J. Clin. Pharmacol. , vol.28 , pp. 367-370
    • Jansen, J.B.M.J.1    Jebbink, M.C.W.2    Douglas, B.R.3    Lamers, C.B.H.W.4
  • 19
    • 0026078928 scopus 로고
    • Progress in the development of potent bombesin-receptorantagonists
    • JENSEN, R.T. and COY, D.H., Progress in the development of potent bombesin-receptorantagonists. TIPS, 12, 13-19 (1991).
    • (1991) TIPS , vol.12 , pp. 13-19
    • Jensen, R.T.1    Coy, D.H.2
  • 21
    • 0027517429 scopus 로고
    • 3]-octreotide: The Rotterdam experience with more than 1000 patients
    • 3]-octreotide: the Rotterdam experience with more than 1000 patients. Europ. J. nucl. Med., 20, 716-731 (1993).
    • (1993) Europ. J. Nucl. Med. , vol.20 , pp. 716-731
    • Krenning, E.P.1
  • 22
    • 0027496213 scopus 로고
    • High-affinity binding sites for gastrin-releasing peptide on human gastric cancer and ménétrier's mucosa
    • PRESTON, S.R., WOODHOUSE, L.F., JONES-BLACKETT, S., WYATT, J.L. and PRIMROSE, J.N., High-affinity binding sites for gastrin-releasing peptide on human gastric cancer and Ménétrier's mucosa. Cancer Res., 53, 5090-5092 (1993).
    • (1993) Cancer Res. , vol.53 , pp. 5090-5092
    • Preston, S.R.1    Woodhouse, L.F.2    Jones-Blackett, S.3    Wyatt, J.L.4    Primrose, J.N.5
  • 23
    • 0027965768 scopus 로고
    • Bombesin antagonist inhibits in vitro and in vivo growth of human gastric cancer and binding of bombesin to its receptors
    • QIN, Y., HALMOS, G., CAI, R-Z., SZOKE, B., ERTL, T. and SCHALLY, A.V., Bombesin antagonist inhibits in vitro and in vivo growth of human gastric cancer and binding of bombesin to its receptors. J. Cancer. Res. clin. Oncol., 120, 519-528 (1994).
    • (1994) J. Cancer. Res. Clin. Oncol. , vol.120 , pp. 519-528
    • Qin, Y.1    Halmos, G.2    Cai, R.-Z.3    Szoke, B.4    Ertl, T.5    Schally, A.V.6
  • 28
    • 0025021426 scopus 로고
    • Desmethionine alkylamide bombesin analogue: A new class of bombesin-receptor antagonist with potent anti-secretory activity in pancreatic acini and anti-mitotic activity in Swiss 3T3 cells
    • WANG, L.H., COY, D.H., TAYLOR, J.E., JIANG, N.Y., KIM, S.H., MOREAU, J-P., HUANG, S.H., MANTEY, S.A., FRUCHT, H. and JENSEN, R.T., Desmethionine alkylamide bombesin analogue: a new class of bombesin-receptor antagonist with potent anti-secretory activity in pancreatic acini and anti-mitotic activity in Swiss 3T3 cells. Biochemistry, 29, 616-622 (1990).
    • (1990) Biochemistry , vol.29 , pp. 616-622
    • Wang, L.H.1    Coy, D.H.2    Taylor, J.E.3    Jiang, N.Y.4    Kim, S.H.5    Moreau, J.-P.6    Huang, S.H.7    Mantey, S.A.8    Frucht, H.9    Jensen, R.T.10
  • 29
    • 0027470822 scopus 로고
    • Ligand binding, internalization, degradation and regulation by guanine nucleotides of bombesin-receptor sub-types: A comparative study
    • WANG, L.H., MANTEY, J.T., FRUCHT, L.H. and JENSEN, R.T., Ligand binding, internalization, degradation and regulation by guanine nucleotides of bombesin-receptor sub-types: a comparative study. Biochem. biophys. Acta, 1175, 232-242 (1993).
    • (1993) Biochem. Biophys. Acta , vol.1175 , pp. 232-242
    • Wang, L.H.1    Mantey, J.T.2    Frucht, L.H.3    Jensen, R.T.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.